Compile Data Set for Download or QSAR
Report error Found 5 Enz. Inhib. hit(s) with all data for entry = 50013559
TargetCholine kinase alpha(Human)
Universidad De Granada

Curated by ChEMBL
LigandPNGBDBM50131885(4,8-diaza-3 (1,4) , 9 (4,1)-dipyridina-1 (1,4), 6 ...)
Affinity DataIC50: 300nMAssay Description:Ex vivo inhibitory activity against human choline kinase was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholine kinase alpha(Human)
Universidad De Granada

Curated by ChEMBL
LigandPNGBDBM50131887(1-(3,5-Bis-{4-[(4-chloro-phenyl)-methyl-amino]-pyr...)
Affinity DataIC50: 1.40E+3nMAssay Description:Ex vivo inhibitory activity against human choline kinase was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholine kinase alpha(Human)
Universidad De Granada

Curated by ChEMBL
LigandPNGBDBM50131884(Bis-pyridinium cyclophane | CHEMBL125434)
Affinity DataIC50: 2.10E+3nMAssay Description:Ex vivo inhibitory activity against human choline kinase was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholine kinase alpha(Human)
Universidad De Granada

Curated by ChEMBL
LigandPNGBDBM50131886(Bis-pyridinium cyclophane | CHEMBL121973)
Affinity DataIC50: 1.32E+4nMAssay Description:Ex vivo inhibitory activity against human choline kinase was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholine kinase alpha(Human)
Universidad De Granada

Curated by ChEMBL
LigandPNGBDBM50131883(Bis-pyridinium cyclophane | CHEMBL341537)
Affinity DataIC50: 2.48E+4nMAssay Description:Ex vivo inhibitory activity against human choline kinase was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed