Compile Data Set for Download or QSAR
Report error Found 11 Enz. Inhib. hit(s) with all data for entry = 50012804
TargetProtein kinase C alpha type(Human)
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50122942(5-(3,5-Bis-trifluoromethyl-phenyl)-penta-2,4-dieno...)
Affinity DataKi:  5.60nMAssay Description:Displacement of PDBU from recombinant Protein kinase C alpha with phosphatidylserineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein kinase C alpha type(Human)
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50122938(5-(3,5-Bis-trifluoromethyl-phenyl)-pentanoic acid ...)
Affinity DataKi:  7.80nMAssay Description:Displacement of PDBU from recombinant Protein kinase C alpha with phosphatidylserineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein kinase C alpha type(Human)
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50122941(5-[4-(3,3,4,4,5,5,6,6,7,7,8,8,8-Tridecafluoro-octy...)
Affinity DataKi:  9.20nMAssay Description:Displacement of PDBU from recombinant Protein kinase C alpha with phosphatidylserineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein kinase C alpha type(Human)
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50122945(5-[4-(3,3,4,4,5,5,6,6,7,7,8,8,8-Tridecafluoro-oct-...)
Affinity DataKi:  11nMAssay Description:Displacement of PDBU from recombinant Protein kinase C alpha with phosphatidylserineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein kinase C alpha type(Human)
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50122940(5-(4-Trifluoromethyl-phenyl)-penta-2,4-dienoic aci...)
Affinity DataKi:  12nMAssay Description:Displacement of PDBU from recombinant Protein kinase C alpha with phosphatidylserineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein kinase C alpha type(Human)
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50122939(5-(4-Trifluoromethyl-phenyl)-pentanoic acid (5-hyd...)
Affinity DataKi:  13nMAssay Description:Displacement of PDBU from recombinant Protein kinase C alpha with phosphatidylserineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein kinase C alpha type(Human)
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50057509(8-Dec-1-ynyl-5-hydroxymethyl-2-isopropyl-1-methyl-...)
Affinity DataKi:  15nMAssay Description:Displacement of PDBU from recombinant Protein kinase C alpha with phosphatidylserineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein kinase C alpha type(Human)
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50122944(5-Phenyl-penta-2,4-dienoic acid (5-hydroxymethyl-2...)
Affinity DataKi:  16nMAssay Description:Displacement of PDBU from recombinant Protein kinase C alpha with phosphatidylserineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein kinase C alpha type(Human)
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50122937(5-Phenyl-pentanoic acid (5-hydroxymethyl-2-isoprop...)
Affinity DataKi:  34nMAssay Description:Displacement of PDBU from recombinant Protein kinase C alpha with phosphatidylserineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein kinase C alpha type(Human)
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50122946(Hexanoic acid [(S)-5-hydroxymethyl-2-((S)-isopropy...)
Affinity DataKi:  225nMAssay Description:Displacement of PDBU from recombinant Protein kinase C alpha with phosphatidylserineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein kinase C alpha type(Human)
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50122943(Hexa-2,4-dienoic acid (5-hydroxymethyl-2-isopropyl...)
Affinity DataKi:  1.97E+3nMAssay Description:Displacement of PDBU from recombinant Protein kinase C alpha with phosphatidylserineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed