Compile Data Set for Download or QSAR
Report error Found 284 Enz. Inhib. hit(s) with all data for entry = 866
LigandChemical structure of BindingDB Monomer ID 6811BDBM6811(18,23-dimethyl-3,13,18-triazahexacyclo[14.7.0.0^{2...)
Affinity DataIC50: 2nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 6832BDBM6832(3-[3-(4-hydroxypiperidin-1-yl)propyl]-6-methoxy-18...)
Affinity DataIC50: 4nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 6846BDBM6846(5-{2-[(4-hydroxycyclohexyl)amino]ethyl}-18-methyl-...)
Affinity DataIC50: 5nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 6838BDBM6838(1-(2-{18-methyl-12,14-dioxo-3,13,18-triazahexacycl...)
Affinity DataIC50: 5nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 6800BDBM6800(6-hydroxy-3,13,18-triazahexacyclo[14.7.0.0^{2,10}....)
Affinity DataIC50: 6nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 6803BDBM6803(6-methoxy-18-methyl-3,13,18-triazahexacyclo[14.7.0...)
Affinity DataIC50: 6nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 6815BDBM6815(6-fluoro-18,23-dimethyl-3,13,18-triazahexacyclo[14...)
Affinity DataIC50: 6nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 6816BDBM6816(6-methoxy-18,23-dimethyl-3,13,18-triazahexacyclo[1...)
Affinity DataIC50: 7nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 6840BDBM6840(5-[2-(4-hydroxypiperidin-1-yl)ethyl]-18-methyl-3,1...)
Affinity DataIC50: 8nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 6818BDBM6818(3-(3-hydroxypropyl)-3,13,18-triazahexacyclo[14.7.0...)
Affinity DataIC50: 8nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 6794BDBM6794(6-fluoro-18-methyl-3,13,18-triazahexacyclo[14.7.0....)
Affinity DataIC50: 9nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 6796BDBM6796(18-methyl-6-(trifluoromethyl)-3,13,18-triazahexacy...)
Affinity DataIC50: 9nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 6801BDBM6801(6-hydroxy-18-methyl-3,13,18-triazahexacyclo[14.7.0...)
Affinity DataIC50: 9nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 6804BDBM6804(6-ethoxy-18-methyl-3,13,18-triazahexacyclo[14.7.0....)
Affinity DataIC50: 10nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 6843BDBM6843(5-{2-[(2-hydroxyethyl)amino]ethyl}-18-methyl-3,13,...)
Affinity DataIC50: 10nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 6797BDBM6797(18-methyl-12,14-dioxo-3,13,18-triazahexacyclo[14.7...)
Affinity DataIC50: 10nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 6842BDBM6842(18-methyl-5-[2-(piperidin-1-yl)ethyl]-3,13,18-tria...)
Affinity DataIC50: 11nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 6794BDBM6794(6-fluoro-18-methyl-3,13,18-triazahexacyclo[14.7.0....)
Affinity DataIC50: 11nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 6797BDBM6797(18-methyl-12,14-dioxo-3,13,18-triazahexacyclo[14.7...)
Affinity DataIC50: 11nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 6822BDBM6822(3-(3-hydroxypropyl)-6-methoxy-18-methyl-3,13,18-tr...)
Affinity DataIC50: 12nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 6818BDBM6818(3-(3-hydroxypropyl)-3,13,18-triazahexacyclo[14.7.0...)
Affinity DataIC50: 12nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 6831BDBM6831(1-(3-{6-methoxy-18-methyl-12,14-dioxo-3,13,18-tria...)
Affinity DataIC50: 13nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 6795BDBM6795(6-bromo-18-methyl-3,13,18-triazahexacyclo[14.7.0.0...)
Affinity DataIC50: 13nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 6837BDBM6837(methyl 1-(2-{18-methyl-12,14-dioxo-3,13,18-triazah...)
Affinity DataIC50: 13nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 6833BDBM6833(6-methoxy-18-methyl-3-[3-(4-methylpiperazin-1-yl)p...)
Affinity DataIC50: 14nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 6839BDBM6839(18-methyl-5-[2-(piperazin-1-yl)ethyl]-3,13,18-tria...)
Affinity DataIC50: 15nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 6844BDBM6844(18-methyl-5-[2-(morpholin-4-yl)ethyl]-3,13,18-tria...)
Affinity DataIC50: 15nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 6812BDBM6812(23-fluoro-18-methyl-3,13,18-triazahexacyclo[14.7.0...)
Affinity DataIC50: 16nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 6800BDBM6800(6-hydroxy-3,13,18-triazahexacyclo[14.7.0.0^{2,10}....)
Affinity DataIC50: 17nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 6813BDBM6813(23-methoxy-18-methyl-3,13,18-triazahexacyclo[14.7....)
Affinity DataIC50: 18nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 6798BDBM6798(6,18-dimethyl-3,13,18-triazahexacyclo[14.7.0.0^{2,...)
Affinity DataIC50: 18nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 6784BDBM6784(18-ethyl-3,13,18-triazahexacyclo[14.7.0.0^{2,10}.0...)
Affinity DataIC50: 19nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 6848BDBM6848(5-{3-[(2-hydroxyethyl)amino]propyl}-18-methyl-3,13...)
Affinity DataIC50: 19nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 6851BDBM6851(5-{3-[(4-hydroxycyclohexyl)amino]propyl}-18-methyl...)
Affinity DataIC50: 19nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 6829BDBM6829(3-{2-[(2-hydroxyethyl)amino]ethyl}-6-methoxy-18-me...)
Affinity DataIC50: 21nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 6835BDBM6835(6-methoxy-18-methyl-3-[3-(morpholin-4-yl)propyl]-3...)
Affinity DataIC50: 21nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 6799BDBM6799(6-ethyl-18-methyl-3,13,18-triazahexacyclo[14.7.0.0...)
Affinity DataIC50: 22nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 6782BDBM6782(3,13,18-triazahexacyclo[14.7.0.0^{2,10}.0^{4,9}.0^...)
Affinity DataIC50: 22nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 6783BDBM6783(18-methyl-3,13,18-triazahexacyclo[14.7.0.0^{2,10}....)
Affinity DataIC50: 22nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 6841BDBM6841(5-{2-[(2S)-2-(hydroxymethyl)pyrrolidin-1-yl]ethyl}...)
Affinity DataIC50: 23nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 6827BDBM6827(3-{2-[(2S)-2-(hydroxymethyl)pyrrolidin-1-yl]ethyl}...)
Affinity DataIC50: 23nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 6830BDBM6830(3-{2-[(4-hydroxycyclohexyl)amino]ethyl}-6-methoxy-...)
Affinity DataIC50: 23nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 6815BDBM6815(6-fluoro-18,23-dimethyl-3,13,18-triazahexacyclo[14...)
Affinity DataIC50: 23nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 6821BDBM6821(3-(2-hydroxyethyl)-6-methoxy-18-methyl-3,13,18-tri...)
Affinity DataIC50: 24nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 6845BDBM6845(18-methyl-5-[2-(thiomorpholin-4-yl)ethyl]-3,13,18-...)
Affinity DataIC50: 24nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 6850BDBM6850(5-[3-(diethylamino)propyl]-18-methyl-3,13,18-triaz...)
Affinity DataIC50: 24nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 6806BDBM6806(6-(benzyloxy)-18-methyl-3,13,18-triazahexacyclo[14...)
Affinity DataIC50: 25nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 6838BDBM6838(1-(2-{18-methyl-12,14-dioxo-3,13,18-triazahexacycl...)
Affinity DataIC50: 25nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 6817BDBM6817(18,23-dimethyl-6-(trifluoromethyl)-3,13,18-triazah...)
Affinity DataIC50: 25nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 6811BDBM6811(18,23-dimethyl-3,13,18-triazahexacyclo[14.7.0.0^{2...)
Affinity DataIC50: 28nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2005
Entry Details Article
PubMed
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