Compile Data Set for Download or QSAR
Report error Found 18 Enz. Inhib. hit(s) with all data for entry = 50000347
TargetPolyunsaturated fatty acid 5-lipoxygenase(Rat)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50004679(CHEMBL85000 | 2-Benzyl-naphthalen-1-ol | 2-Benzyl-...)
Affinity DataIC50: 19nMAssay Description:Inhibitory activity against 5-lipoxygenase of RBL-1 cell lineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1/2(Bovine)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM17638(indometacin | Indocin | 2-{1-[(4-chlorophenyl)carb...)
Affinity DataIC50: 430nMAssay Description:Inhibitory activity against Prostaglandin G/H synthase (bovine seminal vesicles)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetPolyunsaturated fatty acid 5-lipoxygenase(Rat)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50004677(Acetic acid 4-acetoxy-6-chloro-2,3-dimethoxy-napht...)
Affinity DataIC50: 740nMAssay Description:Inhibitory activity against 5-lipoxygenase of RBL-1 cell lineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Rat)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM31768(Nizoral | CHEMBL295698 | Panfungol | Ketoconazole)
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibitory activity against 5-lipoxygenase of RBL-1 cell lineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Rat)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM17638(indometacin | Indocin | 2-{1-[(4-chlorophenyl)carb...)
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibitory activity against 5-lipoxygenase of RBL-1 cell lineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Rat)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50004678(CHEMBL108795 | 2-Imidazol-1-yl-1-(4-pyridin-4-yl-p...)
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibitory activity against 5-lipoxygenase of RBL-1 cell lineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Rat)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50004676(CHEMBL321024 | 1-(4-Fluoro-phenyl)-2-imidazol-1-yl...)
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibitory activity against 5-lipoxygenase of RBL-1 cell lineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1/2(Bovine)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM31768(Nizoral | CHEMBL295698 | Panfungol | Ketoconazole)
Affinity DataIC50: 7.50E+5nMAssay Description:Inhibitory activity against Prostaglandin G/H synthase (bovine seminal vesicles)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1/2(Bovine)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50004678(CHEMBL108795 | 2-Imidazol-1-yl-1-(4-pyridin-4-yl-p...)
Affinity DataIC50: 7.50E+5nMAssay Description:Inhibitory activity against Prostaglandin G/H synthase (bovine seminal vesicles)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1/2(Bovine)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50004676(CHEMBL321024 | 1-(4-Fluoro-phenyl)-2-imidazol-1-yl...)
Affinity DataIC50: 7.50E+5nMAssay Description:Inhibitory activity against Prostaglandin G/H synthase (bovine seminal vesicles)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1/2(Bovine)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50004679(CHEMBL85000 | 2-Benzyl-naphthalen-1-ol | 2-Benzyl-...)
Affinity DataIC50: 7.50E+5nMAssay Description:Inhibitory activity against Prostaglandin G/H synthase (bovine seminal vesicles)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1/2(Bovine)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50004677(Acetic acid 4-acetoxy-6-chloro-2,3-dimethoxy-napht...)
Affinity DataIC50: 7.50E+5nMAssay Description:Inhibitory activity against Prostaglandin G/H synthase (bovine seminal vesicles)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPhospholipase A2, major isoenzyme(Pig)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM17638(indometacin | Indocin | 2-{1-[(4-chlorophenyl)carb...)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibitory activity against phospholipase A2 of Croatalus adamanteusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPhospholipase A2, major isoenzyme(Pig)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM31768(Nizoral | CHEMBL295698 | Panfungol | Ketoconazole)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibitory activity against phospholipase A2 of Croatalus adamanteusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPhospholipase A2, major isoenzyme(Pig)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50004679(CHEMBL85000 | 2-Benzyl-naphthalen-1-ol | 2-Benzyl-...)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibitory activity against phospholipase A2 of Croatalus adamanteusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPhospholipase A2, major isoenzyme(Pig)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50004678(CHEMBL108795 | 2-Imidazol-1-yl-1-(4-pyridin-4-yl-p...)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibitory activity against phospholipase A2 of Croatalus adamanteusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPhospholipase A2, major isoenzyme(Pig)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50004677(Acetic acid 4-acetoxy-6-chloro-2,3-dimethoxy-napht...)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibitory activity against phospholipase A2 of Croatalus adamanteusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPhospholipase A2, major isoenzyme(Pig)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50004676(CHEMBL321024 | 1-(4-Fluoro-phenyl)-2-imidazol-1-yl...)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibitory activity against phospholipase A2 of Croatalus adamanteusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed