Compile Data Set for Download or QSAR
Report error Found 23 Enz. Inhib. hit(s) with all data for entry = 50048566
TargetHistone deacetylase(Human)
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM19149(Zolinza | suberoylanilide hydroxamic acid | CHEMBL...)
Affinity DataIC50: 280nMAssay Description:In vitro inhibitory activity against histone deacetylase (HDAC) isolated from HeLa nuclear extractMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2018
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetHistone deacetylase(Human)
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50222441(CHEMBL114237)
Affinity DataIC50: 1.40E+4nMAssay Description:In vitro inhibitory activity against histone deacetylase (HDAC) isolated from HeLa nuclear extractMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2018
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50222416(CHEMBL344920)
Affinity DataIC50: 1.70E+4nMAssay Description:In vitro inhibitory activity against histone deacetylase (HDAC) isolated from HeLa nuclear extractMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2018
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50222443(CHEMBL264784)
Affinity DataIC50: 1.00E+5nMAssay Description:In vitro inhibitory activity against histone deacetylase (HDAC) isolated from HeLa nuclear extractMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2018
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50222454(CHEMBL137003)
Affinity DataIC50: 1.00E+5nMAssay Description:In vitro inhibitory activity against histone deacetylase (HDAC) isolated from HeLa nuclear extractMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2018
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50222453(CHEMBL137695)
Affinity DataIC50: 1.00E+5nMAssay Description:In vitro inhibitory activity against histone deacetylase (HDAC) isolated from HeLa nuclear extractMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2018
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50222452(CHEMBL137100 | Octanedioic acid phenylamide pyridi...)
Affinity DataIC50: 1.00E+5nMAssay Description:In vitro inhibitory activity against histone deacetylase (HDAC) isolated from HeLa nuclear extractMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2018
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50222451(CHEMBL343377 | Octanedioic acid phenylamide thiazo...)
Affinity DataIC50: 1.00E+5nMAssay Description:In vitro inhibitory activity against histone deacetylase (HDAC) isolated from HeLa nuclear extractMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2018
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50222449(CHEMBL344475)
Affinity DataIC50: 1.00E+5nMAssay Description:In vitro inhibitory activity against histone deacetylase (HDAC) isolated from HeLa nuclear extractMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2018
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50222448(CHEMBL137278)
Affinity DataIC50: 1.00E+5nMAssay Description:In vitro inhibitory activity against histone deacetylase (HDAC) isolated from HeLa nuclear extractMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2018
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50222446(CHEMBL137672)
Affinity DataIC50: 1.00E+5nMAssay Description:In vitro inhibitory activity against histone deacetylase (HDAC) isolated from HeLa nuclear extractMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2018
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50222444(CHEMBL137036)
Affinity DataIC50: 1.00E+5nMAssay Description:In vitro inhibitory activity against histone deacetylase (HDAC) isolated from HeLa nuclear extractMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2018
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50222409(CHEMBL137333)
Affinity DataIC50: 1.00E+5nMAssay Description:In vitro inhibitory activity against histone deacetylase (HDAC) isolated from HeLa nuclear extractMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2018
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50222442(CHEMBL423356)
Affinity DataIC50: 1.00E+5nMAssay Description:In vitro inhibitory activity against histone deacetylase (HDAC) isolated from HeLa nuclear extractMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2018
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50222415(CHEMBL136992)
Affinity DataIC50: 1.00E+5nMAssay Description:In vitro inhibitory activity against histone deacetylase (HDAC) isolated from HeLa nuclear extractMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2018
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50222412(CHEMBL341701)
Affinity DataIC50: 1.00E+5nMAssay Description:In vitro inhibitory activity against histone deacetylase (HDAC) isolated from HeLa nuclear extractMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2018
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50222410(CHEMBL137216 | 7-Ureido-Heptanoic Acid Phenylamide)
Affinity DataIC50: 1.00E+5nMAssay Description:In vitro inhibitory activity against histone deacetylase (HDAC) isolated from HeLa nuclear extractMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2018
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50222414(CHEMBL324053 | CHEBI:61077 | BML-210)
Affinity DataIC50: 1.20E+5nMAssay Description:In vitro inhibitory activity against histone deacetylase (HDAC) isolated from HeLa nuclear extractMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2018
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50222447(CHEMBL138381)
Affinity DataIC50: 1.21E+5nMAssay Description:In vitro inhibitory activity against histone deacetylase (HDAC) isolated from HeLa nuclear extractMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2018
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50222413(CHEMBL112539)
Affinity DataIC50: 1.50E+5nMAssay Description:In vitro inhibitory activity against histone deacetylase (HDAC) isolated from HeLa nuclear extractMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2018
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50222450(CHEMBL137519)
Affinity DataIC50: 3.00E+5nMAssay Description:In vitro inhibitory activity against histone deacetylase (HDAC) isolated from HeLa nuclear extractMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2018
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50222445(CHEMBL422460)
Affinity DataIC50: 6.50E+5nMAssay Description:In vitro inhibitory activity against histone deacetylase (HDAC) isolated from HeLa nuclear extractMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2018
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50222411(CHEMBL136792)
Affinity DataIC50: 1.00E+6nMAssay Description:In vitro inhibitory activity against histone deacetylase (HDAC) isolated from HeLa nuclear extractMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2018
Entry Details Article
PubMed