Compile Data Set for Download or QSAR
Report error Found 10 Enz. Inhib. hit(s) with all data for entry = 50013136
TargetProtein kinase C alpha type(Human)
National Cancer Institute-Frederick

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50085904BDBM50085904(3-Isopropyl-4-methyl-pentanoic acid 2-hydroxymethy...)
Affinity DataKi:  2.90nMAssay Description:Displacement of [20-3H]phorbol-12,13-dibutyrate (PDBu) from recombinant Protein kinase C alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein kinase C alpha type(Human)
National Cancer Institute-Frederick

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50127016BDBM50127016(3-Methyl-butyric acid 3-hydroxymethyl-4-(3-isoprop...)
Affinity DataKi:  11nMAssay Description:Displacement of [20-3H]phorbol-12,13-dibutyrate (PDBu) from recombinant Protein kinase C alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein kinase C alpha type(Human)
National Cancer Institute-Frederick

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50127018BDBM50127018(3-Isopropyl-4-methyl-pentanoic acid 3-hydroxymethy...)
Affinity DataKi:  15nMAssay Description:Displacement of [20-3H]phorbol-12,13-dibutyrate (PDBu) from recombinant Protein kinase C alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein kinase C alpha type(Human)
National Cancer Institute-Frederick

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50127015BDBM50127015(3-Isopropyl-4-methyl-pentanoic acid 3-hydroxymethy...)
Affinity DataKi:  15nMAssay Description:Displacement of [20-3H]phorbol-12,13-dibutyrate (PDBu) from recombinant Protein kinase C alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein kinase C alpha type(Human)
National Cancer Institute-Frederick

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50087241BDBM50087241(3-Isopropyl-4-methyl-pentanoic acid 3-hydroxy-2-(3...)
Affinity DataKi:  29nMAssay Description:Displacement of [20-3H]phorbol-12,13-dibutyrate (PDBu) from recombinant Protein kinase C alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein kinase C alpha type(Human)
National Cancer Institute-Frederick

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50127019BDBM50127019(3-Isopropyl-4-methyl-pentanoic acid 3-hydroxymethy...)
Affinity DataKi:  30nMAssay Description:Displacement of [20-3H]phorbol-12,13-dibutyrate (PDBu) from recombinant Protein kinase C alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein kinase C alpha type(Human)
National Cancer Institute-Frederick

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50127017BDBM50127017(3-Methyl-butyric acid 3-hydroxymethyl-4-(3-isoprop...)
Affinity DataKi:  30nMAssay Description:Displacement of [20-3H]phorbol-12,13-dibutyrate (PDBu) from recombinant Protein kinase C alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein kinase C alpha type(Human)
National Cancer Institute-Frederick

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50100126BDBM50100126(3-Isopropyl-4-methyl-pent-2-enoic acid 1-hydroxyme...)
Affinity DataKi:  31nMAssay Description:Displacement of [20-3H]phorbol-12,13-dibutyrate (PDBu) from recombinant Protein kinase C alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein kinase C alpha type(Human)
National Cancer Institute-Frederick

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50100129BDBM50100129(3-Isopropyl-4-methyl-pentanoic acid 3-hydroxy-2-(3...)
Affinity DataKi:  40nMAssay Description:Displacement of [20-3H]phorbol-12,13-dibutyrate (PDBu) from recombinant Protein kinase C alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein kinase C alpha type(Human)
National Cancer Institute-Frederick

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50100121BDBM50100121(3-Isopropyl-4-methyl-pent-2-enoic acid 1-hydroxyme...)
Affinity DataKi:  330nMAssay Description:Displacement of [20-3H]phorbol-12,13-dibutyrate (PDBu) from recombinant Protein kinase C alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed