Compile Data Set for Download or QSAR
Report error Found 16 Enz. Inhib. hit(s) with all data for entry = 50013747
LigandPNGBDBM50134315(CHEMBL331627 | 7-hydroxy-11-hydroxymethyl-12-methy...)
Affinity DataIC50: 1.70E+4nMAssay Description:Inhibition of [3H]-GGPP incorporation into recombinant human Ha-Ras-CVLL by Geranylgeranyl transferase type IMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50134315(CHEMBL331627 | 7-hydroxy-11-hydroxymethyl-12-methy...)
Affinity DataIC50: 8.00E+4nMAssay Description:Inhibition of [3H]FPP incorporation into recombinant human Ha-Ras-CVLS by farnesyl transferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50134312(Thioacetic acid S-(9-methoxy-2-methyl-1,4-dioxo-1,...)
Affinity DataIC50: 9.03E+4nMAssay Description:Inhibition of [3H]-GGPP incorporation into recombinant human Ha-Ras-CVLL by Geranylgeranyl transferase type IMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50134309(2-Methyl-2,3,10,10a-tetrahydro-pyrazino[1,2-a]indo...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of [3H]FPP incorporation into recombinant human Ha-Ras-CVLS by farnesyl transferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50134311(3-Benzyldisulfanyl-9-methoxy-2-methyl-2,3-dihydro-...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of [3H]-GGPP incorporation into recombinant human Ha-Ras-CVLL by Geranylgeranyl transferase type IMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50134310(9-Methoxy-2-methyl-2,3,10,10a-tetrahydro-pyrazino[...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of [3H]-GGPP incorporation into recombinant human Ha-Ras-CVLL by Geranylgeranyl transferase type IMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50134313(2-Methyl-2,3-dihydro-pyrazino[1,2-a]indole-1,4-dio...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of [3H]-GGPP incorporation into recombinant human Ha-Ras-CVLL by Geranylgeranyl transferase type IMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50134308(3-Benzyldisulfanyl-2-methyl-2,3-dihydro-pyrazino[1...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of [3H]FPP incorporation into recombinant human Ha-Ras-CVLS by farnesyl transferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50134309(2-Methyl-2,3,10,10a-tetrahydro-pyrazino[1,2-a]indo...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of [3H]-GGPP incorporation into recombinant human Ha-Ras-CVLL by Geranylgeranyl transferase type IMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50134314(9-Methoxy-2-methyl-2,3-dihydro-pyrazino[1,2-a]indo...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of [3H]-GGPP incorporation into recombinant human Ha-Ras-CVLL by Geranylgeranyl transferase type IMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50134314(9-Methoxy-2-methyl-2,3-dihydro-pyrazino[1,2-a]indo...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of [3H]FPP incorporation into recombinant human Ha-Ras-CVLS by farnesyl transferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50134313(2-Methyl-2,3-dihydro-pyrazino[1,2-a]indole-1,4-dio...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of [3H]FPP incorporation into recombinant human Ha-Ras-CVLS by farnesyl transferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50134308(3-Benzyldisulfanyl-2-methyl-2,3-dihydro-pyrazino[1...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of [3H]-GGPP incorporation into recombinant human Ha-Ras-CVLL by Geranylgeranyl transferase type IMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50134310(9-Methoxy-2-methyl-2,3,10,10a-tetrahydro-pyrazino[...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of [3H]FPP incorporation into recombinant human Ha-Ras-CVLS by farnesyl transferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50134311(3-Benzyldisulfanyl-9-methoxy-2-methyl-2,3-dihydro-...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of [3H]FPP incorporation into recombinant human Ha-Ras-CVLS by farnesyl transferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50134312(Thioacetic acid S-(9-methoxy-2-methyl-1,4-dioxo-1,...)
Affinity DataIC50: 7.48E+5nMAssay Description:Inhibition of [3H]FPP incorporation into recombinant human Ha-Ras-CVLS by farnesyl transferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed