Compile Data Set for Download or QSAR
Report error Found 16 Enz. Inhib. hit(s) with all data for entry = 50014660
TargetUrokinase-type plasminogen activator(Human)
University of Antwerp

Curated by ChEMBL
LigandPNGBDBM50145689([1-[(S)-2-((R)-2-Benzyloxycarbonylamino-3-hydroxy-...)
Affinity DataIC50: 57nMAssay Description:Inhibitory activity against Urokinase-type plasminogen activatorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetUrokinase-type plasminogen activator(Human)
University of Antwerp

Curated by ChEMBL
LigandPNGBDBM50145688({1-[(S)-2-((R)-2-Benzyloxycarbonylamino-3-hydroxy-...)
Affinity DataIC50: 61nMAssay Description:Inhibitory activity against Urokinase-type plasminogen activatorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetUrokinase-type plasminogen activator(Human)
University of Antwerp

Curated by ChEMBL
LigandPNGBDBM50145690({1-[(S)-2-((R)-2-Benzyloxycarbonylamino-3-hydroxy-...)
Affinity DataIC50: 250nMAssay Description:Inhibitory activity against Urokinase-type plasminogen activatorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProthrombin(Human)
University of Antwerp

Curated by ChEMBL
LigandPNGBDBM50145688({1-[(S)-2-((R)-2-Benzyloxycarbonylamino-3-hydroxy-...)
Affinity DataIC50: 500nMAssay Description:Inhibitory activity against thrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetUrokinase-type plasminogen activator(Human)
University of Antwerp

Curated by ChEMBL
LigandPNGBDBM50145687([(S)-[(S)-2-((R)-2-Benzyloxycarbonylamino-3-hydrox...)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibitory activity against Urokinase-type plasminogen activatorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetUrokinase-type plasminogen activator(Human)
University of Antwerp

Curated by ChEMBL
LigandPNGBDBM50145693([[(S)-2-((R)-2-Benzyloxycarbonylamino-3-hydroxy-pr...)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibitory activity against Urokinase-type plasminogen activatorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetUrokinase-type plasminogen activator(Human)
University of Antwerp

Curated by ChEMBL
LigandPNGBDBM50145691({1-[(S)-2-((R)-2-Benzyloxycarbonylamino-3-hydroxy-...)
Affinity DataIC50: 4.10E+3nMAssay Description:Inhibitory activity against Urokinase-type plasminogen activatorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetUrokinase-type plasminogen activator(Human)
University of Antwerp

Curated by ChEMBL
LigandPNGBDBM50145692([[(S)-2-((R)-2-Benzyloxycarbonylamino-3-hydroxy-pr...)
Affinity DataIC50: 8.40E+3nMAssay Description:Inhibitory activity against Urokinase-type plasminogen activatorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlasminogen(Human)
University of Antwerp

Curated by ChEMBL
LigandPNGBDBM50145688({1-[(S)-2-((R)-2-Benzyloxycarbonylamino-3-hydroxy-...)
Affinity DataIC50: 1.08E+4nMAssay Description:Inhibitory activity against plasminMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTissue-type plasminogen activator(Human)
University of Antwerp

Curated by ChEMBL
LigandPNGBDBM50145689([1-[(S)-2-((R)-2-Benzyloxycarbonylamino-3-hydroxy-...)
Affinity DataIC50: 1.40E+4nMAssay Description:Inhibitory activity against Tissue type plasminogen activatorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlasminogen(Human)
University of Antwerp

Curated by ChEMBL
LigandPNGBDBM50145689([1-[(S)-2-((R)-2-Benzyloxycarbonylamino-3-hydroxy-...)
Affinity DataIC50: 2.20E+4nMAssay Description:Inhibitory activity against plasminMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProthrombin(Human)
University of Antwerp

Curated by ChEMBL
LigandPNGBDBM50145689([1-[(S)-2-((R)-2-Benzyloxycarbonylamino-3-hydroxy-...)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibitory activity against thrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlasminogen(Human)
University of Antwerp

Curated by ChEMBL
LigandPNGBDBM50145687([(S)-[(S)-2-((R)-2-Benzyloxycarbonylamino-3-hydrox...)
Affinity DataIC50: 3.22E+4nMAssay Description:Inhibitory activity against plasminMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
University of Antwerp

Curated by ChEMBL
LigandPNGBDBM50145688({1-[(S)-2-((R)-2-Benzyloxycarbonylamino-3-hydroxy-...)
Affinity DataIC50: 6.50E+4nMAssay Description:Inhibitory activity against Coagulation factor XaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
University of Antwerp

Curated by ChEMBL
LigandPNGBDBM50145689([1-[(S)-2-((R)-2-Benzyloxycarbonylamino-3-hydroxy-...)
Affinity DataIC50: 7.90E+4nMAssay Description:Inhibitory activity against Coagulation factor XaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetUrokinase-type plasminogen activator(Human)
University of Antwerp

Curated by ChEMBL
LigandPNGBDBM16173(3,5-diamino-N-carbamimidoyl-6-chloropyrazine-2-car...)
Affinity DataIC50: 1.07E+5nMAssay Description:Inhibitory activity against Urokinase-type plasminogen activatorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)