Compile Data Set for Download or QSAR
Report error Found 21 Enz. Inhib. hit(s) with all data for entry = 50012616
TargetGlucagon receptor(Human)
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50121047(5-Fluoro-2-[3-(1-hydroxy-ethyl)-2,6-diisopropyl-5-...)
Affinity DataIC50: 10nMAssay Description:Binding affinity of second enantiomer (E2) against human glucagon receptor was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50121049(5-Fluoro-2-[3-(1-hydroxy-ethyl)-2,6-diisopropyl-5-...)
Affinity DataIC50: 12nMAssay Description:Binding affinity of second enantiomer (E2) against human glucagon receptor was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50121045(2-[3-Ethyl-5-(1-hydroxy-ethyl)-2,6-diisopropyl-pyr...)
Affinity DataIC50: 16nMAssay Description:Binding affinity of second enantiomer (E2) against human glucagon receptor was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50121045(2-[3-Ethyl-5-(1-hydroxy-ethyl)-2,6-diisopropyl-pyr...)
Affinity DataIC50: 16nMAssay Description:Binding affinity of second enantiomer (E2) against human glucagon receptor was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50121047(5-Fluoro-2-[3-(1-hydroxy-ethyl)-2,6-diisopropyl-5-...)
Affinity DataIC50: 18nMAssay Description:Binding affinity of first diastereomer (D1) against human glucagon receptor was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50121045(2-[3-Ethyl-5-(1-hydroxy-ethyl)-2,6-diisopropyl-pyr...)
Affinity DataIC50: 20nMAssay Description:Binding affinity of first diastereomer (D1) against human glucagon receptor was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50121046(2-[3-(1-Hydroxy-ethyl)-2,6-diisopropyl-5-propyl-py...)
Affinity DataIC50: 25nMAssay Description:Binding affinity of second enantiomer (E2) against human glucagon receptor was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50121048(2-[3-Butyl-5-(1-hydroxy-ethyl)-2,6-diisopropyl-pyr...)
Affinity DataIC50: 28nMAssay Description:Binding affinity of first diastereomer (D1) against human glucagon receptor was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50121049(5-Fluoro-2-[3-(1-hydroxy-ethyl)-2,6-diisopropyl-5-...)
Affinity DataIC50: 30nMAssay Description:Binding affinity of first diastereomer (D1) against human glucagon receptor was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50121046(2-[3-(1-Hydroxy-ethyl)-2,6-diisopropyl-5-propyl-py...)
Affinity DataIC50: 40nMAssay Description:Binding affinity of first diastereomer (D1) against human glucagon receptor was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50109326((R)-1-[4-(4-Fluoro-phenyl)-2,6-diisopropyl-5-propy...)
Affinity DataIC50: 110nMAssay Description:Binding affinity of first diastereomer (D1) against human glucagon receptor was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50121046(2-[3-(1-Hydroxy-ethyl)-2,6-diisopropyl-5-propyl-py...)
Affinity DataIC50: 190nMAssay Description:Binding affinity of first enantiomer (E1) against human glucagon receptor was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50112476(5-Fluoro-2-(3-hydroxymethyl-2,6-diisopropyl-5-pent...)
Affinity DataIC50: 190nMAssay Description:Binding affinity of first diastereomer (D1) against human glucagon receptor was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50121047(5-Fluoro-2-[3-(1-hydroxy-ethyl)-2,6-diisopropyl-5-...)
Affinity DataIC50: 1.00E+3nMAssay Description:Binding affinity of second diastereomer (D2) against human glucagon receptor was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50121047(5-Fluoro-2-[3-(1-hydroxy-ethyl)-2,6-diisopropyl-5-...)
Affinity DataIC50: 1.00E+3nMAssay Description:Binding affinity of second diastereomer (D2) against human glucagon receptor was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50121048(2-[3-Butyl-5-(1-hydroxy-ethyl)-2,6-diisopropyl-pyr...)
Affinity DataIC50: 1.00E+3nMAssay Description:Binding affinity of second diastereomer (D2) against human glucagon receptor was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50121046(2-[3-(1-Hydroxy-ethyl)-2,6-diisopropyl-5-propyl-py...)
Affinity DataIC50: 1.10E+3nMAssay Description:Binding affinity of second diastereomer (D2) against human glucagon receptor was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50121049(5-Fluoro-2-[3-(1-hydroxy-ethyl)-2,6-diisopropyl-5-...)
Affinity DataIC50: 2.20E+3nMAssay Description:Binding affinity of second diastereomer (D2) against human glucagon receptor was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50121045(2-[3-Ethyl-5-(1-hydroxy-ethyl)-2,6-diisopropyl-pyr...)
Affinity DataIC50: 5.00E+3nMAssay Description:Binding affinity of first enantiomer (E1) against human glucagon receptor was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50109322([4-(4-Fluoro-phenyl)-2,6-diisopropyl-5-(2-methyl-p...)
Affinity DataIC50: 7.00E+3nMAssay Description:Binding affinity of first diastereomer (D1) against human glucagon receptor was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50121049(5-Fluoro-2-[3-(1-hydroxy-ethyl)-2,6-diisopropyl-5-...)
Affinity DataIC50: 8.00E+3nMAssay Description:Binding affinity of first enantiomer (E1) against human glucagon receptor was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed