Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 50014220
LigandPNGBDBM86248(NSC_3019 | CAS_364-98-7 | diazoxide)
Affinity DataEC50:  8.80E+3nMAssay Description:Maximum activation of human KATP (SUR1/Kir6.2) channel expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50139705(4-Nitro-3-(4-nitro-phenyl)-5-trifluoromethyl-1H-py...)
Affinity DataEC50:  700nMAssay Description:Maximum activation of human KATP (SUR1/Kir6.2) channel expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50139708(3-(4-Nitro-phenyl)-5-trifluoromethyl-1H-pyrazole |...)
Affinity DataEC50: >3.00E+4nMAssay Description:Maximum activation of human KATP (SUR1/Kir6.2) channel expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50139710(4-Nitro-3-phenyl-5-trifluoromethyl-1H-pyrazole | C...)
Affinity DataEC50:  3.00E+4nMAssay Description:Maximum activation of human KATP (SUR1/Kir6.2) channel expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50139709(3-(2,4-Bis-trifluoromethyl-phenyl)-4-nitro-5-trifl...)
Affinity DataEC50:  540nMAssay Description:Maximum activation of human KATP (SUR1/Kir6.2) channel expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50139707(4-Nitro-3-(4-nitro-phenyl)-5-trifluoromethyl-isoxa...)
Affinity DataEC50: >3.00E+4nMAssay Description:Maximum activation of human KATP (SUR1/Kir6.2) channel expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50139706(3-(2,4-Dinitro-phenyl)-4-nitro-5-trifluoromethyl-1...)
Affinity DataEC50:  70nMAssay Description:Maximum activation of human KATP (SUR1/Kir6.2) channel expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50139704(3-(2,4-Difluoro-phenyl)-4-nitro-5-trifluoromethyl-...)
Affinity DataEC50:  1.15E+3nMAssay Description:Maximum activation of human KATP (SUR1/Kir6.2) channel expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed