Compile Data Set for Download or QSAR
Report error Found 35 Enz. Inhib. hit(s) with all data for entry = 50013037
TargetMelanocyte-stimulating hormone receptor(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50125748(2-Acetylamino-N-[2-(4-butyryl-4-phenyl-piperidin-1...)
Affinity DataEC50:  0.350nMAssay Description:In vitro effective concentration towards human Melanocortin 1 receptor (MC1R) in SPA-based cAMP assay in melanoma cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50125750(N-[1-[2-(4-Butyryl-4-phenyl-piperidin-1-yl)-1-(4-m...)
Affinity DataEC50:  2.10E+3nMAssay Description:In vitro effective concentration towards human Melanocortin 5 receptor (MC5R) was determined by a SPA-based cAMP assay in melanoma cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50125747(N-[2-(4-Butyryl-4-phenyl-piperidin-1-yl)-1-(4-meth...)
Affinity DataEC50:  77nMAssay Description:In vitro effective concentration towards human Melanocortin 4 receptor (MC4R) was determined by a SPA-based cAMP assay in melanoma cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50125746(1'-[3-(4-methoxyphenyl)-2-(1,2,3,4-tetrahydro-3-is...)
Affinity DataEC50:  220nMAssay Description:In vitro inhibitory concentration against human Melanocortin 1 receptor (MC1R)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50125747(N-[2-(4-Butyryl-4-phenyl-piperidin-1-yl)-1-(4-meth...)
Affinity DataEC50:  2.70E+3nMAssay Description:In vitro effective concentration towards human Melanocortin 5 receptor (MC5R) was determined by a SPA-based cAMP assay in melanoma cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50125749(2-Amino-N-[2-(4-butyryl-4-phenyl-piperidin-1-yl)-1...)
Affinity DataEC50:  2.60E+3nMAssay Description:In vitro effective concentration towards human Melanocortin 4 receptor (MC4R) was determined by a SPA-based cAMP assay in melanoma cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50125750(N-[1-[2-(4-Butyryl-4-phenyl-piperidin-1-yl)-1-(4-m...)
Affinity DataEC50:  2.90nMAssay Description:In vitro effective concentration towards human Melanocortin 4 receptor (MC4R) was determined by a SPA-based cAMP assay in melanoma cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50125748(2-Acetylamino-N-[2-(4-butyryl-4-phenyl-piperidin-1...)
Affinity DataEC50:  23nMAssay Description:In vitro effective concentration towards human Melanocortin 4 receptor (MC4R) was determined by a SPA-based cAMP assay in melanoma cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50125743(N-[2-(4-Butyryl-4-phenyl-piperidin-1-yl)-1-(4-meth...)
Affinity DataEC50:  9.40E+3nMAssay Description:In vitro effective concentration towards human Melanocortin 5 receptor (MC5R) was determined by a SPA-based cAMP assay in melanoma cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50125744(2-Amino-N-[2-(4-butyryl-4-phenyl-piperidin-1-yl)-1...)
Affinity DataEC50:  1.00E+4nMAssay Description:In vitro effective concentration towards human Melanocortin 5 receptor (MC5R) was determined by a SPA-based cAMP assay in melanoma cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50125744(2-Amino-N-[2-(4-butyryl-4-phenyl-piperidin-1-yl)-1...)
Affinity DataEC50:  630nMAssay Description:In vitro effective concentration towards human Melanocortin 4 receptor (MC4R) was determined by a SPA-based cAMP assay in melanoma cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50125750(N-[1-[2-(4-Butyryl-4-phenyl-piperidin-1-yl)-1-(4-m...)
Affinity DataEC50:  0.190nMAssay Description:In vitro inhibitory concentration against human Melanocortin 1 receptor (MC1R)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50125748(2-Acetylamino-N-[2-(4-butyryl-4-phenyl-piperidin-1...)
Affinity DataEC50:  3.90E+3nMAssay Description:In vitro effective concentration towards human Melanocortin 5 receptor (MC5R) was determined by a SPA-based cAMP assay in melanoma cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50125743(N-[2-(4-Butyryl-4-phenyl-piperidin-1-yl)-1-(4-meth...)
Affinity DataEC50:  840nMAssay Description:In vitro effective concentration towards human Melanocortin 4 receptor (MC4R) was determined by a SPA-based cAMP assay in melanoma cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50125749(2-Amino-N-[2-(4-butyryl-4-phenyl-piperidin-1-yl)-1...)
Affinity DataEC50:  4.40E+3nMAssay Description:In vitro effective concentration towards human Melanocortin 5 receptor (MC5R) was determined by a SPA-based cAMP assay in melanoma cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50125745(2-Amino-N-[2-(4-butyryl-4-phenyl-piperidin-1-yl)-1...)
Affinity DataEC50:  510nMAssay Description:In vitro effective concentration towards human Melanocortin 1 receptor (MC1R) in SPA-based cAMP assay in melanoma cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50125743(N-[2-(4-Butyryl-4-phenyl-piperidin-1-yl)-1-(4-meth...)
Affinity DataEC50:  7.00E+3nMAssay Description:In vitro effective concentration towards human Melanocortin 3 receptor (MC3R) was determined by a SPA-based cAMP assay in melanoma cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50125747(N-[2-(4-Butyryl-4-phenyl-piperidin-1-yl)-1-(4-meth...)
Affinity DataEC50:  3.80nMAssay Description:In vitro effective concentration towards human Melanocortin 1 receptor (MC1R) in SPA-based cAMP assay in melanoma cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50125744(2-Amino-N-[2-(4-butyryl-4-phenyl-piperidin-1-yl)-1...)
Affinity DataEC50:  1.70E+3nMAssay Description:In vitro effective concentration towards human Melanocortin 3 receptor (MC3R) was determined by a SPA-based cAMP assay in melanoma cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50125743(N-[2-(4-Butyryl-4-phenyl-piperidin-1-yl)-1-(4-meth...)
Affinity DataEC50:  2.5nMAssay Description:In vitro effective concentration towards human Melanocortin 1 receptor (MC1R) in SPA-based cAMP assay in melanoma cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50125747(N-[2-(4-Butyryl-4-phenyl-piperidin-1-yl)-1-(4-meth...)
Affinity DataEC50:  3.90E+3nMAssay Description:In vitro effective concentration towards human Melanocortin-3 receptor (MC3R) was determined by a SPA-based cAMP assay in melanoma cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50125751(2-Amino-N-[2-(4-butyryl-4-phenyl-piperidin-1-yl)-1...)
Affinity DataEC50:  400nMAssay Description:In vitro effective concentration towards human Melanocortin 1 receptor (MC1R) in SPA-based cAMP assay in melanoma cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50125750(N-[1-[2-(4-Butyryl-4-phenyl-piperidin-1-yl)-1-(4-m...)
Affinity DataEC50:  250nMAssay Description:In vitro effective concentration towards human Melanocortin 3 receptor (MC3R) was determined by a SPA-based cAMP assay in melanoma cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50125744(2-Amino-N-[2-(4-butyryl-4-phenyl-piperidin-1-yl)-1...)
Affinity DataEC50:  1.5nMAssay Description:In vitro effective concentration towards human Melanocortin 1 receptor (MC1R) in SPA-based cAMP assay in melanoma cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50125749(2-Amino-N-[2-(4-butyryl-4-phenyl-piperidin-1-yl)-1...)
Affinity DataEC50:  28nMAssay Description:In vitro effective concentration towards human Melanocortin 1 receptor (MC1R) in SPA-based cAMP assay in melanoma cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50125748(2-Acetylamino-N-[2-(4-butyryl-4-phenyl-piperidin-1...)
Affinity DataEC50:  2.20E+3nMAssay Description:In vitro effective concentration towards human Melanocortin 3 receptor (MC3R) was determined by a SPA-based cAMP assay in melanoma cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50125746(1'-[3-(4-methoxyphenyl)-2-(1,2,3,4-tetrahydro-3-is...)
Affinity DataEC50:  40nMAssay Description:In vitro effective concentration towards human Melanocortin 4 receptor (MC4R) was determined by a SPA-based cAMP assay in melanoma cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50125750(N-[1-[2-(4-Butyryl-4-phenyl-piperidin-1-yl)-1-(4-m...)
Affinity DataIC50: 3.10nMAssay Description:In vitro inhibitory concentration of the compound against human Melanocortin 1 receptor (MC1R)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50125748(2-Acetylamino-N-[2-(4-butyryl-4-phenyl-piperidin-1...)
Affinity DataIC50: 5.10nMAssay Description:In vitro inhibitory concentration of the compound against human Melanocortin 1 receptor (MC1R)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50125747(N-[2-(4-Butyryl-4-phenyl-piperidin-1-yl)-1-(4-meth...)
Affinity DataIC50: 5.5nMAssay Description:In vitro inhibitory concentration of the compound against human Melanocortin 1 receptor (MC1R)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50125743(N-[2-(4-Butyryl-4-phenyl-piperidin-1-yl)-1-(4-meth...)
Affinity DataIC50: 18nMAssay Description:In vitro inhibitory concentration of the compound against human Melanocortin 1 receptor (MC1R)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50125744(2-Amino-N-[2-(4-butyryl-4-phenyl-piperidin-1-yl)-1...)
Affinity DataIC50: 32nMAssay Description:In vitro inhibitory concentration of the compound against human Melanocortin 1 receptor (MC1R)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50125749(2-Amino-N-[2-(4-butyryl-4-phenyl-piperidin-1-yl)-1...)
Affinity DataIC50: 120nMAssay Description:In vitro inhibitory concentration of the compound against human Melanocortin 1 receptor (MC1R)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50125751(2-Amino-N-[2-(4-butyryl-4-phenyl-piperidin-1-yl)-1...)
Affinity DataIC50: 1.30E+3nMAssay Description:In vitro inhibitory concentration of the compound against human Melanocortin 1 receptor (MC1R)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50125745(2-Amino-N-[2-(4-butyryl-4-phenyl-piperidin-1-yl)-1...)
Affinity DataIC50: 1.50E+3nMAssay Description:In vitro inhibitory concentration of the compound against human Melanocortin 1 receptor (MC1R)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed