Compile Data Set for Download or QSAR
Report error Found 23 Enz. Inhib. hit(s) with all data for entry = 50012892
TargetMelanocyte-stimulating hormone receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50123944(9-Benzyl-6-(3-guanidino-propyl)-12-(3H-imidazol-4-...)
Affinity DataEC50:  2.70E+3nMAssay Description:Agonistic activity towards Melanocortin 1 receptor in the Xenopus frog skin assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50123943(c[Pro-D-Nal(2')-Arg-Trp-Glu]-Val-Val-Gly-NH2 | CHE...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonistic activity towards Melanocortin 1 receptor in the Xenopus frog skin assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50123950(c[His-D-Nal(2')-Arg-Trp-Glu]-Val-Val-Gly-NH2 | CHE...)
Affinity DataEC50:  60nMAssay Description:Agonistic activity towards Melanocortin 1 receptor in the Xenopus frog skin assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50123951(9-Benzyl-6-(3-guanidino-propyl)-12-(3H-imidazol-4-...)
Affinity DataEC50:  313nMAssay Description:Agonistic activity towards Melanocortin 1 receptor in the Xenopus frog skin assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50123940(c[Gly-Pro-D-Nal(2')-Arg-Trp-Glu]-Val-Val-Gly-NH2 |...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonistic activity towards Melanocortin 1 receptor in the Xenopus frog skin assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50123949(c[gamma-Abu-His-D-Nal(2')-Arg-Trp-Glu]-Val-Val-Gly...)
Affinity DataEC50:  23nMAssay Description:Agonistic activity towards Melanocortin 1 receptor in the Xenopus frog skin assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50123946(5-Benzyl-8-(3-guanidino-propyl)-2-(3H-imidazol-4-y...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonistic activity towards Melanocortin 1 receptor in the Xenopus frog skin assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50123947(c[6-Ahx-His-phe-Arg-Trp-Glu]-Val-Val-Gly-NH2 | CHE...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonistic activity towards Melanocortin 1 receptor in the Xenopus frog skin assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50123948(c[beta-Ala-His-D-phe-Arg-Trp-Glu]-Val-Val-Gly-NH2 ...)
Affinity DataEC50:  31nMAssay Description:Agonistic activity towards Melanocortin 1 receptor in the Xenopus frog skin assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50123945(c[6-Ahx-His-D-phe-Arg-Trp-Glu]-Val-Val-Gly-NH2 | C...)
Affinity DataEC50:  23nMAssay Description:Agonistic activity towards Melanocortin 1 receptor in the Xenopus frog skin assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50123936(19-Benzyl-16-(3-guanidino-propyl)-13-(1H-indol-3-y...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonistic activity towards Melanocortin 1 receptor in the Xenopus frog skin assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50123935(8-Benzyl-11-(3-guanidino-propyl)-5-(3H-imidazol-4-...)
Affinity DataEC50:  510nMAssay Description:Agonistic activity towards Melanocortin 1 receptor in the Xenopus frog skin assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50123942(c[beta-Ala-His-D-Nal(2')-Arg-Trp-Glu]-Val-Val-Gly-...)
Affinity DataEC50:  2nMAssay Description:Agonistic activity towards Melanocortin 1 receptor in the Xenopus frog skin assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50123941(8-Benzyl-11-(3-guanidino-propyl)-5-(3H-imidazol-4-...)
Affinity DataEC50:  5.20E+3nMAssay Description:Agonistic activity towards Melanocortin 1 receptor in the Xenopus frog skin assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50123939(5-Benzyl-8-(3-guanidino-propyl)-2-(3H-imidazol-4-y...)
Affinity DataEC50:  825nMAssay Description:Agonistic activity towards Melanocortin 1 receptor in the Xenopus frog skin assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50123938(c[Gly-His-D-Nal(2')-Arg-Trp-Glu]-Val-Val-Gly-NH2 |...)
Affinity DataEC50:  60nMAssay Description:Agonistic activity towards Melanocortin 1 receptor in the Xenopus frog skin assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50123937(4-[8-Benzyl-17-{1-[1-(carbamoylmethyl-carbamoyl)-2...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonistic activity towards Melanocortin 1 receptor in the Xenopus frog skin assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50123937(4-[8-Benzyl-17-{1-[1-(carbamoylmethyl-carbamoyl)-2...)
Affinity DataIC50: 440nMAssay Description:Antagonistic activity towards Melanocortin 1 receptor in Xenopus frog skin using competitive binding in the presence of 500 pM of alpha-melanocyte st...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50123939(5-Benzyl-8-(3-guanidino-propyl)-2-(3H-imidazol-4-y...)
Affinity DataIC50: 455nMAssay Description:Antagonistic activity towards Melanocortin 1 receptor in Xenopus frog skin using competitive binding in the presence of 500 pM of alpha-melanocyte st...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50123940(c[Gly-Pro-D-Nal(2')-Arg-Trp-Glu]-Val-Val-Gly-NH2 |...)
Affinity DataIC50: 637nMAssay Description:Antagonistic activity towards Melanocortin 1 receptor in Xenopus frog skin using competitive binding in the presence of 500 pM of alpha-melanocyte st...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50123943(c[Pro-D-Nal(2')-Arg-Trp-Glu]-Val-Val-Gly-NH2 | CHE...)
Affinity DataIC50: 1.50E+3nMAssay Description:Antagonistic activity towards Melanocortin 1 receptor in Xenopus frog skin using competitive binding in the presence of 500 pM of alpha-melanocyte st...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50123946(5-Benzyl-8-(3-guanidino-propyl)-2-(3H-imidazol-4-y...)
Affinity DataIC50: 8.20E+3nMAssay Description:Antagonistic activity towards Melanocortin 1 receptor in Xenopus frog skin using competitive binding in the presence of 500 pM of alpha-melanocyte st...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50123936(19-Benzyl-16-(3-guanidino-propyl)-13-(1H-indol-3-y...)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonistic activity towards Melanocortin 1 receptor in Xenopus frog skin using competitive binding in the presence of 500 pM of alpha-melanocyte st...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed