Compile Data Set for Download or QSAR
Report error Found 9 Enz. Inhib. hit(s) with all data for entry = 5419
TargetMetabotropic glutamate receptor 5(Rat)
Merck Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50084137(2-Methyl-6-phenylethynyl-pyridine | CHEMBL66654 | ...)
Affinity DataKi:  0.300nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2012
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 1(Rat)
Merck Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50030629(4-(Amino-carboxy-methyl)-benzoic acid | (S)-4CPG |...)
Affinity DataKi:  1.10E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2012
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 2(Human)
Merck Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50030630(AIDA | AIDC | 1-Amino-indan-1,5-dicarboxylic acid(...)
Affinity DataKi:  1.10E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2012
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Rat)
Merck Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM86230(NSC_2866 | CAS_146-48-5 | YOHIMBINE)
Affinity DataKi:  7.60E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2012
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Rat)
Merck Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM86232(NSC_2325 | CAS_2325 | Benoxathian)
Affinity DataKi:  7.60E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Rat)
Merck Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM86231(CAS_51-55-8 | NSC_3661 | Atropine,(-) | ATROPINE |...)
Affinity DataKi:  7.60E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Merck Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM22869(6-chloro-10-(4-methylpiperazin-1-yl)-2,9-diazatric...)
Affinity DataKi:  7.60E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2012
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 2B(Rat)
Merck Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50032651(1-[(1S,2S)-2-Hydroxy-2-(4-hydroxy-phenyl)-1-methyl...)
Affinity DataKi:  7.60E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2012
Entry Details Article
PubMed
TargetRetinoic acid receptor RXR-alpha(Rat)
Merck Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM86153(CAS_180081 | NSC_180081 | MK-801)
Affinity DataKi:  7.60E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2012
Entry Details Article
PubMed