Report error Found 60 Enz. Inhib. hit(s) with all data for entry = 50014050
Affinity DataKi: 0.400nMAssay Description:Binding affinity at dopamine receptor D3 on Sf9 cells by [125I]IABN displacement.More data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:Binding affinity at dopamine receptor D3 on Sf9 cells by [125I]IABN displacement.More data for this Ligand-Target Pair
Affinity DataKi: 0.900nMAssay Description:Binding affinity at dopamine receptor D3 on Sf9 cells by [125I]IABN displacement.More data for this Ligand-Target Pair
Affinity DataKi: 1.40nMAssay Description:Binding affinity at dopamine receptor D3 on Sf9 cells by [125I]IABN displacement.More data for this Ligand-Target Pair
Affinity DataKi: 1.40nMAssay Description:Binding affinity at dopamine receptor D3 on Sf9 cells by [125I]IABN displacement.More data for this Ligand-Target Pair
Affinity DataKi: 2.10nMAssay Description:Binding affinity at dopamine receptor D3 on Sf9 cells by [125I]IABN displacement.More data for this Ligand-Target Pair
Affinity DataKi: 3.20nMAssay Description:Binding affinity at dopamine receptor D3 on Sf9 cells by [125I]IABN displacement.More data for this Ligand-Target Pair
Affinity DataKi: 3.80nMAssay Description:Binding affinity at dopamine receptor D3 on Sf9 cells by [125I]IABN displacement.More data for this Ligand-Target Pair
Affinity DataKi: 3.90nMAssay Description:Binding affinity at dopamine receptor D3 on Sf9 cells by [125I]IABN displacement.More data for this Ligand-Target Pair
Affinity DataKi: 5.80nMAssay Description:Binding affinity at dopamine receptor D2 on Sf9 cells by [125I]IABN displacement.More data for this Ligand-Target Pair
Affinity DataKi: 8nMAssay Description:Binding affinity at dopamine receptor D3 on Sf9 cells by [125I]IABN displacement.More data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Binding affinity at dopamine receptor D3 on Sf9 cells by [125I]IABN displacement.More data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Human)
Wake Forest University School of Medicine
Curated by ChEMBL
Wake Forest University School of Medicine
Curated by ChEMBL
Affinity DataKi: 15nMAssay Description:Inhibition of [3H](+)-pentazocine binding to Sigma opioid receptor of guiena pig brain membraneMore data for this Ligand-Target Pair
Affinity DataKi: 18nMAssay Description:Binding affinity at dopamine receptor D3 on Sf9 cells by [125I]IABN displacement.More data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Human)
Wake Forest University School of Medicine
Curated by ChEMBL
Wake Forest University School of Medicine
Curated by ChEMBL
Affinity DataKi: 18nMAssay Description:Inhibition of [3H](+)-pentazocine binding to Sigma opioid receptor of guiena pig brain membraneMore data for this Ligand-Target Pair
Affinity DataKi: 21nMAssay Description:Binding affinity at dopamine receptor D3 on Sf9 cells by [125I]IABN displacement.More data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Human)
Wake Forest University School of Medicine
Curated by ChEMBL
Wake Forest University School of Medicine
Curated by ChEMBL
Affinity DataKi: 22nMAssay Description:Inhibition of [3H](+)-pentazocine binding to Sigma opioid receptor of guiena pig brain membraneMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Human)
Wake Forest University School of Medicine
Curated by ChEMBL
Wake Forest University School of Medicine
Curated by ChEMBL
Affinity DataKi: 28nMAssay Description:Inhibition of [3H](+)-pentazocine binding to Sigma opioid receptor of guiena pig brain membraneMore data for this Ligand-Target Pair
Affinity DataKi: 30nMAssay Description:Binding affinity at dopamine receptor D2 on Sf9 cells by [125I]IABN displacement.More data for this Ligand-Target Pair
Affinity DataKi: 33nMAssay Description:Binding affinity at dopamine receptor D2 on Sf9 cells by [125I]IABN displacement.More data for this Ligand-Target Pair
Affinity DataKi: 48nMAssay Description:Binding affinity for human dopamine receptor D4 using [125I]IABN as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 58nMAssay Description:Binding affinity at dopamine receptor D2 on Sf9 cells by [125I]IABN displacement.More data for this Ligand-Target Pair
Affinity DataKi: 59nMAssay Description:Binding affinity at dopamine receptor D2 on Sf9 cells by [125I]IABN displacement.More data for this Ligand-Target Pair
Affinity DataKi: 82nMAssay Description:Binding affinity at dopamine receptor D3 on Sf9 cells by [125I]IABN displacement.More data for this Ligand-Target Pair
Affinity DataKi: 89nMAssay Description:Binding affinity at dopamine receptor D2 on Sf9 cells by [125I]IABN displacement.More data for this Ligand-Target Pair
Affinity DataKi: 107nMAssay Description:Binding affinity at dopamine receptor D2 on Sf9 cells by [125I]IABN displacement.More data for this Ligand-Target Pair
Affinity DataKi: 107nMAssay Description:Binding affinity at dopamine receptor D3 on Sf9 cells by [125I]IABN displacement.More data for this Ligand-Target Pair
Affinity DataKi: 127nMAssay Description:Binding affinity at dopamine receptor D3 on Sf9 cells by [125I]IABN displacement.More data for this Ligand-Target Pair
Affinity DataKi: 132nMAssay Description:Binding affinity at dopamine receptor D2 on Sf9 cells by [125I]IABN displacement.More data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Human)
Wake Forest University School of Medicine
Curated by ChEMBL
Wake Forest University School of Medicine
Curated by ChEMBL
Affinity DataKi: 189nMAssay Description:Inhibition of [3H](+)-pentazocine binding to Sigma opioid receptor of guiena pig brain membraneMore data for this Ligand-Target Pair
Affinity DataKi: 217nMAssay Description:Binding affinity at dopamine receptor D2 on Sf9 cells by [125I]IABN displacement.More data for this Ligand-Target Pair
Affinity DataKi: 241nMAssay Description:Binding affinity at dopamine receptor D2 on Sf9 cells by [125I]IABN displacement.More data for this Ligand-Target Pair
Affinity DataKi: 262nMAssay Description:Binding affinity at dopamine receptor D2 on Sf9 cells by [125I]IABN displacement.More data for this Ligand-Target Pair
Affinity DataKi: 265nMAssay Description:Binding affinity for human dopamine receptor D4 using [125I]IABN as radioligandMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Human)
Wake Forest University School of Medicine
Curated by ChEMBL
Wake Forest University School of Medicine
Curated by ChEMBL
Affinity DataKi: 277nMAssay Description:Inhibition of [3H](+)-pentazocine binding to Sigma opioid receptor of guiena pig brain membraneMore data for this Ligand-Target Pair
Affinity DataKi: 311nMAssay Description:Binding affinity at dopamine receptor D3 on Sf9 cells by [125I]IABN displacement.More data for this Ligand-Target Pair
Affinity DataKi: 313nMAssay Description:Binding affinity at dopamine receptor D3 on Sf9 cells by [125I]IABN displacement.More data for this Ligand-Target Pair
Affinity DataKi: 430nMAssay Description:Binding affinity at dopamine receptor D2 on Sf9 cells by [125I]IABN displacement.More data for this Ligand-Target Pair
Affinity DataKi: 488nMAssay Description:Binding affinity at dopamine receptor D3 on Sf9 cells by [125I]IABN displacement.More data for this Ligand-Target Pair
Affinity DataKi: 627nMAssay Description:Binding affinity at dopamine receptor D3 on Sf9 cells by [125I]IABN displacement.More data for this Ligand-Target Pair
Affinity DataKi: 642nMAssay Description:Binding affinity at dopamine receptor D2 on Sf9 cells by [125I]IABN displacement.More data for this Ligand-Target Pair
Affinity DataKi: 714nMAssay Description:Binding affinity at dopamine receptor D2 on Sf9 cells by [125I]IABN displacement.More data for this Ligand-Target Pair
Affinity DataKi: 741nMAssay Description:Binding affinity at dopamine receptor D2 on Sf9 cells by [125I]IABN displacement.More data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Human)
Wake Forest University School of Medicine
Curated by ChEMBL
Wake Forest University School of Medicine
Curated by ChEMBL
Affinity DataKi: 751nMAssay Description:Inhibition of [3H](+)-pentazocine binding to Sigma opioid receptor of guiena pig brain membraneMore data for this Ligand-Target Pair
Affinity DataKi: 800nMAssay Description:Binding affinity for human dopamine receptor D4 using [125I]IABN as radioligandMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Human)
Wake Forest University School of Medicine
Curated by ChEMBL
Wake Forest University School of Medicine
Curated by ChEMBL
Affinity DataKi: 809nMAssay Description:Inhibition of [3H](+)-pentazocine binding to Sigma opioid receptor of guiena pig brain membraneMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Human)
Wake Forest University School of Medicine
Curated by ChEMBL
Wake Forest University School of Medicine
Curated by ChEMBL
Affinity DataKi: 1.16E+3nMAssay Description:Inhibition of [3H](+)-pentazocine binding to Sigma opioid receptor of guiena pig brain membraneMore data for this Ligand-Target Pair
Affinity DataKi: 1.35E+3nMAssay Description:Binding affinity for human dopamine receptor D4 using [125I]IABN as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 2.19E+3nMAssay Description:Binding affinity at dopamine receptor D2 on Sf9 cells by [125I]IABN displacement.More data for this Ligand-Target Pair
Affinity DataKi: 2.20E+3nMAssay Description:Binding affinity at dopamine receptor D2 on Sf9 cells by [125I]IABN displacement.More data for this Ligand-Target Pair



















