Compile Data Set for Download or QSAR
Report error Found 43 Enz. Inhib. hit(s) with all data for entry = 50013709
TargetCruzipain(Trypanosoma cruzi)
University of Cape Town

Curated by ChEMBL
LigandPNGBDBM50133630((3Z)-5-iodo-1H-indole-2,3-dione 3-thiosemicarbazon...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibitory activity against Trypanosoma brucei rhodesiense cysteine protease rhodesainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCruzipain(Trypanosoma cruzi)
University of Cape Town

Curated by ChEMBL
LigandPNGBDBM50133632(1-(3-Methoxy-benzyl)-5-methyl-1H-indole-2,3-dione ...)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibitory activity against the Trypanosoma cruzi cysteine protease cruzainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCruzipain(Trypanosoma cruzi)
University of Cape Town

Curated by ChEMBL
LigandPNGBDBM50133620(1-Biphenyl-2-ylmethyl-5-methyl-1H-indole-2,3-dione...)
Affinity DataIC50: 2.80E+3nMAssay Description:Inhibitory activity against the Trypanosoma cruzi cysteine protease cruzainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFalcipain 2(malaria parasite P. falciparum)
University of Cape Town

Curated by ChEMBL
LigandPNGBDBM50133627((3Z)-5-nitro-1H-indole-2,3-dione 3-thiosemicarbazo...)
Affinity DataIC50: 4.40E+3nMAssay Description:Inhibitory activity against Falcipain-2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCruzipain(Trypanosoma cruzi)
University of Cape Town

Curated by ChEMBL
LigandPNGBDBM50133623((3Z)-5-chloro-1H-indole-2,3-dione 3-thiosemicarbaz...)
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibitory activity against Trypanosoma brucei rhodesiense cysteine protease rhodesainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCruzipain(Trypanosoma cruzi)
University of Cape Town

Curated by ChEMBL
LigandPNGBDBM50133622(5-Chloro-1-(4-chloro-benzyl)-1H-indole-2,3-dione |...)
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibitory activity against the Trypanosoma cruzi cysteine protease cruzainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCruzipain(Trypanosoma cruzi)
University of Cape Town

Curated by ChEMBL
LigandPNGBDBM50133618((3Z)-5-bromo-1H-indole-2,3-dione 3-thiosemicarbazo...)
Affinity DataIC50: 7.00E+3nMAssay Description:Inhibitory activity against Trypanosoma brucei rhodesiense cysteine protease rhodesainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCruzipain(Trypanosoma cruzi)
University of Cape Town

Curated by ChEMBL
LigandPNGBDBM50133615((3Z)-1H-indole-2,3-dione 3-thiosemicarbazone | CHE...)
Affinity DataIC50: 8.00E+3nMAssay Description:Inhibitory activity against the Trypanosoma cruzi cysteine protease cruzainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCruzipain(Trypanosoma cruzi)
University of Cape Town

Curated by ChEMBL
LigandPNGBDBM50133615((3Z)-1H-indole-2,3-dione 3-thiosemicarbazone | CHE...)
Affinity DataIC50: 8.00E+3nMAssay Description:Inhibitory activity against the Trypanosoma cruzi cysteine protease cruzainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCruzipain(Trypanosoma cruzi)
University of Cape Town

Curated by ChEMBL
LigandPNGBDBM50133630((3Z)-5-iodo-1H-indole-2,3-dione 3-thiosemicarbazon...)
Affinity DataIC50: 9.00E+3nMAssay Description:Inhibitory activity against the Trypanosoma cruzi cysteine protease cruzainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFalcipain 2(malaria parasite P. falciparum)
University of Cape Town

Curated by ChEMBL
LigandPNGBDBM50133620(1-Biphenyl-2-ylmethyl-5-methyl-1H-indole-2,3-dione...)
Affinity DataIC50: 9.20E+3nMAssay Description:Inhibitory activity against Falcipain-2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFalcipain 2(malaria parasite P. falciparum)
University of Cape Town

Curated by ChEMBL
LigandPNGBDBM50133619((3Z)-5-chloro-7-methyl-1H-indole-2,3-dione 3-thios...)
Affinity DataIC50: 9.40E+3nMAssay Description:Inhibitory activity against Falcipain-2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCruzipain(Trypanosoma cruzi)
University of Cape Town

Curated by ChEMBL
LigandPNGBDBM50133619((3Z)-5-chloro-7-methyl-1H-indole-2,3-dione 3-thios...)
Affinity DataIC50: 1.05E+4nMAssay Description:Inhibitory activity against the Trypanosoma cruzi cysteine protease cruzainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCruzipain(Trypanosoma cruzi)
University of Cape Town

Curated by ChEMBL
LigandPNGBDBM50133619((3Z)-5-chloro-7-methyl-1H-indole-2,3-dione 3-thios...)
Affinity DataIC50: 1.05E+4nMAssay Description:Inhibitory activity against the Trypanosoma cruzi cysteine protease cruzainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFalcipain 2(malaria parasite P. falciparum)
University of Cape Town

Curated by ChEMBL
LigandPNGBDBM50133626((3Z)-5,7-dimethyl-1H-indole-2,3-dione 3-thiosemica...)
Affinity DataIC50: 1.32E+4nMAssay Description:Inhibitory activity against Falcipain-2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCruzipain(Trypanosoma cruzi)
University of Cape Town

Curated by ChEMBL
LigandPNGBDBM50133628((3Z)-5-methyl-1H-indole-2,3-dione 3-thiosemicarbaz...)
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibitory activity against the Trypanosoma cruzi cysteine protease cruzainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCruzipain(Trypanosoma cruzi)
University of Cape Town

Curated by ChEMBL
LigandPNGBDBM50133624((3Z)-5-fluoro-1H-indole-2,3-dione 3-thiosemicarbaz...)
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibitory activity against Trypanosoma brucei rhodesiense cysteine protease rhodesainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCruzipain(Trypanosoma cruzi)
University of Cape Town

Curated by ChEMBL
LigandPNGBDBM50133631(1-Benzenesulfonyl-1H-indole-2,3-dione | CHEMBL1198...)
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibitory activity against the Trypanosoma cruzi cysteine protease cruzainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCruzipain(Trypanosoma cruzi)
University of Cape Town

Curated by ChEMBL
LigandPNGBDBM50133626((3Z)-5,7-dimethyl-1H-indole-2,3-dione 3-thiosemica...)
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibitory activity against Trypanosoma brucei rhodesiense cysteine protease rhodesainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCruzipain(Trypanosoma cruzi)
University of Cape Town

Curated by ChEMBL
LigandPNGBDBM50133626((3Z)-5,7-dimethyl-1H-indole-2,3-dione 3-thiosemica...)
Affinity DataIC50: 1.60E+4nMAssay Description:Inhibitory activity against the Trypanosoma cruzi cysteine protease cruzainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCruzipain(Trypanosoma cruzi)
University of Cape Town

Curated by ChEMBL
LigandPNGBDBM50133627((3Z)-5-nitro-1H-indole-2,3-dione 3-thiosemicarbazo...)
Affinity DataIC50: 1.70E+4nMAssay Description:Inhibitory activity against Trypanosoma brucei rhodesiense cysteine protease rhodesainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCruzipain(Trypanosoma cruzi)
University of Cape Town

Curated by ChEMBL
LigandPNGBDBM50133618((3Z)-5-bromo-1H-indole-2,3-dione 3-thiosemicarbazo...)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibitory activity against the Trypanosoma cruzi cysteine protease cruzainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCruzipain(Trypanosoma cruzi)
University of Cape Town

Curated by ChEMBL
LigandPNGBDBM50133623((3Z)-5-chloro-1H-indole-2,3-dione 3-thiosemicarbaz...)
Affinity DataIC50: 2.10E+4nMAssay Description:Inhibitory activity against the Trypanosoma cruzi cysteine protease cruzainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFalcipain 2(malaria parasite P. falciparum)
University of Cape Town

Curated by ChEMBL
LigandPNGBDBM50133632(1-(3-Methoxy-benzyl)-5-methyl-1H-indole-2,3-dione ...)
Affinity DataIC50: 2.19E+4nMAssay Description:Inhibitory activity against Falcipain-2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFalcipain 2(malaria parasite P. falciparum)
University of Cape Town

Curated by ChEMBL
LigandPNGBDBM50133630((3Z)-5-iodo-1H-indole-2,3-dione 3-thiosemicarbazon...)
Affinity DataIC50: 2.87E+4nMAssay Description:Inhibitory activity against Falcipain-2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFalcipain 2(malaria parasite P. falciparum)
University of Cape Town

Curated by ChEMBL
LigandPNGBDBM50133618((3Z)-5-bromo-1H-indole-2,3-dione 3-thiosemicarbazo...)
Affinity DataIC50: 2.96E+4nMAssay Description:Inhibitory activity against Falcipain-2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCruzipain(Trypanosoma cruzi)
University of Cape Town

Curated by ChEMBL
LigandPNGBDBM50133629(2,3-Dioxo-2,3-dihydro-indole-1-carboxylic acid ben...)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibitory activity against the Trypanosoma cruzi cysteine protease cruzainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCruzipain(Trypanosoma cruzi)
University of Cape Town

Curated by ChEMBL
LigandPNGBDBM50133627((3Z)-5-nitro-1H-indole-2,3-dione 3-thiosemicarbazo...)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibitory activity against the Trypanosoma cruzi cysteine protease cruzainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCruzipain(Trypanosoma cruzi)
University of Cape Town

