Compile Data Set for Download or QSAR
Report error Found 23 Enz. Inhib. hit(s) with all data for entry = 50013599
TargetDNA-dependent protein kinase catalytic subunit(Human)
University of Newcastle

Curated by ChEMBL
LigandPNGBDBM50132355(2-(4-Chloro-phenyl)-6-morpholin-4-yl-pyran-4-one |...)
Affinity DataIC50: 180nMAssay Description:In vitro inhibition of DNA-dependent protein kinase(DNA-PK) from HeLa (human carcinoma) cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDNA-dependent protein kinase catalytic subunit(Human)
University of Newcastle

Curated by ChEMBL
LigandPNGBDBM50132371(2-morpholino-6-(4-(naphthalen-1-yl)phenyl)-4H-thio...)
Affinity DataIC50: 190nMAssay Description:In vitro inhibition of DNA-dependent protein kinase(DNA-PK) from HeLa (human carcinoma) cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDNA-dependent protein kinase catalytic subunit(Human)
University of Newcastle

Curated by ChEMBL
LigandPNGBDBM50132361(2-(4-methoxyphenyl)-6-morpholino-4H-pyran-4-one | ...)
Affinity DataIC50: 220nMAssay Description:In vitro inhibition of DNA-dependent protein kinase(DNA-PK) from HeLa (human carcinoma) cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDNA-dependent protein kinase catalytic subunit(Human)
University of Newcastle

Curated by ChEMBL
LigandPNGBDBM50098126(LY-293646 | 2-morpholino-4H-benzo[h]chromen-4-one ...)
Affinity DataIC50: 230nMAssay Description:In vitro inhibition of DNA-dependent protein kinase(DNA-PK) from HeLa (human carcinoma) cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDNA-dependent protein kinase catalytic subunit(Human)
University of Newcastle

Curated by ChEMBL
LigandPNGBDBM50132368(6-(4-(4-methylnaphthalen-1-yl)phenyl)-2-morpholin-...)
Affinity DataIC50: 260nMAssay Description:In vitro inhibition of DNA-dependent protein kinase(DNA-PK) from HeLa (human carcinoma) cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDNA-dependent protein kinase catalytic subunit(Human)
University of Newcastle

Curated by ChEMBL
LigandPNGBDBM50132365(6-(4-methoxyphenyl)-2-morpholin-4-yl-4H-thiopyran-...)
Affinity DataIC50: 280nMAssay Description:In vitro inhibition of DNA-dependent protein kinase(DNA-PK) from HeLa (human carcinoma) cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDNA-dependent protein kinase catalytic subunit(Human)
University of Newcastle

Curated by ChEMBL
LigandPNGBDBM50132373(2-(4-(benzo[b]thiophen-3-yl)phenyl)-6-morpholino-4...)
Affinity DataIC50: 330nMAssay Description:In vitro inhibition of DNA-dependent protein kinase(DNA-PK) from HeLa (human carcinoma) cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDNA-dependent protein kinase catalytic subunit(Human)
University of Newcastle

Curated by ChEMBL
LigandPNGBDBM50132370(2-(4-fluorophenyl)-6-morpholino-4H-pyran-4-one | 2...)
Affinity DataIC50: 350nMAssay Description:In vitro inhibition of DNA-dependent protein kinase(DNA-PK) from HeLa (human carcinoma) cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDNA-dependent protein kinase catalytic subunit(Human)
University of Newcastle

Curated by ChEMBL
LigandPNGBDBM50132366(2-(4'-Hydroxy-biphenyl-3-yl)-6-morpholin-4-yl-thio...)
Affinity DataIC50: 350nMAssay Description:In vitro inhibition of DNA-dependent protein kinase(DNA-PK) from HeLa (human carcinoma) cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDNA-dependent protein kinase catalytic subunit(Human)
University of Newcastle

Curated by ChEMBL
LigandPNGBDBM50132363(2-(2-methoxyphenyl)-6-morpholino-4H-pyran-4-one | ...)
Affinity DataIC50: 380nMAssay Description:In vitro inhibition of DNA-dependent protein kinase(DNA-PK) from HeLa (human carcinoma) cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDNA-dependent protein kinase catalytic subunit(Human)
University of Newcastle

Curated by ChEMBL
LigandPNGBDBM50132358(6-(4-t-butylphenyl)-2-(4-morpholin-4-yl)pyran-4-on...)
Affinity DataIC50: 480nMAssay Description:In vitro inhibition of DNA-dependent protein kinase(DNA-PK) from HeLa (human carcinoma) cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDNA-dependent protein kinase catalytic subunit(Human)
University of Newcastle

