Compile Data Set for Download or QSAR
Report error Found 30 Enz. Inhib. hit(s) with all data for entry = 50014511
TargetDisintegrin and metalloproteinase domain-containing protein 17(Human)
Hokkaido Collaboration Center N-21

Curated by ChEMBL
LigandPNGBDBM50141577((2R,3R,4R,5R)-1-(4-But-2-ynyloxy-benzenesulfonyl)-...)
Affinity DataIC50: 28nMAssay Description:Inhibition of heparin-binding HB-EGF sheddingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Human)
Hokkaido Collaboration Center N-21

Curated by ChEMBL
LigandPNGBDBM50143732((2R,3R,4R,5R)-1-(4-Benzyloxy-benzenesulfonyl)-3,4,...)
Affinity DataIC50: 84nMAssay Description:Inhibition of heparin-binding HB-EGF sheddingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Human)
Hokkaido Collaboration Center N-21

Curated by ChEMBL
LigandPNGBDBM50143729((2R,3R,4R,5R)-3,4,5-Trihydroxy-1-(4-phenoxy-benzen...)
Affinity DataIC50: 340nMAssay Description:Inhibition of heparin-binding HB-EGF sheddingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Human)
Hokkaido Collaboration Center N-21

Curated by ChEMBL
LigandPNGBDBM50131385((2R,3R,4R,5S)-N,3,4,5-tetrahydroxy-1-(4-phenoxyphe...)
Affinity DataIC50: 350nMAssay Description:Inhibition of heparin-binding HB-EGF sheddingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Human)
Hokkaido Collaboration Center N-21

Curated by ChEMBL
LigandPNGBDBM50143731((2R,3R,4R,5R)-3,4,5-Trihydroxy-1-(4-methoxy-benzen...)
Affinity DataIC50: 450nMAssay Description:Inhibition of heparin-binding HB-EGF sheddingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Human)
Hokkaido Collaboration Center N-21

Curated by ChEMBL
LigandPNGBDBM50143730((2R,3R,4R,5R)-1-(Biphenyl-4-sulfonyl)-3,4,5-trihyd...)
Affinity DataIC50: 2.10E+4nMAssay Description:Inhibition of heparin-binding HB-EGF sheddingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMatrix metalloproteinase-9(Human)
Hokkaido Collaboration Center N-21

Curated by ChEMBL
LigandPNGBDBM50131385((2R,3R,4R,5S)-N,3,4,5-tetrahydroxy-1-(4-phenoxyphe...)
Affinity DataKi:  0.0600nMAssay Description:Inhibition of human recombinant matrix metalloprotease 9More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMatrix metalloproteinase-9(Human)
Hokkaido Collaboration Center N-21

Curated by ChEMBL
LigandPNGBDBM50143729((2R,3R,4R,5R)-3,4,5-Trihydroxy-1-(4-phenoxy-benzen...)
Affinity DataKi:  0.0970nMAssay Description:Inhibition of human recombinant matrix metalloprotease 9More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetStromelysin-1(Human)
Hokkaido Collaboration Center N-21

Curated by ChEMBL
LigandPNGBDBM50143729((2R,3R,4R,5R)-3,4,5-Trihydroxy-1-(4-phenoxy-benzen...)
Affinity DataKi:  0.350nMAssay Description:Inhibition of human recombinant matrix metalloprotease 3More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetStromelysin-1(Human)
Hokkaido Collaboration Center N-21

Curated by ChEMBL
LigandPNGBDBM50131385((2R,3R,4R,5S)-N,3,4,5-tetrahydroxy-1-(4-phenoxyphe...)
Affinity DataKi:  0.510nMAssay Description:Inhibition of human recombinant matrix metalloprotease 3More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Human)
Hokkaido Collaboration Center N-21

Curated by ChEMBL
LigandPNGBDBM50141577((2R,3R,4R,5R)-1-(4-But-2-ynyloxy-benzenesulfonyl)-...)
Affinity DataKi:  0.530nMAssay Description:Inhibition of human tumor necrosis factor alpha converting enzymeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Human)
Hokkaido Collaboration Center N-21

Curated by ChEMBL
LigandPNGBDBM50143732((2R,3R,4R,5R)-1-(4-Benzyloxy-benzenesulfonyl)-3,4,...)
Affinity DataKi:  1.70nMAssay Description:Inhibition of human tumor necrosis factor alpha converting enzymeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetStromelysin-1(Human)
Hokkaido Collaboration Center N-21

Curated by ChEMBL
LigandPNGBDBM50143731((2R,3R,4R,5R)-3,4,5-Trihydroxy-1-(4-methoxy-benzen...)
Affinity DataKi:  2nMAssay Description:Inhibition of human recombinant matrix metalloprotease 3More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMatrix metalloproteinase-9(Human)
Hokkaido Collaboration Center N-21

Curated by ChEMBL
LigandPNGBDBM50143731((2R,3R,4R,5R)-3,4,5-Trihydroxy-1-(4-methoxy-benzen...)
Affinity DataKi:  2nMAssay Description:Inhibition of human recombinant matrix metalloprotease 9More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetStromelysin-1(Human)
Hokkaido Collaboration Center N-21

Curated by ChEMBL
LigandPNGBDBM50143732((2R,3R,4R,5R)-1-(4-Benzyloxy-benzenesulfonyl)-3,4,...)
Affinity DataKi:  2.10nMAssay Description:Inhibition of human recombinant matrix metalloprotease 3More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Human)
Hokkaido Collaboration Center N-21

Curated by ChEMBL
LigandPNGBDBM50131385((2R,3R,4R,5S)-N,3,4,5-tetrahydroxy-1-(4-phenoxyphe...)
Affinity DataKi:  2.30nMAssay Description:Inhibition of human tumor necrosis factor alpha converting enzymeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetStromelysin-1(Human)
Hokkaido Collaboration Center N-21

Curated by ChEMBL
LigandPNGBDBM50141577((2R,3R,4R,5R)-1-(4-But-2-ynyloxy-benzenesulfonyl)-...)
Affinity DataKi:  3.30nMAssay Description:Inhibition of human recombinant matrix metalloprotease 3More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetInterstitial collagenase(Human)
Hokkaido Collaboration Center N-21

Curated by ChEMBL
LigandPNGBDBM50143729((2R,3R,4R,5R)-3,4,5-Trihydroxy-1-(4-phenoxy-benzen...)
Affinity DataKi:  5.30nMAssay Description:Inhibition of human recombinant matrix metalloprotease 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Human)
Hokkaido Collaboration Center N-21

Curated by ChEMBL
LigandPNGBDBM50143729((2R,3R,4R,5R)-3,4,5-Trihydroxy-1-(4-phenoxy-benzen...)
Affinity DataKi:  6.20nMAssay Description:Inhibition of human tumor necrosis factor alpha converting enzymeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMatrix metalloproteinase-9(Human)
Hokkaido Collaboration Center N-21

Curated by ChEMBL
LigandPNGBDBM50143732((2R,3R,4R,5R)-1-(4-Benzyloxy-benzenesulfonyl)-3,4,...)
Affinity DataKi:  7.40nMAssay Description:Inhibition of human recombinant matrix metalloprotease 9More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetInterstitial collagenase(Human)
Hokkaido Collaboration Center N-21

Curated by ChEMBL
LigandPNGBDBM50131385((2R,3R,4R,5S)-N,3,4,5-tetrahydroxy-1-(4-phenoxyphe...)
Affinity DataKi:  8nMAssay Description:Inhibition of human recombinant matrix metalloprotease 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMatrix metalloproteinase-9(Human)
Hokkaido Collaboration Center N-21

Curated by ChEMBL
LigandPNGBDBM50141577((2R,3R,4R,5R)-1-(4-But-2-ynyloxy-benzenesulfonyl)-...)
Affinity DataKi:  14nMAssay Description:Inhibition of human recombinant matrix metalloprotease 9More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Human)
Hokkaido Collaboration Center N-21

Curated by ChEMBL
LigandPNGBDBM50143731((2R,3R,4R,5R)-3,4,5-Trihydroxy-1-(4-methoxy-benzen...)
Affinity DataKi:  15nMAssay Description:Inhibition of human tumor necrosis factor alpha converting enzymeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Human)
Hokkaido Collaboration Center N-21

Curated by ChEMBL
LigandPNGBDBM50143730((2R,3R,4R,5R)-1-(Biphenyl-4-sulfonyl)-3,4,5-trihyd...)
Affinity DataKi:  21nMAssay Description:Inhibition of human tumor necrosis factor alpha converting enzymeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetInterstitial collagenase(Human)
Hokkaido Collaboration Center N-21

Curated by ChEMBL
LigandPNGBDBM50143731((2R,3R,4R,5R)-3,4,5-Trihydroxy-1-(4-methoxy-benzen...)
Affinity DataKi:  26nMAssay Description:Inhibition of human recombinant matrix metalloprotease 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMatrix metalloproteinase-9(Human)
Hokkaido Collaboration Center N-21

Curated by ChEMBL
LigandPNGBDBM50143730((2R,3R,4R,5R)-1-(Biphenyl-4-sulfonyl)-3,4,5-trihyd...)
Affinity DataKi:  47nMAssay Description:Inhibition of human recombinant matrix metalloprotease 9More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetStromelysin-1(Human)
Hokkaido Collaboration Center N-21

Curated by ChEMBL
LigandPNGBDBM50143730((2R,3R,4R,5R)-1-(Biphenyl-4-sulfonyl)-3,4,5-trihyd...)
Affinity DataKi:  50nMAssay Description:Inhibition of human recombinant matrix metalloprotease 3More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetInterstitial collagenase(Human)
Hokkaido Collaboration Center N-21

Curated by ChEMBL
LigandPNGBDBM50141577((2R,3R,4R,5R)-1-(4-But-2-ynyloxy-benzenesulfonyl)-...)
Affinity DataKi:  128nMAssay Description:Inhibition of human recombinant matrix metalloprotease 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetInterstitial collagenase(Human)
Hokkaido Collaboration Center N-21

Curated by ChEMBL
LigandPNGBDBM50143730((2R,3R,4R,5R)-1-(Biphenyl-4-sulfonyl)-3,4,5-trihyd...)
Affinity DataKi:  162nMAssay Description:Inhibition of human recombinant matrix metalloprotease 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetInterstitial collagenase(Human)
Hokkaido Collaboration Center N-21

Curated by ChEMBL
LigandPNGBDBM50143732((2R,3R,4R,5R)-1-(4-Benzyloxy-benzenesulfonyl)-3,4,...)
Affinity DataKi: >850nMAssay Description:Inhibition of human recombinant matrix metalloprotease 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed