Compile Data Set for Download or QSAR
Report error Found 17 Enz. Inhib. hit(s) with all data for entry = 50048546
Target5-hydroxytryptamine receptor 7(Human)
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50220557(CHEMBL422869)
Affinity DataKi:  2nMAssay Description:Ability to displace the radioligand [3H]5-carboximidotryptamine ([3H]-5-CT) from cloned human 5-hydroxytryptamine 7 receptor expressed in COS-7 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2018
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 7(Human)
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50116963(2a-[4-(4-Phenyl-3,6-dihydro-2H-pyridin-1-yl)-butyl...)
Affinity DataKi:  2.10nMAssay Description:Ability to displace the radioligand [3H]5-carboximidotryptamine ([3H]-5-CT) from cloned human 5-hydroxytryptamine 7 receptor expressed in COS-7 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2018
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 7(Human)
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50220558(CHEMBL418888)
Affinity DataKi:  3.5nMAssay Description:Ability to displace the radioligand [3H]5-carboximidotryptamine ([3H]-5-CT) from cloned human 5-hydroxytryptamine 7 receptor expressed in COS-7 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2018
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 7(Human)
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50220504(CHEMBL348410)
Affinity DataKi:  5nMAssay Description:Ability to displace the radioligand [3H]5-carboximidotryptamine ([3H]-5-CT) from cloned human 5-hydroxytryptamine 7 receptor expressed in COS-7 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2018
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 7(Human)
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50220503(CHEMBL348890)
Affinity DataKi:  7.20nMAssay Description:Binding affinity towards 5-HT7 receptor by the displacement of [3H]-5-CT] in human recombinant receptors in mammalian cellMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2018
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 7(Human)
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50220503(CHEMBL348890)
Affinity DataKi:  7.20nMAssay Description:Ability to displace the radioligand [3H]5-carboximidotryptamine ([3H]-5-CT) from cloned human 5-hydroxytryptamine 7 receptor expressed in COS-7 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2018
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50220558(CHEMBL418888)
Affinity DataKi:  66nMAssay Description:Binding affinity towards 5-hydroxytryptamine 2 receptor by the displacement of [3H]ketanserin in rat cerebral cortex membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2018
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50116963(2a-[4-(4-Phenyl-3,6-dihydro-2H-pyridin-1-yl)-butyl...)
Affinity DataKi:  98nMAssay Description:Binding affinity towards 5-hydroxytryptamine 2 receptor by the displacement of [3H]ketanserin in rat cerebral cortex membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2018
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50220557(CHEMBL422869)
Affinity DataKi:  229nMAssay Description:Binding affinity towards 5-hydroxytryptamine 2 receptor by the displacement of [3H]ketanserin in rat cerebral cortex membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2018
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50220504(CHEMBL348410)
Affinity DataKi:  316nMAssay Description:Binding affinity towards 5-hydroxytryptamine 2 receptor by the displacement of [3H]ketanserin in rat cerebral cortex membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2018
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50220503(CHEMBL348890)
Affinity DataKi:  316nMAssay Description:Binding affinity towards 5-HT1A receptor by the displacement of [3H]-8-OH-DPAT] in human recombinant receptors in mammalian cellMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2018
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1B(Human)
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50220503(CHEMBL348890)
Affinity DataKi: <1.00E+3nMAssay Description:Binding affinity towards 5-HT1B receptor by the displacement of [3H]-5-CT] in human recombinant receptors in mammalian cellMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2018
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Guinea pig)
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50220503(CHEMBL348890)
Affinity DataKi: <1.00E+3nMAssay Description:Binding affinity towards 5-HT4 receptor by the displacement of [3H]GR-113808 in guinea-pig striatumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2018
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50220503(CHEMBL348890)
Affinity DataKi: <1.00E+3nMAssay Description:Binding affinity towards 5-HT2C receptor by the displacement of [3H]mesulergine] in human recombinant receptors in mammalian cellMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2018
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50220503(CHEMBL348890)
Affinity DataKi: <1.00E+3nMAssay Description:Binding affinity towards human recombinant 5-hydroxytryptamine 7 receptor by the displacement of [3H]-5-CT]More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2018
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50220503(CHEMBL348890)
Affinity DataKi: <1.00E+3nMAssay Description:Binding affinity towards 5-HT2 receptor by the displacement of [3H]-ketanserin] in rat cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2018
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50220503(CHEMBL348890)
Affinity DataKi: <1.00E+3nMAssay Description:Binding affinity towards 5-hydroxytryptamine 2 receptor by the displacement of [3H]ketanserin in rat cerebral cortex membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2018
Entry Details Article
PubMed