Curated by ChEMBL
LigandPNGBDBM50132360(6-(3-fluorophenyl)-2-(4-morpholin-4-yl)pyran-4-one...)
Affinity DataIC50: 530nMAssay Description:In vitro inhibition of DNA-dependent protein kinase(DNA-PK) from HeLa (human carcinoma) cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDNA-dependent protein kinase catalytic subunit(Human)
University of Newcastle

Curated by ChEMBL
LigandPNGBDBM50132369(6-(4-chlorophenyl)-2-morpholin-4-yl-4H-thiopyran-4...)
Affinity DataIC50: 530nMAssay Description:In vitro inhibition of DNA-dependent protein kinase(DNA-PK) from HeLa (human carcinoma) cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDNA-dependent protein kinase catalytic subunit(Human)
University of Newcastle

Curated by ChEMBL
LigandPNGBDBM50132356(2-(3-methoxyphenyl)-6-morpholino-4H-pyran-4-one | ...)
Affinity DataIC50: 540nMAssay Description:In vitro inhibition of DNA-dependent protein kinase(DNA-PK) from HeLa (human carcinoma) cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDNA-dependent protein kinase catalytic subunit(Human)
University of Newcastle

Curated by ChEMBL
LigandPNGBDBM50132367(6-(4-bromophenyl)-2-morpholin-4-yl-4H-thiopyran-4-...)
Affinity DataIC50: 680nMAssay Description:In vitro inhibition of DNA-dependent protein kinase(DNA-PK) from HeLa (human carcinoma) cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDNA-dependent protein kinase catalytic subunit(Human)
University of Newcastle

Curated by ChEMBL
LigandPNGBDBM50132364(2-morpholin-4-yl-6-phenyl-4H-thiopyran-4-one | 2-M...)
Affinity DataIC50: 720nMAssay Description:In vitro inhibition of DNA-dependent protein kinase(DNA-PK) from HeLa (human carcinoma) cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDNA-dependent protein kinase catalytic subunit(Human)
University of Newcastle

Curated by ChEMBL
LigandPNGBDBM50132354(2-(3-Bromo-phenyl)-6-morpholin-4-yl-thiopyran-4-on...)
Affinity DataIC50: 800nMAssay Description:In vitro inhibition of DNA-dependent protein kinase(DNA-PK) from HeLa (human carcinoma) cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDNA-dependent protein kinase catalytic subunit(Human)
University of Newcastle

Curated by ChEMBL
LigandPNGBDBM50132357((E)-3-[3'-(6-Morpholin-4-yl-4-oxo-4H-thiopyran-2-y...)
Affinity DataIC50: 840nMAssay Description:In vitro inhibition of DNA-dependent protein kinase(DNA-PK) from HeLa (human carcinoma) cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDNA-dependent protein kinase catalytic subunit(Human)
University of Newcastle

Curated by ChEMBL
LigandPNGBDBM50132362(2-(3'-hydroxy-biphenyl-3-yl)-6-morpholin-4-yl-thio...)
Affinity DataIC50: 920nMAssay Description:In vitro inhibition of DNA-dependent protein kinase(DNA-PK) from HeLa (human carcinoma) cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDNA-dependent protein kinase catalytic subunit(Human)
University of Newcastle

Curated by ChEMBL
LigandPNGBDBM50132372(6-(4-t-butylphenyl)-2-morpholin-4-yl-4H-thiopyran-...)
Affinity DataIC50: 920nMAssay Description:In vitro inhibition of DNA-dependent protein kinase(DNA-PK) from HeLa (human carcinoma) cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDNA-dependent protein kinase catalytic subunit(Human)
University of Newcastle

Curated by ChEMBL
LigandPNGBDBM50132359(2-morpholino-6-phenyl-4H-pyran-4-one | 2-Morpholin...)
Affinity DataIC50: 1.10E+3nMAssay Description:In vitro inhibition of DNA-dependent protein kinase(DNA-PK) from HeLa (human carcinoma) cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDNA-dependent protein kinase catalytic subunit(Human)
University of Newcastle

Curated by ChEMBL
LigandPNGBDBM12915(CHEMBL98350 | 2-(morpholin-4-yl)-8-phenyl-4H-chrom...)
Affinity DataIC50: 1.40E+3nMAssay Description:In vitro inhibition of DNA-dependent protein kinase(DNA-PK) from HeLa (human carcinoma) cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDNA-dependent protein kinase catalytic subunit(Human)
University of Newcastle

Curated by ChEMBL
LigandPNGBDBM12915(CHEMBL98350 | 2-(morpholin-4-yl)-8-phenyl-4H-chrom...)
Affinity DataKi:  6.00E+3nMAssay Description:Affinity for DNA-dependent protein kinase(DNA-PK) from HeLa cell extractMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed