Compile Data Set for Download or QSAR
Report error Found 46 Enz. Inhib. hit(s) with all data for entry = 50037231
TargetDelta-type opioid receptor(Rat)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50123658(3-[(R)-((2S,5R)-4-Allyl-2,5-dimethyl-piperazin-1-y...)
Affinity DataKi:  0.180nMAssay Description:Binding affinity of compound evaluated for Opioid receptor delta 1 isolated from rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50123658(3-[(R)-((2S,5R)-4-Allyl-2,5-dimethyl-piperazin-1-y...)
Affinity DataKi:  0.180nMAssay Description:Binding affinity of compound evaluated for Opioid receptor delta 1 isolated from rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50123658(3-[(R)-((2S,5R)-4-Allyl-2,5-dimethyl-piperazin-1-y...)
Affinity DataKi:  0.460nMAssay Description:Inhibition of [3H]DAMGO binding to mu opioid receptor of rat brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50123658(3-[(R)-((2S,5R)-4-Allyl-2,5-dimethyl-piperazin-1-y...)
Affinity DataKi:  0.460nMAssay Description:Inhibition of [3H]DAMGO binding to mu opioid receptor of rat brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50000092(Analog of 14-(Arylhydroxyamino)codeinone | 4-methy...)
Affinity DataKi:  1nMAssay Description:Inhibition of [3H]DAMGO binding to mu opioid receptor of rat brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50123655(3-[(S)-((2S,5R)-4-Allyl-2,5-dimethyl-piperazin-1-y...)
Affinity DataKi:  1.06nMAssay Description:Binding affinity of compound evaluated for Opioid receptor delta 1 isolated from rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50123647(3-[(R)-((2S,5R)-4-Allyl-2,5-dimethyl-piperazin-1-y...)
Affinity DataKi:  1.06nMAssay Description:Inhibition of [3H]DAMGO binding to mu opioid receptor of rat brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50123654({3-[(R)-((2S,5R)-4-Allyl-2,5-dimethyl-piperazin-1-...)
Affinity DataKi:  1.18nMAssay Description:Binding affinity of compound evaluated for Opioid receptor delta 1 isolated from rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50123664(3-[(R)-((2S,5R)-4-Allyl-2,5-dimethyl-piperazin-1-y...)
Affinity DataKi:  1.26nMAssay Description:Binding affinity of compound evaluated for Opioid receptor delta 1 isolated from rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50123647(3-[(R)-((2S,5R)-4-Allyl-2,5-dimethyl-piperazin-1-y...)
Affinity DataKi:  1.37nMAssay Description:Binding affinity of compound evaluated for Opioid receptor delta 1 isolated from rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50123649(3-[(R)-((2S,5R)-4-Allyl-2,5-dimethyl-piperazin-1-y...)
Affinity DataKi:  1.40nMAssay Description:Binding affinity of compound evaluated for Opioid receptor delta 1 isolated from rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50123649(3-[(R)-((2S,5R)-4-Allyl-2,5-dimethyl-piperazin-1-y...)
Affinity DataKi:  1.49nMAssay Description:Inhibition of [3H]DAMGO binding to mu opioid receptor of rat brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50008984(N-(1-Phenethyl-piperidin-4-yl)-N-phenyl-propionami...)
Affinity DataKi:  1.5nMAssay Description:Inhibition of [3H]DAMGO binding to mu opioid receptor of rat brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetMu-type opioid receptor(Rat)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50123655(3-[(S)-((2S,5R)-4-Allyl-2,5-dimethyl-piperazin-1-y...)
Affinity DataKi:  1.55nMAssay Description:Inhibition of [3H]DAMGO binding to mu opioid receptor of rat brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50123665(3-[(R)-((2S,5R)-4-Allyl-2,5-dimethyl-piperazin-1-y...)
Affinity DataKi:  1.58nMAssay Description:Inhibition of [3H]DAMGO binding to mu opioid receptor of rat brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50123665(3-[(R)-((2S,5R)-4-Allyl-2,5-dimethyl-piperazin-1-y...)
Affinity DataKi:  1.69nMAssay Description:Binding affinity of compound evaluated for Opioid receptor delta 1 isolated from rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50123662(3-[(R)-((2S,5R)-4-Allyl-2,5-dimethyl-piperazin-1-y...)
Affinity DataKi:  1.75nMAssay Description:Binding affinity of compound evaluated for Opioid receptor delta 1 isolated from rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50039026(4-[(R)-((2S,5R)-4-Allyl-2,5-dimethyl-piperazin-1-y...)
Affinity DataKi:  1.80nMAssay Description:Binding affinity of compound evaluated for Opioid receptor delta 1 isolated from rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50123664(3-[(R)-((2S,5R)-4-Allyl-2,5-dimethyl-piperazin-1-y...)
Affinity DataKi:  1.82nMAssay Description:Inhibition of [3H]DAMGO binding to mu opioid receptor of rat brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50123657(3-[(R)-((2S,5R)-4-Allyl-2,5-dimethyl-piperazin-1-y...)
Affinity DataKi:  1.88nMAssay Description:Binding affinity of compound evaluated for Opioid receptor delta 1 isolated from rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50123660(3-[(R)-((2S,5R)-4-Allyl-2,5-dimethyl-piperazin-1-y...)
Affinity DataKi:  1.92nMAssay Description:Binding affinity of compound evaluated for Opioid receptor delta 1 isolated from rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50123656(3-[(R)-((2S,5R)-4-Allyl-2,5-dimethyl-piperazin-1-y...)
Affinity DataKi:  2.01nMAssay Description:Binding affinity of compound evaluated for Opioid receptor delta 1 isolated from rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50123652(3-[(S)-((2S,5R)-4-Allyl-2,5-dimethyl-piperazin-1-y...)
Affinity DataKi:  2.10nMAssay Description:Binding affinity of compound evaluated for Opioid receptor delta 1 isolated from rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50123657(3-[(R)-((2S,5R)-4-Allyl-2,5-dimethyl-piperazin-1-y...)
Affinity DataKi:  2.16nMAssay Description:Inhibition of [3H]DAMGO binding to mu opioid receptor of rat brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50123650(3-[(R)-((2S,5R)-4-Allyl-2,5-dimethyl-piperazin-1-y...)
Affinity DataKi:  2.17nMAssay Description:Binding affinity of compound evaluated for Opioid receptor delta 1 isolated from rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50123662(3-[(R)-((2S,5R)-4-Allyl-2,5-dimethyl-piperazin-1-y...)
Affinity DataKi:  2.19nMAssay Description:Inhibition of [3H]DAMGO binding to mu opioid receptor of rat brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50123648(3-[(R)-((2S,5R)-4-Allyl-2,5-dimethyl-piperazin-1-y...)
Affinity DataKi:  2.31nMAssay Description:Binding affinity of compound evaluated for Opioid receptor delta 1 isolated from rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50123656(3-[(R)-((2S,5R)-4-Allyl-2,5-dimethyl-piperazin-1-y...)
Affinity DataKi:  2.35nMAssay Description:Inhibition of [3H]DAMGO binding to mu opioid receptor of rat brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50123660(3-[(R)-((2S,5R)-4-Allyl-2,5-dimethyl-piperazin-1-y...)
Affinity DataKi:  2.37nMAssay Description:Inhibition of [3H]DAMGO binding to mu opioid receptor of rat brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50123653(3-[(R)-((2S,5R)-4-Allyl-2,5-dimethyl-piperazin-1-y...)
Affinity DataKi:  2.41nMAssay Description:Binding affinity of compound evaluated for Opioid receptor delta 1 isolated from rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50123654({3-[(R)-((2S,5R)-4-Allyl-2,5-dimethyl-piperazin-1-...)
Affinity DataKi:  2.55nMAssay Description:Inhibition of [3H]DAMGO binding to mu opioid receptor of rat brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50123646(3-[(R)-((2S,5R)-4-Allyl-2,5-dimethyl-piperazin-1-y...)
Affinity DataKi:  2.73nMAssay Description:Binding affinity of compound evaluated for Opioid receptor delta 1 isolated from rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50123648(3-[(R)-((2S,5R)-4-Allyl-2,5-dimethyl-piperazin-1-y...)
Affinity DataKi:  2.74nMAssay Description:Inhibition of [3H]DAMGO binding to mu opioid receptor of rat brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50123651(3-[(R)-((2S,5R)-4-Allyl-2,5-dimethyl-piperazin-1-y...)
Affinity DataKi:  2.75nMAssay Description:Binding affinity of compound evaluated for Opioid receptor delta 1 isolated from rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50123653(3-[(R)-((2S,5R)-4-Allyl-2,5-dimethyl-piperazin-1-y...)
Affinity DataKi:  2.78nMAssay Description:Inhibition of [3H]DAMGO binding to mu opioid receptor of rat brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50123652(3-[(S)-((2S,5R)-4-Allyl-2,5-dimethyl-piperazin-1-y...)
Affinity DataKi:  3.20nMAssay Description:Inhibition of [3H]DAMGO binding to mu opioid receptor of rat brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50123650(3-[(R)-((2S,5R)-4-Allyl-2,5-dimethyl-piperazin-1-y...)
Affinity DataKi:  3.39nMAssay Description:Inhibition of [3H]DAMGO binding to mu opioid receptor of rat brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50123646(3-[(R)-((2S,5R)-4-Allyl-2,5-dimethyl-piperazin-1-y...)
Affinity DataKi:  3.46nMAssay Description:Inhibition of [3H]DAMGO binding to mu opioid receptor of rat brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50123659(3-[(R)-((2S,5R)-4-Allyl-2,5-dimethyl-piperazin-1-y...)
Affinity DataKi:  6.95nMAssay Description:Binding affinity of compound evaluated for Opioid receptor delta 1 isolated from rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50123651(3-[(R)-((2S,5R)-4-Allyl-2,5-dimethyl-piperazin-1-y...)
Affinity DataKi:  7.06nMAssay Description:Inhibition of [3H]DAMGO binding to mu opioid receptor of rat brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50123659(3-[(R)-((2S,5R)-4-Allyl-2,5-dimethyl-piperazin-1-y...)
Affinity DataKi:  7.08nMAssay Description:Inhibition of [3H]DAMGO binding to mu opioid receptor of rat brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50123661(3-[(R)-((2S,5R)-4-Allyl-2,5-dimethyl-piperazin-1-y...)
Affinity DataKi:  8.88nMAssay Description:Inhibition of [3H]DAMGO binding to mu opioid receptor of rat brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50123661(3-[(R)-((2S,5R)-4-Allyl-2,5-dimethyl-piperazin-1-y...)
Affinity DataKi:  9.20nMAssay Description:Binding affinity of compound evaluated for Opioid receptor delta 1 isolated from rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50039026(4-[(R)-((2S,5R)-4-Allyl-2,5-dimethyl-piperazin-1-y...)
Affinity DataKi:  15nMAssay Description:Inhibition of [3H]DAMGO binding to mu opioid receptor of rat brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50000092(Analog of 14-(Arylhydroxyamino)codeinone | 4-methy...)
Affinity DataKi:  90nMAssay Description:Binding affinity of compound evaluated for Opioid receptor delta 1 isolated from rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50008984(N-(1-Phenethyl-piperidin-4-yl)-N-phenyl-propionami...)
Affinity DataKi:  400nMAssay Description:Binding affinity of compound evaluated for Opioid receptor delta 1 isolated from rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed