Compile Data Set for Download or QSAR
Report error Found 28 Enz. Inhib. hit(s) with all data for entry = 50000353
TargetAdenosine receptor A1(Rat)
Marion Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50004724(CHEMBL109310 | 5-Methyl-1-phenyl-6-propoxy-1,5-dih...)
Affinity DataIC50: 4.30E+3nMAssay Description:Inhibition of [3H]CHA binding to Adenosine A1 receptor in rat cerebral cortical membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Marion Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50004720(CHEMBL334046 | 6-Methoxy-5-methyl-1-phenyl-1,5-dih...)
Affinity DataIC50: 4.80E+3nMAssay Description:Inhibition of [3H]CHA binding to Adenosine A1 receptor in rat cerebral cortical membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Marion Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50004718(CHEMBL322512 | 5,7-Dimethyl-1-phenyl-1,7-dihydro-p...)
Affinity DataIC50: 3.30E+4nMAssay Description:Inhibition of [3H]CHA binding to Adenosine A1 receptor in rat cerebral cortical membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Marion Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50004723(CHEMBL322801 | 5-Methyl-1-phenyl-7-propyl-1,7-dihy...)
Affinity DataIC50: 3.50E+4nMAssay Description:Inhibition of [3H]CHA binding to Adenosine A1 receptor in rat cerebral cortical membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Marion Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50004711(CHEMBL420489 | 3-Phenyl-2-(9-phenyl-2-propoxy-9H-p...)
Affinity DataKi:  96nMAssay Description:Inhibition of [3H]CHA binding to Adenosine A1 receptor in rat cerebral cortical membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Rat)
Marion Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50455626(CHEMBL2112507)
Affinity DataKi:  310nMAssay Description:Inhibition of [3H]NECA binding to Adenosine A2 receptor in rat brain striatumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Marion Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50455625(CHEMBL2111718)
Affinity DataKi:  350nMAssay Description:Inhibition of [3H]CHA binding to Adenosine A1 receptor in whole rat brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Marion Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50455625(CHEMBL2111718)
Affinity DataKi:  350nMAssay Description:Inhibition of [3H]CHA binding to Adenosine A1 receptor in rat cerebral cortical membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Rat)
Marion Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50455625(CHEMBL2111718)
Affinity DataKi:  370nMAssay Description:Inhibition of [3H]NECA binding to Adenosine A2 receptor in rat brain striatumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Rat)
Marion Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50455625(CHEMBL2111718)
Affinity DataKi:  370nMAssay Description:Inhibition of [3H]NECA binding to Adenosine A2 receptor in rat brain striatumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Marion Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50004715(CHEMBL322270 | 3-Phenyl-2-(9-phenyl-2-propoxy-9H-p...)
Affinity DataKi:  440nMAssay Description:Inhibition of [3H]CHA binding to Adenosine A1 receptor in rat cerebral cortical membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Marion Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50004713(CHEMBL320319 | (R)-2-Benzyl-7-phenyl-5-propoxy-2,7...)
Affinity DataKi:  620nMAssay Description:Inhibition of [3H]CHA binding to Adenosine A1 receptor in rat cerebral cortical membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Marion Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50455626(CHEMBL2112507)
Affinity DataKi:  1.00E+3nMAssay Description:Inhibition of [3H]CHA binding to Adenosine A1 receptor in rat cerebral cortical membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Rat)
Marion Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50455624(CHEMBL2112500)
Affinity DataKi:  1.40E+3nMAssay Description:Inhibition of [3H]NECA binding to Adenosine A2 receptor in rat brain striatumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Rat)
Marion Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50004721(7-Benzyl-3-phenyl-5-propoxy-6,7-dihydro-3H-1,3,4,5...)
Affinity DataKi:  1.60E+3nMAssay Description:Inhibition of [3H]NECA binding to Adenosine A2 receptor in rat brain striatumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Marion Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50004722((R)-8-Benzyl-3-phenyl-5-propoxy-7,8-dihydro-3H-imi...)
Affinity DataKi:  3.20E+3nMAssay Description:Inhibition of [3H]CHA binding to Adenosine A1 receptor in rat cerebral cortical membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Rat)
Marion Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50004714((S)-2-Benzyl-7-phenyl-5-propoxy-2,7-dihydro-3H-imi...)
Affinity DataKi:  3.30E+3nMAssay Description:Inhibition of [3H]NECA binding to Adenosine A2 receptor in rat brain striatumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Rat)
Marion Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50004711(CHEMBL420489 | 3-Phenyl-2-(9-phenyl-2-propoxy-9H-p...)
Affinity DataKi:  5.60E+3nMAssay Description:Inhibition of [3H]NECA binding to Adenosine A2 receptor in rat brain striatumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Marion Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50455624(CHEMBL2112500)
Affinity DataKi:  6.30E+3nMAssay Description:Inhibition of [3H]CHA binding to Adenosine A1 receptor in rat cerebral cortical membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Marion Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50004716(CHEMBL111729 | 2-Methyl-3,6-diphenyl-4-propoxy-2,6...)
Affinity DataKi:  7.40E+3nMAssay Description:Inhibition of [3H]CHA binding to Adenosine A1 receptor in rat cerebral cortical membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Marion Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50004721(7-Benzyl-3-phenyl-5-propoxy-6,7-dihydro-3H-1,3,4,5...)
Affinity DataKi:  9.00E+3nMAssay Description:Inhibition of [3H]CHA binding to Adenosine A1 receptor in rat cerebral cortical membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Marion Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50004714((S)-2-Benzyl-7-phenyl-5-propoxy-2,7-dihydro-3H-imi...)
Affinity DataKi:  9.40E+3nMAssay Description:Inhibition of [3H]CHA binding to Adenosine A1 receptor in rat cerebral cortical membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Rat)
Marion Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50004716(CHEMBL111729 | 2-Methyl-3,6-diphenyl-4-propoxy-2,6...)
Affinity DataKi:  1.10E+4nMAssay Description:Inhibition of [3H]NECA binding to Adenosine A2 receptor in rat brain striatumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Rat)
Marion Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50004715(CHEMBL322270 | 3-Phenyl-2-(9-phenyl-2-propoxy-9H-p...)
Affinity DataKi:  3.00E+4nMAssay Description:Inhibition of [3H]NECA binding to Adenosine A2 receptor in rat brain striatumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Marion Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50004710(2-Methyl-3,6-diphenyl-4-propoxy-2,6-dihydro-3H-1,3...)
Affinity DataKi:  3.30E+4nMAssay Description:Inhibition of [3H]CHA binding to Adenosine A1 receptor in rat cerebral cortical membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Rat)
Marion Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50004710(2-Methyl-3,6-diphenyl-4-propoxy-2,6-dihydro-3H-1,3...)
Affinity DataKi:  4.50E+4nMAssay Description:Inhibition of [3H]NECA binding to Adenosine A2 receptor in rat brain striatumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Rat)
Marion Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50004722((R)-8-Benzyl-3-phenyl-5-propoxy-7,8-dihydro-3H-imi...)
Affinity DataKi:  7.20E+4nMAssay Description:Inhibition of [3H]NECA binding to Adenosine A2 receptor in rat brain striatumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Rat)
Marion Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50004713(CHEMBL320319 | (R)-2-Benzyl-7-phenyl-5-propoxy-2,7...)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of [3H]NECA binding to Adenosine A2 receptor in rat brain striatumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed