Compile Data Set for Download or QSAR
Report error Found 22 Enz. Inhib. hit(s) with all data for entry = 5387
TargetTyrosine-protein kinase Lck(Human)
University of Dundee

Curated by PDSP Ki Database
LigandPNGBDBM25116(cid_1400 | CHEMBL306380 | 1-tert-butyl-3-(4-methyl...)
Affinity DataKi:  50nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2012
Entry Details Article
PubMed
TargetTyrosine-protein kinase Lck(Human)
University of Dundee

Curated by PDSP Ki Database
LigandPNGBDBM50142887(1-tert-Butyl-3-(4-chloro-phenyl)-1H-pyrazolo[3,4-d...)
Affinity DataKi:  60nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2012
Entry Details Article
PubMed
TargetCyclin-dependent kinase 2(Human)
University of Dundee

Curated by PDSP Ki Database
LigandPNGBDBM7262(NSC 705701 | BDBM84528 | alsterpaullone | 9-Nitrop...)
Affinity DataKi:  80nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2012
Entry Details Article
PubMed
TargetCyclin-dependent kinase 2(Human)
University of Dundee

Curated by PDSP Ki Database
LigandPNGBDBM27216((2R)-2-({6-[(3-chlorophenyl)amino]-9-(propan-2-yl)...)
Affinity DataKi:  100nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2012
Entry Details Article
PubMed
TargetNinein(Human)
University of Dundee

Curated by PDSP Ki Database
LigandPNGBDBM7262(NSC 705701 | BDBM84528 | alsterpaullone | 9-Nitrop...)
Affinity DataKi:  110nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2012
Entry Details Article
PubMed
TargetNinein(Human)
University of Dundee

Curated by PDSP Ki Database
LigandPNGBDBM7393(Indirubin-3 -monoxime | 3-[(2Z,3E)-3-(hydroxyimino...)
Affinity DataKi:  190nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2012
Entry Details Article
PubMed
TargetNinein(Human)
University of Dundee

Curated by PDSP Ki Database
LigandPNGBDBM7266(cid_3820 | NSC 664704 | 9-bromopaullone | 14-bromo...)
Affinity DataKi:  230nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2012
Entry Details Article
PubMed
TargetCyclin-dependent kinase 2(Human)
University of Dundee

Curated by PDSP Ki Database
LigandPNGBDBM7533(2,6,9-Trisubstituted purine deriv. 28 | (2R)-2-[[6...)
Affinity DataKi:  250nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2012
Entry Details Article
PubMed
TargetTyrosine-protein kinase Lck(Human)
University of Dundee

Curated by PDSP Ki Database
LigandPNGBDBM7393(Indirubin-3 -monoxime | 3-[(2Z,3E)-3-(hydroxyimino...)
Affinity DataKi:  300nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2012
Entry Details Article
PubMed
LigandPNGBDBM27216((2R)-2-({6-[(3-chlorophenyl)amino]-9-(propan-2-yl)...)
Affinity DataKi:  300nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2012
Entry Details Article
PubMed
LigandPNGBDBM50070942((-)-Epigallocatechin-3-o-gallate | (-)-Epigallocat...)
Affinity DataKi:  330nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2012
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase Sgk1(Human)
University of Dundee

Curated by PDSP Ki Database
LigandPNGBDBM7393(Indirubin-3 -monoxime | 3-[(2Z,3E)-3-(hydroxyimino...)
Affinity DataKi:  380nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2012
Entry Details Article
PubMed
TargetTyrosine-protein kinase Lck(Human)
University of Dundee

Curated by PDSP Ki Database
LigandPNGBDBM7262(NSC 705701 | BDBM84528 | alsterpaullone | 9-Nitrop...)
Affinity DataKi:  470nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2012
Entry Details Article
PubMed
TargetTyrosine-protein kinase Lck(Human)
University of Dundee

Curated by PDSP Ki Database
LigandPNGBDBM7266(cid_3820 | NSC 664704 | 9-bromopaullone | 14-bromo...)
Affinity DataKi:  470nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2012
Entry Details Article
PubMed
TargetCyclin-dependent kinase 2(Human)
University of Dundee

Curated by PDSP Ki Database
LigandPNGBDBM7393(Indirubin-3 -monoxime | 3-[(2Z,3E)-3-(hydroxyimino...)
Affinity DataKi:  590nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2012
Entry Details Article
PubMed
TargetCyclin-dependent kinase 2(Human)
University of Dundee

Curated by PDSP Ki Database
LigandPNGBDBM7266(cid_3820 | NSC 664704 | 9-bromopaullone | 14-bromo...)
Affinity DataKi:  670nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2012
Entry Details Article
PubMed
TargetTyrosine-protein kinase CSK(Human)
University of Dundee

Curated by PDSP Ki Database
LigandPNGBDBM50142887(1-tert-Butyl-3-(4-chloro-phenyl)-1H-pyrazolo[3,4-d...)
Affinity DataKi:  730nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2012
Entry Details Article
PubMed
TargetCasein kinase I isoform delta(Rat)
University of Dundee

Curated by PDSP Ki Database
LigandPNGBDBM25116(cid_1400 | CHEMBL306380 | 1-tert-butyl-3-(4-methyl...)
Affinity DataKi:  1.06E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2012
Entry Details Article
PubMed
TargetCasein kinase I isoform delta(Rat)
University of Dundee

Curated by PDSP Ki Database
LigandPNGBDBM50142887(1-tert-Butyl-3-(4-chloro-phenyl)-1H-pyrazolo[3,4-d...)
Affinity DataKi:  1.29E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2012
Entry Details Article
PubMed
LigandPNGBDBM7533(2,6,9-Trisubstituted purine deriv. 28 | (2R)-2-[[6...)
Affinity DataKi:  3.10E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2012
Entry Details Article
PubMed
TargetCasein kinase I isoform delta(Rat)
University of Dundee

Curated by PDSP Ki Database
LigandPNGBDBM50013720(CHEMBL65063 | PP3 | cid_4879 | 1-Phenyl-1H-pyrazol...)
Affinity DataKi:  9.90E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2012
Entry Details Article
PubMed
TargetCasein kinase I isoform delta(Rat)
University of Dundee

Curated by PDSP Ki Database
LigandPNGBDBM7533(2,6,9-Trisubstituted purine deriv. 28 | (2R)-2-[[6...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2012
Entry Details Article
PubMed