Compile Data Set for Download or QSAR
Report error Found 15 Enz. Inhib. hit(s) with all data for entry = 50036042
TargetPlatelet-activating factor receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50002827(CHEMBL118105 | 1-{3-(3-Hydroxy-propoxy)-2-propoxy-...)
Affinity DataKi:  1.90nMAssay Description:Inhibition of the binding of [3H]C18-Platelet activating factor to human platelet membrane preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50002828(CHEMBL117413 | 1-{3-(3-Morpholin-4-yl-propoxy)-2-p...)
Affinity DataKi:  2.5nMAssay Description:Inhibition of the binding of [3H]C18-Platelet activating factor to human platelet membrane preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50002827(CHEMBL118105 | 1-{3-(3-Hydroxy-propoxy)-2-propoxy-...)
Affinity DataKi:  2.90nMAssay Description:In vitro effect on inhibition of the binding of [3H]C18-Platelet activating factor to human PMN membranes preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50002824(CHEMBL334115 | (S)-5-{3-Methoxy-2-propoxy-5-[(2S,5...)
Affinity DataKi:  2.90nMAssay Description:Inhibition of the binding of [3H]C18-Platelet activating factor to human platelet membrane preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50002826(CHEMBL407427 | 1-{3-(3-Imidazol-1-yl-propoxy)-2-pr...)
Affinity DataKi:  3nMAssay Description:Inhibition of the binding of [3H]C18-Platelet activating factor to human platelet membrane preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50002823(CHEMBL299944 | 2-{3-Methoxy-2-propoxy-5-[(2S,5S)-5...)
Affinity DataKi:  3.20nMAssay Description:In vitro effect on inhibition of the binding of [3H]C18-Platelet activating factor to human PMN membranes preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50002825(CHEMBL116072 | (R)-5-{3-Methoxy-2-propoxy-5-[(2S,5...)
Affinity DataKi:  3.70nMAssay Description:Inhibition of the binding of [3H]C18-Platelet activating factor to human platelet membrane preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50002824(CHEMBL334115 | (S)-5-{3-Methoxy-2-propoxy-5-[(2S,5...)
Affinity DataKi:  3.70nMAssay Description:In vitro effect on inhibition of the binding of [3H]C18-Platelet activating factor to human PMN membranes preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50002825(CHEMBL116072 | (R)-5-{3-Methoxy-2-propoxy-5-[(2S,5...)
Affinity DataKi:  3.72nMAssay Description:Inhibition of the binding of [3H]C18-Platelet activating factor to human platelet membrane preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50002823(CHEMBL299944 | 2-{3-Methoxy-2-propoxy-5-[(2S,5S)-5...)
Affinity DataKi:  6.30nMAssay Description:Inhibition of the binding of [3H]C18-Platelet activating factor to human platelet membrane preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM81972(CAS_75614-93-6 | (S)-(+)-ALPHA-METHYL-1H-IMIDAZOLE...)
Affinity DataKi:  9nMAssay Description:Inhibition of the binding of [3H]C18-Platelet activating factor to human platelet membrane preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50366241(L-652731 | CHEMBL297624)
Affinity DataKi:  103nMAssay Description:Inhibition of the binding of [3H]C18-Platelet activating factor to human platelet membrane preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50002822(CHEMBL325491 | (-)-trans 42s,5S)-2-[3-[(2-Oxopropy...)
Affinity DataKi:  110nMAssay Description:Inhibition of the binding of [3H]C18-Platelet activating factor to human platelet membrane preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50002822(CHEMBL325491 | (-)-trans 42s,5S)-2-[3-[(2-Oxopropy...)
Affinity DataKi:  174nMAssay Description:In vitro effect on inhibition of the binding of [3H]C18-Platelet activating factor to human PMN membranes preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50002830(CHEMBL112481 | (2R,3R,4R,5S)-2,5-Bis-(3,4-dimethox...)
Affinity DataKi:  1.00E+3nMAssay Description:Inhibition of the binding of [3H]C18-Platelet activating factor to human platelet membrane preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed