Compile Data Set for Download or QSAR
Report error Found 40 Enz. Inhib. hit(s) with all data for entry = 50000158
TargetD(2) dopamine receptor(Rat)
E. Merck Darmstadt

Curated by ChEMBL
LigandPNGBDBM50002173(CHEMBL431367 | roxindole | 3-(4-(3,6-dihydro-4-phe...)
Affinity DataIC50: 6nMAssay Description:Compound was evaluated for its ability to displace tritiated receptor ligand in rat striatal membranes 3[H]spiperone, a dopamine antagonistMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
E. Merck Darmstadt

Curated by ChEMBL
LigandPNGBDBM50002169(CHEMBL130502 | 3-[4-(4-Phenyl-3,6-dihydro-2H-pyrid...)
Affinity DataIC50: 8nMAssay Description:Evaluated for its ability to displace tritiated receptor ligand in rat striatal membranes 3[H]spiperone, a dopamine antagonistMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
E. Merck Darmstadt

Curated by ChEMBL
LigandPNGBDBM50002175(CHEMBL130659 | 6-Methoxy-3-[4-(4-phenyl-3,6-dihydr...)
Affinity DataIC50: 9nMAssay Description:Evaluated for its ability to displace tritiated receptor ligand in rat striatal membranes 3[H]spiperone, a dopamine antagonistMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
E. Merck Darmstadt

Curated by ChEMBL
LigandPNGBDBM50002158(CHEMBL338710 | 5-Fluoro-3-[4-(4-phenyl-3,6-dihydro...)
Affinity DataIC50: 10nMAssay Description:Evaluated for its ability to displace tritiated receptor ligand in rat striatal membranes 3[H]spiperone, a dopamine antagonistMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
E. Merck Darmstadt

Curated by ChEMBL
LigandPNGBDBM50002177(CHEMBL130327 | 5-Methoxy-3-[4-(4-phenyl-3,6-dihydr...)
Affinity DataIC50: 20nMAssay Description:Evaluated for its ability to displace tritiated receptor ligand in rat striatal membranes 3[H]spiperone, a dopamine antagonistMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
E. Merck Darmstadt

Curated by ChEMBL
LigandPNGBDBM50002174(CHEMBL132270 | 3-{4-[4-(2-Fluoro-phenyl)-3,6-dihyd...)
Affinity DataIC50: 20nMAssay Description:Evaluated for its ability to displace tritiated receptor ligand in rat striatal membranes 3[H]spiperone, a dopamine antagonistMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
E. Merck Darmstadt

Curated by ChEMBL
LigandPNGBDBM50002176(CHEMBL130614 | 3-[6-(4-Phenyl-3,6-dihydro-2H-pyrid...)
Affinity DataIC50: 40nMAssay Description:Evaluated for its ability to displace tritiated receptor ligand in rat striatal membranes 3[H]spiperone, a dopamine antagonistMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
E. Merck Darmstadt

Curated by ChEMBL
LigandPNGBDBM50002170(CHEMBL131841 | 3-[3-(4-Phenyl-3,6-dihydro-2H-pyrid...)
Affinity DataIC50: 50nMAssay Description:Evaluated for its ability to displace tritiated receptor ligand in rat striatal membranes 3[H]spiperone, a dopamine antagonistMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
E. Merck Darmstadt

Curated by ChEMBL
LigandPNGBDBM50002162(CHEMBL338849 | 2-Methyl-3-[4-(4-phenyl-3,6-dihydro...)
Affinity DataIC50: 50nMAssay Description:Evaluated for its ability to displace tritiated receptor ligand in rat striatal membranes 3[H]spiperone, a dopamine antagonistMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
E. Merck Darmstadt

Curated by ChEMBL
LigandPNGBDBM50002160(CHEMBL132446 | 5-Chloro-3-[4-(4-phenyl-3,6-dihydro...)
Affinity DataIC50: 50nMAssay Description:Evaluated for its ability to displace tritiated receptor ligand in rat striatal membranes 3[H]spiperone, a dopamine antagonistMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
E. Merck Darmstadt

Curated by ChEMBL
LigandPNGBDBM50002167(CHEMBL419957 | 3-[5-(4-Phenyl-3,6-dihydro-2H-pyrid...)
Affinity DataIC50: 60nMAssay Description:Evaluated for its ability to displace tritiated receptor ligand in rat striatal membranes 3[H]spiperone, a dopamine antagonistMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
E. Merck Darmstadt

Curated by ChEMBL
LigandPNGBDBM50002171(CHEMBL64344 | 3-{4-[4-(4-Fluoro-phenyl)-3,6-dihydr...)
Affinity DataIC50: 90nMAssay Description:Evaluated for its ability to displace tritiated receptor ligand in rat striatal membranes 3[H]spiperone, a dopamine antagonistMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
E. Merck Darmstadt

Curated by ChEMBL
LigandPNGBDBM50002164(CHEMBL59335 | 3-[4-(4-Phenyl-piperidin-1-yl)-butyl...)
Affinity DataIC50: 100nMAssay Description:Evaluated for its ability to displace tritiated receptor ligand in rat striatal membranes 3[H]spiperone, a dopamine antagonistMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
E. Merck Darmstadt

Curated by ChEMBL
LigandPNGBDBM50002166(CHEMBL130501 | 3-{4-[4-(4-Chloro-phenyl)-3,6-dihyd...)
Affinity DataIC50: 100nMAssay Description:Evaluated for its ability to displace tritiated receptor ligand in rat striatal membranes 3[H]spiperone, a dopamine antagonistMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
E. Merck Darmstadt

Curated by ChEMBL
LigandPNGBDBM50002159(CHEMBL131356 | 1-Methyl-3-[4-(4-phenyl-3,6-dihydro...)
Affinity DataIC50: 100nMAssay Description:Evaluated for its ability to displace tritiated receptor ligand in rat striatal membranes 3[H]spiperone, a dopamine antagonistMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
E. Merck Darmstadt

Curated by ChEMBL
LigandPNGBDBM50002165(CHEMBL131711 | 3-{4-[4-(2-Chloro-phenyl)-3,6-dihyd...)
Affinity DataIC50: 100nMAssay Description:Evaluated for its ability to displace tritiated receptor ligand in rat striatal membranes 3[H]spiperone, a dopamine antagonistMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
E. Merck Darmstadt

Curated by ChEMBL
LigandPNGBDBM50002163(CHEMBL127609 | 3-[2-(4-Phenyl-3,6-dihydro-2H-pyrid...)
Affinity DataIC50: 100nMAssay Description:Evaluated for its ability to displace tritiated receptor ligand in rat striatal membranes 3[H]spiperone, a dopamine antagonistMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
E. Merck Darmstadt

Curated by ChEMBL
LigandPNGBDBM50002172(CHEMBL44231 | 3-[4-(4-Phenyl-3,6-dihydro-2H-pyridi...)
Affinity DataIC50: 105nMAssay Description:Compound was evaluated for its ability to displace tritiated receptor ligand in rat striatal membranes [3H]ADTN, a dopamine agonistMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
E. Merck Darmstadt

Curated by ChEMBL
LigandPNGBDBM50002168(CHEMBL339954 | 3-{4-[4-(4-Methoxy-phenyl)-3,6-dihy...)
Affinity DataIC50: 700nMAssay Description:Evaluated for its ability to displace tritiated receptor ligand in rat striatal membranes 3[H]spiperone, a dopamine antagonistMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
E. Merck Darmstadt

Curated by ChEMBL
LigandPNGBDBM50002161(CHEMBL130605 | 3-[4-(3,6-Dihydro-2H-pyridin-1-yl)-...)
Affinity DataIC50: 1.00E+3nMAssay Description:Evaluated for its ability to displace tritiated receptor ligand in rat striatal membranes 3[H]spiperone, a dopamine antagonistMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
E. Merck Darmstadt

Curated by ChEMBL
LigandPNGBDBM50002173(CHEMBL431367 | roxindole | 3-(4-(3,6-dihydro-4-phe...)
Affinity DataKi:  0.880nMAssay Description:Evaluated for its ability to displace tritiated receptor ligand in rat striatal membranes [3H]ADTN, a dopamine agonistMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
E. Merck Darmstadt

Curated by ChEMBL
LigandPNGBDBM50002158(CHEMBL338710 | 5-Fluoro-3-[4-(4-phenyl-3,6-dihydro...)
Affinity DataKi:  1.60nMAssay Description:Evaluated for its ability to displace tritiated receptor ligand in rat striatal membranes [3H]ADTN, a dopamine agonistMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
E. Merck Darmstadt

Curated by ChEMBL
LigandPNGBDBM50002175(CHEMBL130659 | 6-Methoxy-3-[4-(4-phenyl-3,6-dihydr...)
Affinity DataKi:  1.80nMAssay Description:Evaluated for its ability to displace tritiated receptor ligand in rat striatal membranes [3H]ADTN, a dopamine agonistMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
E. Merck Darmstadt

Curated by ChEMBL
LigandPNGBDBM50002169(CHEMBL130502 | 3-[4-(4-Phenyl-3,6-dihydro-2H-pyrid...)
Affinity DataKi:  2.5nMAssay Description:Evaluated for its ability to displace tritiated receptor ligand in rat striatal membranes [3H]ADTN, a dopamine agonistMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
E. Merck Darmstadt

Curated by ChEMBL
LigandPNGBDBM50002160(CHEMBL132446 | 5-Chloro-3-[4-(4-phenyl-3,6-dihydro...)
Affinity DataKi:  3.10nMAssay Description:Evaluated for its ability to displace tritiated receptor ligand in rat striatal membranes [3H]ADTN, a dopamine agonistMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
E. Merck Darmstadt

Curated by ChEMBL
LigandPNGBDBM50002174(CHEMBL132270 | 3-{4-[4-(2-Fluoro-phenyl)-3,6-dihyd...)
Affinity DataKi:  4nMAssay Description:Evaluated for its ability to displace tritiated receptor ligand in rat striatal membranes [3H]ADTN, a dopamine agonistMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
E. Merck Darmstadt

Curated by ChEMBL
LigandPNGBDBM50002176(CHEMBL130614 | 3-[6-(4-Phenyl-3,6-dihydro-2H-pyrid...)
Affinity DataKi:  4.30nMAssay Description:Evaluated for its ability to displace tritiated receptor ligand in rat striatal membranes [3H]ADTN, a dopamine agonistMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
E. Merck Darmstadt

Curated by ChEMBL
LigandPNGBDBM50002177(CHEMBL130327 | 5-Methoxy-3-[4-(4-phenyl-3,6-dihydr...)
Affinity DataKi:  4.40nMAssay Description:Evaluated for its ability to displace tritiated receptor ligand in rat striatal membranes [3H]ADTN, a dopamine agonistMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
E. Merck Darmstadt

Curated by ChEMBL
LigandPNGBDBM50002162(CHEMBL338849 | 2-Methyl-3-[4-(4-phenyl-3,6-dihydro...)
Affinity DataKi:  5.40nMAssay Description:Evaluated for its ability to displace tritiated receptor ligand in rat striatal membranes [3H]ADTN, a dopamine agonistMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
E. Merck Darmstadt

Curated by ChEMBL
LigandPNGBDBM50002172(CHEMBL44231 | 3-[4-(4-Phenyl-3,6-dihydro-2H-pyridi...)
Affinity DataKi:  6.40nMAssay Description:Compound was evaluated for its ability to displace tritiated receptor ligand in rat striatal membranes [3H]ADTN, a dopamine agonistMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
E. Merck Darmstadt

Curated by ChEMBL
LigandPNGBDBM50002170(CHEMBL131841 | 3-[3-(4-Phenyl-3,6-dihydro-2H-pyrid...)
Affinity DataKi:  12nMAssay Description:Evaluated for its ability to displace tritiated receptor ligand in rat striatal membranes [3H]ADTN, a dopamine agonistMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
E. Merck Darmstadt

Curated by ChEMBL
LigandPNGBDBM50002167(CHEMBL419957 | 3-[5-(4-Phenyl-3,6-dihydro-2H-pyrid...)
Affinity DataKi:  13nMAssay Description:Evaluated for its ability to displace tritiated receptor ligand in rat striatal membranes [3H]ADTN, a dopamine agonistMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
E. Merck Darmstadt

Curated by ChEMBL
LigandPNGBDBM50002159(CHEMBL131356 | 1-Methyl-3-[4-(4-phenyl-3,6-dihydro...)
Affinity DataKi:  15nMAssay Description:Evaluated for its ability to displace tritiated receptor ligand in rat striatal membranes [3H]ADTN, a dopamine agonistMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
E. Merck Darmstadt

Curated by ChEMBL
LigandPNGBDBM50002171(CHEMBL64344 | 3-{4-[4-(4-Fluoro-phenyl)-3,6-dihydr...)
Affinity DataKi:  15nMAssay Description:Evaluated for its ability to displace tritiated receptor ligand in rat striatal membranes [3H]ADTN, a dopamine agonistMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
E. Merck Darmstadt

Curated by ChEMBL
LigandPNGBDBM50002165(CHEMBL131711 | 3-{4-[4-(2-Chloro-phenyl)-3,6-dihyd...)
Affinity DataKi:  21nMAssay Description:Evaluated for its ability to displace tritiated receptor ligand in rat striatal membranes [3H]ADTN, a dopamine agonistMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
E. Merck Darmstadt

Curated by ChEMBL
LigandPNGBDBM50002168(CHEMBL339954 | 3-{4-[4-(4-Methoxy-phenyl)-3,6-dihy...)
Affinity DataKi:  41nMAssay Description:Evaluated for its ability to displace tritiated receptor ligand in rat striatal membranes [3H]ADTN, a dopamine agonistMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
E. Merck Darmstadt

Curated by ChEMBL
LigandPNGBDBM50002166(CHEMBL130501 | 3-{4-[4-(4-Chloro-phenyl)-3,6-dihyd...)
Affinity DataKi:  46nMAssay Description:Evaluated for its ability to displace tritiated receptor ligand in rat striatal membranes [3H]ADTN, a dopamine agonistMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
E. Merck Darmstadt

Curated by ChEMBL
LigandPNGBDBM50002163(CHEMBL127609 | 3-[2-(4-Phenyl-3,6-dihydro-2H-pyrid...)
Affinity DataKi:  81nMAssay Description:Evaluated for its ability to displace tritiated receptor ligand in rat striatal membranes [3H]ADTN, a dopamine agonistMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
E. Merck Darmstadt

Curated by ChEMBL
LigandPNGBDBM50002164(CHEMBL59335 | 3-[4-(4-Phenyl-piperidin-1-yl)-butyl...)
Affinity DataKi: >100nMAssay Description:Evaluated for its ability to displace tritiated receptor ligand in rat striatal membranes [3H]ADTN, a dopamine agonistMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
E. Merck Darmstadt

Curated by ChEMBL
LigandPNGBDBM50002161(CHEMBL130605 | 3-[4-(3,6-Dihydro-2H-pyridin-1-yl)-...)
Affinity DataKi: >1.00E+3nMAssay Description:Evaluated for its ability to displace tritiated receptor ligand in rat striatal membranes [3H]ADTN, a dopamine agonistMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed