Compile Data Set for Download or QSAR
Report error Found 19 Enz. Inhib. hit(s) with all data for entry = 50037283
TargetNitric oxide synthase, inducible(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50139793((S)-6-Acetimidoylamino-2-(S)-amino-5-fluoro-hexano...)
Affinity DataIC50: 2.36E+3nMAssay Description:Inhibition concentration against Inducible nitric oxide synthase (iNOS) at 10 uM concentrationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetNitric oxide synthase, inducible(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50063300(l-NIL | CHEMBL1744034 | (L-N6-1-iminoethyl)lysine ...)
Affinity DataIC50: 4.90E+3nMAssay Description:Inhibition concentration against Inducible nitric oxide synthase (iNOS) at 10 uM concentrationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetNitric oxide synthase, inducible(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50139792(6-Acetimidoylamino-2-amino-5-fluoro-hexanoic acid ...)
Affinity DataIC50: 7.84E+3nMAssay Description:Inhibition concentration against Inducible nitric oxide synthase (iNOS) at 10 uM concentrationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetNitric oxide synthase, inducible(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50139797((S)-6-Acetimidoylamino-2-amino-5,5-difluoro-hexano...)
Affinity DataIC50: 8.75E+3nMAssay Description:Inhibition concentration against Inducible nitric oxide synthase (iNOS) at 10 uM concentrationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetNitric oxide synthase, inducible(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50139794(6-Acetimidoylamino-2-amino-5,5-difluoro-hexanoic a...)
Affinity DataIC50: 2.14E+4nMAssay Description:Inhibition concentration against Inducible nitric oxide synthase (iNOS) at 10 uM concentrationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetNitric oxide synthase, brain(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50139793((S)-6-Acetimidoylamino-2-(S)-amino-5-fluoro-hexano...)
Affinity DataIC50: 2.17E+4nMAssay Description:Inhibition concentration against Neuronal nitric oxide synthase (nNOS) at 10 uM concentrationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetNitric oxide synthase, endothelial(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50139796((R)-6-Acetimidoylamino-2-(S)-amino-5-fluoro-hexano...)
Affinity DataIC50: 2.82E+4nMAssay Description:Inhibition concentration against Endothelial nitric oxide synthase (eNOS) at 10 uM concentrationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetNitric oxide synthase, brain(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50139797((S)-6-Acetimidoylamino-2-amino-5,5-difluoro-hexano...)
Affinity DataIC50: 3.38E+4nMAssay Description:Inhibition concentration against Neuronal nitric oxide synthase (nNOS) at 10 uM concentrationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetNitric oxide synthase, brain(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50063300(l-NIL | CHEMBL1744034 | (L-N6-1-iminoethyl)lysine ...)
Affinity DataIC50: 3.50E+4nMAssay Description:Inhibition concentration against Neuronal nitric oxide synthase (nNOS) at 10 uM concentrationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetNitric oxide synthase, inducible(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50139795((S)-6-Acetimidoylamino-2-(R)-amino-5-fluoro-hexano...)
Affinity DataIC50: 4.78E+4nMAssay Description:Inhibition concentration against Inducible nitric oxide synthase (iNOS) at 10 uM concentrationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetNitric oxide synthase, endothelial(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50139797((S)-6-Acetimidoylamino-2-amino-5,5-difluoro-hexano...)
Affinity DataIC50: 5.75E+4nMAssay Description:Inhibition concentration against Endothelial nitric oxide synthase (eNOS) at 10 uM concentrationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetNitric oxide synthase, brain(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50139792(6-Acetimidoylamino-2-amino-5-fluoro-hexanoic acid ...)
Affinity DataIC50: 7.04E+4nMAssay Description:Inhibition concentration against Neuronal nitric oxide synthase (nNOS) at 10 uM concentrationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetNitric oxide synthase, endothelial(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50139793((S)-6-Acetimidoylamino-2-(S)-amino-5-fluoro-hexano...)
Affinity DataIC50: 8.10E+4nMAssay Description:Inhibition concentration against Endothelial nitric oxide synthase (eNOS) at 10 uM concentrationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetNitric oxide synthase, endothelial(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50063300(l-NIL | CHEMBL1744034 | (L-N6-1-iminoethyl)lysine ...)
Affinity DataIC50: 1.38E+5nMAssay Description:Inhibition concentration against Endothelial nitric oxide synthase (eNOS) at 10 uM concentrationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetNitric oxide synthase, endothelial(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50139794(6-Acetimidoylamino-2-amino-5,5-difluoro-hexanoic a...)
Affinity DataIC50: 1.39E+5nMAssay Description:Inhibition concentration against Endothelial nitric oxide synthase (eNOS) at 10 uM concentrationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetNitric oxide synthase, brain(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50139794(6-Acetimidoylamino-2-amino-5,5-difluoro-hexanoic a...)
Affinity DataIC50: 1.40E+5nMAssay Description:Inhibition concentration against Neuronal nitric oxide synthase (nNOS) at 10 uM concentrationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetNitric oxide synthase, endothelial(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50139792(6-Acetimidoylamino-2-amino-5-fluoro-hexanoic acid ...)
Affinity DataIC50: 1.82E+5nMAssay Description:Inhibition concentration against Endothelial nitric oxide synthase (eNOS) at 10 uM concentrationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetNitric oxide synthase, brain(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50139795((S)-6-Acetimidoylamino-2-(R)-amino-5-fluoro-hexano...)
Affinity DataIC50: 3.11E+5nMAssay Description:Inhibition concentration against Neuronal nitric oxide synthase (nNOS) at 10 uM concentrationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetNitric oxide synthase, endothelial(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50139795((S)-6-Acetimidoylamino-2-(R)-amino-5-fluoro-hexano...)
Affinity DataIC50: 3.74E+5nMAssay Description:Inhibition concentration against Endothelial nitric oxide synthase (eNOS) at 10 uM concentrationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed