Compile Data Set for Download or QSAR
Report error Found 89 Enz. Inhib. hit(s) with all data for entry = 4033
TargetGlycylpeptide N-tetradecanoyltransferase(Yeast)
Nippon Roche Research Center

LigandPNGBDBM50121720(CHEMBL355497 | Non peptidic, 5 | (1-METHYL-1H-IMID...)
Affinity DataIC50: 1nMAssay Description:Inhibition activity against C. albicans Nmt and human Nmt as assessed by IC50 using myristoyl-CoA (0.5 uM) and peptide substrate GLTISKLFRR-NH2 (0.5 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2011
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetGlycylpeptide N-tetradecanoyltransferase(Yeast)
Nippon Roche Research Center

LigandPNGBDBM50109879(Non peptidic, 4 | CHEMBL155301 | {3-[2-(2,3-Difluo...)
Affinity DataIC50: 4nMAssay Description:Inhibition activity against C. albicans Nmt and human Nmt as assessed by IC50 using myristoyl-CoA (0.5 uM) and peptide substrate GLTISKLFRR-NH2 (0.5 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2011
Entry Details Article
PubMed
TargetGlycylpeptide N-tetradecanoyltransferase 1(Human)
Nippon Roche Research Center

LigandPNGBDBM50109879(Non peptidic, 4 | CHEMBL155301 | {3-[2-(2,3-Difluo...)
Affinity DataIC50: 62nMAssay Description:Inhibition activity against C. albicans Nmt and human Nmt as assessed by IC50 using myristoyl-CoA (0.5 uM) and peptide substrate GLTISKLFRR-NH2 (0.5 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2011
Entry Details Article
PubMed
TargetGlycylpeptide N-tetradecanoyltransferase 1(Human)
Nippon Roche Research Center

LigandPNGBDBM50121720(CHEMBL355497 | Non peptidic, 5 | (1-METHYL-1H-IMID...)
Affinity DataIC50: 69nMAssay Description:Inhibition activity against C. albicans Nmt and human Nmt as assessed by IC50 using myristoyl-CoA (0.5 uM) and peptide substrate GLTISKLFRR-NH2 (0.5 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2011
Entry Details Article
PubMed
TargetGlycylpeptide N-tetradecanoyltransferase(Yeast)
Nippon Roche Research Center

LigandPNGBDBM43855(N-[4-(3,4,5,6-tetrahydro-2H-azepin-7-ylsulfamoyl)p...)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition activity against C. albicans Nmt and human Nmt as assessed by IC50 using myristoyl-CoA (0.5 uM) and peptide substrate GLTISKLFRR-NH2 (0.5 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2011
Entry Details Article
PubMed
TargetGlycylpeptide N-tetradecanoyltransferase 1(Human)
Nippon Roche Research Center

LigandPNGBDBM43856(cid_3596078 | 4-ethoxy-N-[[6-fluoranyl-1,1-bis(oxi...)
Affinity DataIC50: 8.80E+4nMAssay Description:Inhibition activity against C. albicans Nmt and human Nmt as assessed by IC50 using myristoyl-CoA (0.5 uM) and peptide substrate GLTISKLFRR-NH2 (0.5 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2011
Entry Details Article
PubMed
TargetGlycylpeptide N-tetradecanoyltransferase 1(Human)
Nippon Roche Research Center

LigandPNGBDBM43854(MLS000774113 | 2-[(veratroylhydrazono)methyl]benzo...)
Affinity DataIC50: 1.40E+5nMAssay Description:Inhibition activity against C. albicans Nmt and human Nmt as assessed by IC50 using myristoyl-CoA (0.5 uM) and peptide substrate GLTISKLFRR-NH2 (0.5 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2011
Entry Details Article
PubMed
TargetGlycylpeptide N-tetradecanoyltransferase 1(Human)
Nippon Roche Research Center

LigandPNGBDBM96235(4-[2-hydroxy-3-(propan-2-ylamino)propoxy]-3-methyl...)
Affinity DataIC50: 1.94E+5nMAssay Description:Inhibition activity against C. albicans Nmt and human Nmt as assessed by IC50 using myristoyl-CoA (0.5 uM) and peptide substrate GLTISKLFRR-NH2 (0.5 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2011
Entry Details Article
PubMed
TargetGlycylpeptide N-tetradecanoyltransferase 1(Human)
Nippon Roche Research Center

LigandPNGBDBM43855(N-[4-(3,4,5,6-tetrahydro-2H-azepin-7-ylsulfamoyl)p...)
Affinity DataIC50: 5.70E+5nMAssay Description:Inhibition activity against C. albicans Nmt and human Nmt as assessed by IC50 using myristoyl-CoA (0.5 uM) and peptide substrate GLTISKLFRR-NH2 (0.5 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2011
Entry Details Article
PubMed
TargetGlycylpeptide N-tetradecanoyltransferase(Yeast)
Nippon Roche Research Center

LigandPNGBDBM43856(cid_3596078 | 4-ethoxy-N-[[6-fluoranyl-1,1-bis(oxi...)
Affinity DataKi:  20nMAssay Description:Inhibition activity against C. albicans Nmt and human Nmt as assessed by IC50 using myristoyl-CoA (0.5 uM) and peptide substrate GLTISKLFRR-NH2 (0.5 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2011
Entry Details Article
PubMed
TargetGlycylpeptide N-tetradecanoyltransferase(Yeast)
Nippon Roche Research Center

LigandPNGBDBM43856(cid_3596078 | 4-ethoxy-N-[[6-fluoranyl-1,1-bis(oxi...)
Affinity DataKi:  30nMAssay Description:Inhibition activity against C. albicans Nmt and human Nmt as assessed by IC50 using myristoyl-CoA (0.5 uM) and peptide substrate GLTISKLFRR-NH2 (0.5 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2011
Entry Details Article
PubMed
TargetGlycylpeptide N-tetradecanoyltransferase(Yeast)
Nippon Roche Research Center

LigandPNGBDBM43856(cid_3596078 | 4-ethoxy-N-[[6-fluoranyl-1,1-bis(oxi...)
Affinity DataKi:  30nMAssay Description:Inhibition activity against C. albicans Nmt and human Nmt as assessed by IC50 using myristoyl-CoA (0.5 uM) and peptide substrate GLTISKLFRR-NH2 (0.5 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2011
Entry Details Article
PubMed
TargetGlycylpeptide N-tetradecanoyltransferase(Yeast)
Nippon Roche Research Center

LigandPNGBDBM43856(cid_3596078 | 4-ethoxy-N-[[6-fluoranyl-1,1-bis(oxi...)
Affinity DataKi:  30nMAssay Description:Inhibition activity against C. albicans Nmt and human Nmt as assessed by IC50 using myristoyl-CoA (0.5 uM) and peptide substrate GLTISKLFRR-NH2 (0.5 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2011
Entry Details Article
PubMed
TargetGlycylpeptide N-tetradecanoyltransferase(Yeast)
Nippon Roche Research Center

LigandPNGBDBM43856(cid_3596078 | 4-ethoxy-N-[[6-fluoranyl-1,1-bis(oxi...)
Affinity DataKi:  30nMAssay Description:Inhibition activity against C. albicans Nmt and human Nmt as assessed by IC50 using myristoyl-CoA (0.5 uM) and peptide substrate GLTISKLFRR-NH2 (0.5 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2011
Entry Details Article
PubMed
TargetGlycylpeptide N-tetradecanoyltransferase(Yeast)
Nippon Roche Research Center

LigandPNGBDBM43856(cid_3596078 | 4-ethoxy-N-[[6-fluoranyl-1,1-bis(oxi...)
Affinity DataKi:  30nM IC50: 30nMAssay Description:Inhibition activity against C. albicans Nmt and human Nmt as assessed by IC50 using myristoyl-CoA (0.5 uM) and peptide substrate GLTISKLFRR-NH2 (0.5 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2011
Entry Details Article
PubMed
TargetGlycylpeptide N-tetradecanoyltransferase(Yeast)
Nippon Roche Research Center

LigandPNGBDBM43856(cid_3596078 | 4-ethoxy-N-[[6-fluoranyl-1,1-bis(oxi...)
Affinity DataKi:  40nMAssay Description:Inhibition activity against C. albicans Nmt and human Nmt as assessed by IC50 using myristoyl-CoA (0.5 uM) and peptide substrate GLTISKLFRR-NH2 (0.5 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2011
Entry Details Article
PubMed
TargetGlycylpeptide N-tetradecanoyltransferase(Yeast)
Nippon Roche Research Center

LigandPNGBDBM43856(cid_3596078 | 4-ethoxy-N-[[6-fluoranyl-1,1-bis(oxi...)
Affinity DataKi:  40nMAssay Description:Inhibition activity against C. albicans Nmt and human Nmt as assessed by IC50 using myristoyl-CoA (0.5 uM) and peptide substrate GLTISKLFRR-NH2 (0.5 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2011
Entry Details Article
PubMed
TargetGlycylpeptide N-tetradecanoyltransferase(Yeast)
Nippon Roche Research Center

LigandPNGBDBM96235(4-[2-hydroxy-3-(propan-2-ylamino)propoxy]-3-methyl...)
Affinity DataKi:  50nMAssay Description:Inhibition activity against C. albicans Nmt and human Nmt as assessed by IC50 using myristoyl-CoA (0.5 uM) and peptide substrate GLTISKLFRR-NH2 (0.5 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2011
Entry Details Article
PubMed
TargetGlycylpeptide N-tetradecanoyltransferase(Yeast)
Nippon Roche Research Center

LigandPNGBDBM43856(cid_3596078 | 4-ethoxy-N-[[6-fluoranyl-1,1-bis(oxi...)
Affinity DataKi:  50nMAssay Description:Inhibition activity against C. albicans Nmt and human Nmt as assessed by IC50 using myristoyl-CoA (0.5 uM) and peptide substrate GLTISKLFRR-NH2 (0.5 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2011
Entry Details Article
PubMed
TargetGlycylpeptide N-tetradecanoyltransferase(Yeast)
Nippon Roche Research Center

LigandPNGBDBM43856(cid_3596078 | 4-ethoxy-N-[[6-fluoranyl-1,1-bis(oxi...)
Affinity DataKi:  50nMAssay Description:Inhibition activity against C. albicans Nmt and human Nmt as assessed by IC50 using myristoyl-CoA (0.5 uM) and peptide substrate GLTISKLFRR-NH2 (0.5 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2011
Entry Details Article
PubMed
TargetGlycylpeptide N-tetradecanoyltransferase(Yeast)
Nippon Roche Research Center

LigandPNGBDBM43856(cid_3596078 | 4-ethoxy-N-[[6-fluoranyl-1,1-bis(oxi...)
Affinity DataKi:  70nMAssay Description:Inhibition activity against C. albicans Nmt and human Nmt as assessed by IC50 using myristoyl-CoA (0.5 uM) and peptide substrate GLTISKLFRR-NH2 (0.5 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2011
Entry Details Article
PubMed
TargetGlycylpeptide N-tetradecanoyltransferase(Yeast)
Nippon Roche Research Center

LigandPNGBDBM43856(cid_3596078 | 4-ethoxy-N-[[6-fluoranyl-1,1-bis(oxi...)
Affinity DataKi:  70nMAssay Description:Inhibition activity against C. albicans Nmt and human Nmt as assessed by IC50 using myristoyl-CoA (0.5 uM) and peptide substrate GLTISKLFRR-NH2 (0.5 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2011
Entry Details Article
PubMed
TargetGlycylpeptide N-tetradecanoyltransferase(Yeast)
Nippon Roche Research Center

LigandPNGBDBM43856(cid_3596078 | 4-ethoxy-N-[[6-fluoranyl-1,1-bis(oxi...)
Affinity DataKi:  70nMAssay Description:Inhibition activity against C. albicans Nmt and human Nmt as assessed by IC50 using myristoyl-CoA (0.5 uM) and peptide substrate GLTISKLFRR-NH2 (0.5 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2011
Entry Details Article
PubMed
TargetGlycylpeptide N-tetradecanoyltransferase(Yeast)
Nippon Roche Research Center

LigandPNGBDBM43854(MLS000774113 | 2-[(veratroylhydrazono)methyl]benzo...)
Affinity DataKi:  80nMAssay Description:Inhibition activity against C. albicans Nmt and human Nmt as assessed by IC50 using myristoyl-CoA (0.5 uM) and peptide substrate GLTISKLFRR-NH2 (0.5 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2011
Entry Details Article
PubMed
TargetGlycylpeptide N-tetradecanoyltransferase(Yeast)
Nippon Roche Research Center

LigandPNGBDBM43856(cid_3596078 | 4-ethoxy-N-[[6-fluoranyl-1,1-bis(oxi...)
Affinity DataKi:  90nMAssay Description:Inhibition activity against C. albicans Nmt and human Nmt as assessed by IC50 using myristoyl-CoA (0.5 uM) and peptide substrate GLTISKLFRR-NH2 (0.5 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2011
Entry Details Article
PubMed
TargetGlycylpeptide N-tetradecanoyltransferase(Yeast)
Nippon Roche Research Center

LigandPNGBDBM43856(cid_3596078 | 4-ethoxy-N-[[6-fluoranyl-1,1-bis(oxi...)
Affinity DataKi:  90nMAssay Description:Inhibition activity against C. albicans Nmt and human Nmt as assessed by IC50 using myristoyl-CoA (0.5 uM) and peptide substrate GLTISKLFRR-NH2 (0.5 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2011
Entry Details Article
PubMed
TargetGlycylpeptide N-tetradecanoyltransferase(Yeast)
Nippon Roche Research Center

LigandPNGBDBM43856(cid_3596078 | 4-ethoxy-N-[[6-fluoranyl-1,1-bis(oxi...)
Affinity DataKi:  100nMAssay Description:Inhibition activity against C. albicans Nmt and human Nmt as assessed by IC50 using myristoyl-CoA (0.5 uM) and peptide substrate GLTISKLFRR-NH2 (0.5 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2011
Entry Details Article
PubMed
TargetGlycylpeptide N-tetradecanoyltransferase(Yeast)
Nippon Roche Research Center

LigandPNGBDBM43856(cid_3596078 | 4-ethoxy-N-[[6-fluoranyl-1,1-bis(oxi...)
Affinity DataKi:  110nMAssay Description:Inhibition activity against C. albicans Nmt and human Nmt as assessed by IC50 using myristoyl-CoA (0.5 uM) and peptide substrate GLTISKLFRR-NH2 (0.5 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2011
Entry Details Article
PubMed
TargetGlycylpeptide N-tetradecanoyltransferase(Yeast)
Nippon Roche Research Center

LigandPNGBDBM96235(4-[2-hydroxy-3-(propan-2-ylamino)propoxy]-3-methyl...)
Affinity DataKi:  140nMAssay Description:Inhibition activity against C. albicans Nmt and human Nmt as assessed by IC50 using myristoyl-CoA (0.5 uM) and peptide substrate GLTISKLFRR-NH2 (0.5 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2011
Entry Details Article
PubMed
TargetGlycylpeptide N-tetradecanoyltransferase(Yeast)
Nippon Roche Research Center

LigandPNGBDBM43854(MLS000774113 | 2-[(veratroylhydrazono)methyl]benzo...)
Affinity DataKi:  150nMAssay Description:Inhibition activity against C. albicans Nmt and human Nmt as assessed by IC50 using myristoyl-CoA (0.5 uM) and peptide substrate GLTISKLFRR-NH2 (0.5 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2011
Entry Details Article
PubMed
TargetGlycylpeptide N-tetradecanoyltransferase(Yeast)
Nippon Roche Research Center

LigandPNGBDBM43856(cid_3596078 | 4-ethoxy-N-[[6-fluoranyl-1,1-bis(oxi...)
Affinity DataKi:  150nMAssay Description:Inhibition activity against C. albicans Nmt and human Nmt as assessed by IC50 using myristoyl-CoA (0.5 uM) and peptide substrate GLTISKLFRR-NH2 (0.5 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2011
Entry Details Article
PubMed
TargetGlycylpeptide N-tetradecanoyltransferase(Yeast)
Nippon Roche Research Center

LigandPNGBDBM43854(MLS000774113 | 2-[(veratroylhydrazono)methyl]benzo...)
Affinity DataKi:  180nMAssay Description:Inhibition activity against C. albicans Nmt and human Nmt as assessed by IC50 using myristoyl-CoA (0.5 uM) and peptide substrate GLTISKLFRR-NH2 (0.5 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2011
Entry Details Article
PubMed
TargetGlycylpeptide N-tetradecanoyltransferase(Yeast)
Nippon Roche Research Center

LigandPNGBDBM43854(MLS000774113 | 2-[(veratroylhydrazono)methyl]benzo...)
Affinity DataKi:  200nMAssay Description:Inhibition activity against C. albicans Nmt and human Nmt as assessed by IC50 using myristoyl-CoA (0.5 uM) and peptide substrate GLTISKLFRR-NH2 (0.5 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2011
Entry Details Article
PubMed
TargetGlycylpeptide N-tetradecanoyltransferase(Yeast)
Nippon Roche Research Center

LigandPNGBDBM43856(cid_3596078 | 4-ethoxy-N-[[6-fluoranyl-1,1-bis(oxi...)
Affinity DataKi:  220nMAssay Description:Inhibition activity against C. albicans Nmt and human Nmt as assessed by IC50 using myristoyl-CoA (0.5 uM) and peptide substrate GLTISKLFRR-NH2 (0.5 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2011
Entry Details Article
PubMed
TargetGlycylpeptide N-tetradecanoyltransferase(Yeast)
Nippon Roche Research Center

LigandPNGBDBM43856(cid_3596078 | 4-ethoxy-N-[[6-fluoranyl-1,1-bis(oxi...)
Affinity DataKi:  240nMAssay Description:Inhibition activity against C. albicans Nmt and human Nmt as assessed by IC50 using myristoyl-CoA (0.5 uM) and peptide substrate GLTISKLFRR-NH2 (0.5 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2011
Entry Details Article
PubMed
TargetGlycylpeptide N-tetradecanoyltransferase(Yeast)
Nippon Roche Research Center

LigandPNGBDBM96235(4-[2-hydroxy-3-(propan-2-ylamino)propoxy]-3-methyl...)
Affinity DataKi:  240nMAssay Description:Inhibition activity against C. albicans Nmt and human Nmt as assessed by IC50 using myristoyl-CoA (0.5 uM) and peptide substrate GLTISKLFRR-NH2 (0.5 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2011
Entry Details Article
PubMed
TargetGlycylpeptide N-tetradecanoyltransferase(Yeast)
Nippon Roche Research Center

LigandPNGBDBM43854(MLS000774113 | 2-[(veratroylhydrazono)methyl]benzo...)
Affinity DataKi:  250nMAssay Description:Inhibition activity against C. albicans Nmt and human Nmt as assessed by IC50 using myristoyl-CoA (0.5 uM) and peptide substrate GLTISKLFRR-NH2 (0.5 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2011
Entry Details Article
PubMed
TargetGlycylpeptide N-tetradecanoyltransferase(Yeast)
Nippon Roche Research Center

LigandPNGBDBM43854(MLS000774113 | 2-[(veratroylhydrazono)methyl]benzo...)
Affinity DataKi:  250nM IC50: 830nMAssay Description:Inhibition activity against C. albicans Nmt and human Nmt as assessed by IC50 using myristoyl-CoA (0.5 uM) and peptide substrate GLTISKLFRR-NH2 (0.5 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2011
Entry Details Article
PubMed
TargetGlycylpeptide N-tetradecanoyltransferase(Yeast)
Nippon Roche Research Center

LigandPNGBDBM96235(4-[2-hydroxy-3-(propan-2-ylamino)propoxy]-3-methyl...)
Affinity DataKi:  260nMAssay Description:Inhibition activity against C. albicans Nmt and human Nmt as assessed by IC50 using myristoyl-CoA (0.5 uM) and peptide substrate GLTISKLFRR-NH2 (0.5 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2011
Entry Details Article
PubMed
TargetGlycylpeptide N-tetradecanoyltransferase(Yeast)
Nippon Roche Research Center

LigandPNGBDBM43854(MLS000774113 | 2-[(veratroylhydrazono)methyl]benzo...)
Affinity DataKi:  270nMAssay Description:Inhibition activity against C. albicans Nmt and human Nmt as assessed by IC50 using myristoyl-CoA (0.5 uM) and peptide substrate GLTISKLFRR-NH2 (0.5 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2011
Entry Details Article
PubMed
TargetGlycylpeptide N-tetradecanoyltransferase(Yeast)
Nippon Roche Research Center

LigandPNGBDBM96235(4-[2-hydroxy-3-(propan-2-ylamino)propoxy]-3-methyl...)
Affinity DataKi:  280nMAssay Description:Inhibition activity against C. albicans Nmt and human Nmt as assessed by IC50 using myristoyl-CoA (0.5 uM) and peptide substrate GLTISKLFRR-NH2 (0.5 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2011
Entry Details Article
PubMed
TargetGlycylpeptide N-tetradecanoyltransferase(Yeast)
Nippon Roche Research Center

LigandPNGBDBM43854(MLS000774113 | 2-[(veratroylhydrazono)methyl]benzo...)
Affinity DataKi:  300nMAssay Description:Inhibition activity against C. albicans Nmt and human Nmt as assessed by IC50 using myristoyl-CoA (0.5 uM) and peptide substrate GLTISKLFRR-NH2 (0.5 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2011
Entry Details Article
PubMed
TargetGlycylpeptide N-tetradecanoyltransferase(Yeast)
Nippon Roche Research Center

LigandPNGBDBM43854(MLS000774113 | 2-[(veratroylhydrazono)methyl]benzo...)
Affinity DataKi:  350nMAssay Description:Inhibition activity against C. albicans Nmt and human Nmt as assessed by IC50 using myristoyl-CoA (0.5 uM) and peptide substrate GLTISKLFRR-NH2 (0.5 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2011
Entry Details Article
PubMed
TargetGlycylpeptide N-tetradecanoyltransferase(Yeast)
Nippon Roche Research Center

LigandPNGBDBM96235(4-[2-hydroxy-3-(propan-2-ylamino)propoxy]-3-methyl...)
Affinity DataKi:  360nMAssay Description:Inhibition activity against C. albicans Nmt and human Nmt as assessed by IC50 using myristoyl-CoA (0.5 uM) and peptide substrate GLTISKLFRR-NH2 (0.5 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2011
Entry Details Article
PubMed
TargetGlycylpeptide N-tetradecanoyltransferase(Yeast)
Nippon Roche Research Center

LigandPNGBDBM96235(4-[2-hydroxy-3-(propan-2-ylamino)propoxy]-3-methyl...)
Affinity DataKi:  390nMAssay Description:Inhibition activity against C. albicans Nmt and human Nmt as assessed by IC50 using myristoyl-CoA (0.5 uM) and peptide substrate GLTISKLFRR-NH2 (0.5 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2011
Entry Details Article
PubMed
TargetGlycylpeptide N-tetradecanoyltransferase(Yeast)
Nippon Roche Research Center

LigandPNGBDBM96235(4-[2-hydroxy-3-(propan-2-ylamino)propoxy]-3-methyl...)
Affinity DataKi:  420nMAssay Description:Inhibition activity against C. albicans Nmt and human Nmt as assessed by IC50 using myristoyl-CoA (0.5 uM) and peptide substrate GLTISKLFRR-NH2 (0.5 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2011
Entry Details Article
PubMed
TargetGlycylpeptide N-tetradecanoyltransferase(Yeast)
Nippon Roche Research Center

LigandPNGBDBM96235(4-[2-hydroxy-3-(propan-2-ylamino)propoxy]-3-methyl...)
Affinity DataKi:  450nMAssay Description:Inhibition activity against C. albicans Nmt and human Nmt as assessed by IC50 using myristoyl-CoA (0.5 uM) and peptide substrate GLTISKLFRR-NH2 (0.5 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2011
Entry Details Article
PubMed
TargetGlycylpeptide N-tetradecanoyltransferase(Yeast)
Nippon Roche Research Center

LigandPNGBDBM96235(4-[2-hydroxy-3-(propan-2-ylamino)propoxy]-3-methyl...)
Affinity DataKi:  450nMAssay Description:Inhibition activity against C. albicans Nmt and human Nmt as assessed by IC50 using myristoyl-CoA (0.5 uM) and peptide substrate GLTISKLFRR-NH2 (0.5 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2011
Entry Details Article
PubMed
TargetGlycylpeptide N-tetradecanoyltransferase(Yeast)
Nippon Roche Research Center

LigandPNGBDBM96235(4-[2-hydroxy-3-(propan-2-ylamino)propoxy]-3-methyl...)
Affinity DataKi:  450nMAssay Description:Inhibition activity against C. albicans Nmt and human Nmt as assessed by IC50 using myristoyl-CoA (0.5 uM) and peptide substrate GLTISKLFRR-NH2 (0.5 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2011
Entry Details Article
PubMed
TargetGlycylpeptide N-tetradecanoyltransferase(Yeast)
Nippon Roche Research Center

LigandPNGBDBM43856(cid_3596078 | 4-ethoxy-N-[[6-fluoranyl-1,1-bis(oxi...)
Affinity DataKi:  460nMAssay Description:Inhibition activity against C. albicans Nmt and human Nmt as assessed by IC50 using myristoyl-CoA (0.5 uM) and peptide substrate GLTISKLFRR-NH2 (0.5 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2011
Entry Details Article
PubMed
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