Compile Data Set for Download or QSAR
Report error Found 23 Enz. Inhib. hit(s) with all data for entry = 50048589
LigandPNGBDBM20461(Zostrix | (E)-N-[(4-hydroxy-3-methoxyphenyl)methyl...)
Affinity DataEC50:  30nMAssay Description:In vitro agonist activity, increased [Ca2+] influx, at vanilloid receptor of rat dorsal root gangliaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2018
Entry Details Article
PubMedPDB3D3D Structure (crystal)
LigandPNGBDBM20315(3-[(4-tert-butylphenyl)methyl]-1-[(4-methanesulfon...)
Affinity DataIC50: 110nMAssay Description:In vitro antagonist activity at the vanilloid receptor in rat DRG neurons.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2018
Entry Details Article
PubMed
LigandPNGBDBM50223778(CHEMBL164875)
Affinity DataIC50: 300nMAssay Description:In vitro antagonist activity at the vanilloid receptor in rat DRG neurons.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2018
Entry Details Article
PubMed
LigandPNGBDBM20284(N-[2-(4-chlorophenyl)ethyl]-7,8-dihydroxy-2,3,4,5-...)
Affinity DataIC50: 650nMAssay Description:In vitro antagonist activity at the vanilloid receptor in rat DRG neurons.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2018
Entry Details Article
PubMedPDB3D3D Structure (crystal)
LigandPNGBDBM50139640(N-4-Substituted-benzyl-N'-tert-butylbenzyl thioure...)
Affinity DataIC50: 1.00E+3nMAssay Description:In vitro antagonist activity at the vanilloid receptor in rat DRG neurons.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2018
Entry Details Article
PubMed
LigandPNGBDBM50223786(CHEMBL165036)
Affinity DataIC50: 1.30E+3nMAssay Description:In vitro antagonist activity at the vanilloid receptor in rat DRG neurons.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2018
Entry Details Article
PubMed
LigandPNGBDBM50223825(CHEMBL351511)
Affinity DataIC50: 1.50E+3nMAssay Description:In vitro antagonist activity at the vanilloid receptor in rat DRG neurons.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2018
Entry Details Article
PubMed
LigandPNGBDBM50223785(CHEMBL163834)
Affinity DataIC50: 2.50E+3nMAssay Description:In vitro antagonist activity at the vanilloid receptor in rat DRG neurons.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2018
Entry Details Article
PubMed
LigandPNGBDBM50223779(CHEMBL167960)
Affinity DataIC50: 2.50E+3nMAssay Description:In vitro antagonist activity at the vanilloid receptor in rat DRG neurons.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2018
Entry Details Article
PubMed
LigandPNGBDBM50223823(CHEMBL355156)
Affinity DataIC50: 3.80E+3nMAssay Description:In vitro antagonist activity at the vanilloid receptor in rat DRG neurons.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2018
Entry Details Article
PubMed
LigandPNGBDBM50223775(CHEMBL165254)
Affinity DataIC50: 4.10E+3nMAssay Description:In vitro antagonist activity at the vanilloid receptor in rat DRG neurons.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2018
Entry Details Article
PubMed
LigandPNGBDBM50223822(CHEMBL434280)
Affinity DataIC50: 4.50E+3nMAssay Description:In vitro antagonist activity at the vanilloid receptor in rat DRG neurons.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2018
Entry Details Article
PubMed
LigandPNGBDBM50223774(CHEMBL165129)
Affinity DataEC50:  7.00E+3nMAssay Description:In vitro agonist activity, increased [Ca2+] influx, at vanilloid receptor of rat dorsal root gangliaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2018
Entry Details Article
PubMed
LigandPNGBDBM50223780(CHEMBL166987)
Affinity DataIC50: 9.30E+3nMAssay Description:In vitro antagonist activity at the vanilloid receptor in rat DRG neurons.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2018
Entry Details Article
PubMed
LigandPNGBDBM50223824(CHEMBL168070)
Affinity DataIC50: 1.17E+4nMAssay Description:In vitro antagonist activity at the vanilloid receptor in rat DRG neurons.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2018
Entry Details Article
PubMed
LigandPNGBDBM50223784(CHEMBL164380)
Affinity DataIC50: 1.24E+4nMAssay Description:In vitro antagonist activity at the vanilloid receptor in rat DRG neurons.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2018
Entry Details Article
PubMed
LigandPNGBDBM50223777(CHEMBL163678)
Affinity DataIC50: 1.24E+4nMAssay Description:In vitro antagonist activity at the vanilloid receptor in rat DRG neurons.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2018
Entry Details Article
PubMed
LigandPNGBDBM50223776(CHEMBL354812)
Affinity DataIC50: 1.46E+4nMAssay Description:In vitro antagonist activity at the vanilloid receptor in rat DRG neurons.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2018
Entry Details Article
PubMed
LigandPNGBDBM50223772(CHEMBL164768)
Affinity DataIC50: 3.00E+4nMAssay Description:In vitro antagonist activity at vanilloid receptor in rat dorsal root ganglia (partial at 30 uM)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2018
Entry Details Article
PubMed
LigandPNGBDBM50223773(CHEMBL166988)
Affinity DataEC50: >3.00E+4nMAssay Description:In vitro agonist activity, increased [Ca2+] influx, at vanilloid receptor of rat dorsal root ganglia (partial at 30 uM)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2018
Entry Details Article
PubMed
LigandPNGBDBM50223781(CHEMBL167338)
Affinity DataIC50: 3.00E+4nMAssay Description:In vitro antagonist activity at vanilloid receptor in rat dorsal root ganglia (partial at 30 uM)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2018
Entry Details Article
PubMed
LigandPNGBDBM50223782(CHEMBL349647)
Affinity DataEC50: >3.00E+4nMAssay Description:In vitro agonist activity, increased [Ca2+] influx, at vanilloid receptor of rat dorsal root ganglia (partial at 30 uM)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2018
Entry Details Article
PubMed
LigandPNGBDBM50223773(CHEMBL166988)
Affinity DataIC50: 3.00E+4nMAssay Description:In vitro antagonist activity at vanilloid receptor in rat dorsal root ganglia (partial at 30 uM)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2018
Entry Details Article
PubMed