Curated by ChEMBL
LigandPNGBDBM50133624((3Z)-5-fluoro-1H-indole-2,3-dione 3-thiosemicarbaz...)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibitory activity against the Trypanosoma cruzi cysteine protease cruzainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFalcipain 2(malaria parasite P. falciparum)
University of Cape Town

Curated by ChEMBL
LigandPNGBDBM50133622(5-Chloro-1-(4-chloro-benzyl)-1H-indole-2,3-dione |...)
Affinity DataIC50: 3.12E+4nMAssay Description:Inhibitory activity against Falcipain-2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFalcipain 2(malaria parasite P. falciparum)
University of Cape Town

Curated by ChEMBL
LigandPNGBDBM50133623((3Z)-5-chloro-1H-indole-2,3-dione 3-thiosemicarbaz...)
Affinity DataIC50: 3.28E+4nMAssay Description:Inhibitory activity against Falcipain-2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFalcipain 2(malaria parasite P. falciparum)
University of Cape Town

Curated by ChEMBL
LigandPNGBDBM50133634(5-Chloro-1-(3-methoxy-benzyl)-1H-indole-2,3-dione ...)
Affinity DataIC50: 3.46E+4nMAssay Description:Inhibitory activity against Falcipain-2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFalcipain 2(malaria parasite P. falciparum)
University of Cape Town

Curated by ChEMBL
LigandPNGBDBM50133624((3Z)-5-fluoro-1H-indole-2,3-dione 3-thiosemicarbaz...)
Affinity DataIC50: 3.86E+4nMAssay Description:Inhibitory activity against Falcipain-2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFalcipain 2(malaria parasite P. falciparum)
University of Cape Town

Curated by ChEMBL
LigandPNGBDBM50133615((3Z)-1H-indole-2,3-dione 3-thiosemicarbazone | CHE...)
Affinity DataIC50: 3.88E+4nMAssay Description:Inhibitory activity against Falcipain-2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFalcipain 2(malaria parasite P. falciparum)
University of Cape Town

Curated by ChEMBL
LigandPNGBDBM22817(5-nitro-2,3-dihydro-1H-indole-2,3-dione | CHEMBL11...)
Affinity DataIC50: 4.26E+4nMAssay Description:Inhibitory activity against Falcipain-2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFalcipain 2(malaria parasite P. falciparum)
University of Cape Town

Curated by ChEMBL
LigandPNGBDBM50133628((3Z)-5-methyl-1H-indole-2,3-dione 3-thiosemicarbaz...)
Affinity DataIC50: 4.39E+4nMAssay Description:Inhibitory activity against Falcipain-2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFalcipain 2(malaria parasite P. falciparum)
University of Cape Town

Curated by ChEMBL
LigandPNGBDBM50133625(1-Benzyl-5-chloro-1H-indole-2,3-dione | CHEMBL3366...)
Affinity DataIC50: 4.69E+4nMAssay Description:Inhibitory activity against Falcipain-2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCruzipain(Trypanosoma cruzi)
University of Cape Town

Curated by ChEMBL
LigandPNGBDBM50133628((3Z)-5-methyl-1H-indole-2,3-dione 3-thiosemicarbaz...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibitory activity against Cruzain;range is 20-50More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCruzipain(Trypanosoma cruzi)
University of Cape Town

Curated by ChEMBL
LigandPNGBDBM50133621(1-(2,5-Dimethyl-benzyl)-5-methyl-1H-indole-2,3-dio...)
Affinity DataIC50: 8.00E+4nMAssay Description:Inhibitory activity against the Trypanosoma cruzi cysteine protease cruzainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCruzipain(Trypanosoma cruzi)
University of Cape Town

Curated by ChEMBL
LigandPNGBDBM50133633(5-Chloro-2,3-dioxo-2,3-dihydro-indole-1-carboxylic...)
Affinity DataIC50: 8.00E+4nMAssay Description:Inhibitory activity against the Trypanosoma cruzi cysteine protease cruzainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCruzipain(Trypanosoma cruzi)
University of Cape Town

Curated by ChEMBL
LigandPNGBDBM50133617(1-Benzyl-5-iodo-1H-indole-2,3-dione | 1-benzyl-5-i...)
Affinity DataIC50: 9.00E+4nMAssay Description:Inhibitory activity against the Trypanosoma cruzi cysteine protease cruzainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCruzipain(Trypanosoma cruzi)
University of Cape Town

Curated by ChEMBL
LigandPNGBDBM50133625(1-Benzyl-5-chloro-1H-indole-2,3-dione | CHEMBL3366...)
Affinity DataIC50: 9.00E+4nMAssay Description:Inhibitory activity against the Trypanosoma cruzi cysteine protease cruzainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCruzipain(Trypanosoma cruzi)
University of Cape Town

Curated by ChEMBL
LigandPNGBDBM50133616(1-Benzoyl-1H-indole-2,3-dione | CHEMBL118830)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibitory activity against the Trypanosoma cruzi cysteine protease cruzainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed