Compile Data Set for Download or QSAR
Report error Found 23 Enz. Inhib. hit(s) with all data for entry = 50035246
TargetMelanocyte-stimulating hormone receptor(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50116866(Bu-His-DPhe-Arg(CN)-Trp-Gly-NH2 | CHEMBL311750)
Affinity DataEC50:  15nMAssay Description:Agonist potency for human Melanocortin 1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50116867((S)-2-{(R)-2-[(S)-2-Butylamino-3-(3H-imidazol-4-yl...)
Affinity DataEC50:  950nMAssay Description:Agonist potency for human Melanocortin 1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50116868((S)-2-{(R)-2-[(S)-2-Butylamino-3-(3H-imidazol-4-yl...)
Affinity DataEC50:  350nMAssay Description:Agonist potency for human Melanocortin 1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50116864((S)-2-{(R)-2-[(S)-2-Butylamino-3-(3H-imidazol-4-yl...)
Affinity DataEC50:  1.67E+3nMAssay Description:Agonist potency towards human Melanocortin 4 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50116873((S)-2-{(R)-2-[(S)-2-Butylamino-3-(3H-imidazol-4-yl...)
Affinity DataEC50:  20nMAssay Description:Agonist potency towards human Melanocortin 4 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50116874((S)-2-{(R)-2-[(S)-2-Butylamino-3-(3H-imidazol-4-yl...)
Affinity DataEC50:  1nMAssay Description:Agonist potency for human Melanocortin 1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50116874((S)-2-{(R)-2-[(S)-2-Butylamino-3-(3H-imidazol-4-yl...)
Affinity DataEC50:  10nMAssay Description:Agonist potency towards human Melanocortin 4 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50116865((S)-5-Amino-2-{(R)-2-[(S)-2-butylamino-3-(3H-imida...)
Affinity DataEC50:  900nMAssay Description:Agonist potency for human Melanocortin 1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50116873((S)-2-{(R)-2-[(S)-2-Butylamino-3-(3H-imidazol-4-yl...)
Affinity DataEC50:  10nMAssay Description:Agonist potency for human Melanocortin 1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50116870((S)-2-Butylamino-N-{(R)-1-[(S)-1-[(S)-1-(carbamoyl...)
Affinity DataEC50:  1.70E+3nMAssay Description:Agonist potency for human Melanocortin 1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50029747((4S)-4-{[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-[({[(2S...)
Affinity DataEC50:  0.800nMAssay Description:Agonist potency for human Melanocortin 1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50116872((S)-2-{(R)-2-[(S)-2-Butylamino-3-(3H-imidazol-4-yl...)
Affinity DataEC50:  255nMAssay Description:Agonist potency for human Melanocortin 1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM82411(CAS_75921-69-6 | NDP-MSH)
Affinity DataEC50:  0.5nMAssay Description:Agonist potency for human Melanocortin 1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50029747((4S)-4-{[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-[({[(2S...)
Affinity DataEC50:  25nMAssay Description:Agonist potency towards human Melanocortin 4 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50116870((S)-2-Butylamino-N-{(R)-1-[(S)-1-[(S)-1-(carbamoyl...)
Affinity DataEC50:  1.42E+3nMAssay Description:Agonist potency towards human Melanocortin 4 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50116869((S)-6-Benzylamino-2-{(R)-2-[(S)-2-butylamino-3-(3H...)
Affinity DataEC50:  85nMAssay Description:Agonist potency for human Melanocortin 1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50116869((S)-6-Benzylamino-2-{(R)-2-[(S)-2-butylamino-3-(3H...)
Affinity DataEC50:  4.80E+3nMAssay Description:Agonist potency towards human Melanocortin 4 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50116868((S)-2-{(R)-2-[(S)-2-Butylamino-3-(3H-imidazol-4-yl...)
Affinity DataEC50:  3.28E+3nMAssay Description:Agonist potency towards human Melanocortin 4 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50116867((S)-2-{(R)-2-[(S)-2-Butylamino-3-(3H-imidazol-4-yl...)
Affinity DataEC50:  760nMAssay Description:Agonist potency towards human Melanocortin 4 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50116866(Bu-His-DPhe-Arg(CN)-Trp-Gly-NH2 | CHEMBL311750)
Affinity DataEC50:  70nMAssay Description:Agonist potency towards human Melanocortin 4 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50116865((S)-5-Amino-2-{(R)-2-[(S)-2-butylamino-3-(3H-imida...)
Affinity DataEC50:  2.50E+3nMAssay Description:Agonist potency towards human Melanocortin 4 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50116864((S)-2-{(R)-2-[(S)-2-Butylamino-3-(3H-imidazol-4-yl...)
Affinity DataEC50:  60nMAssay Description:Agonist potency for human Melanocortin 1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM82411(CAS_75921-69-6 | NDP-MSH)
Affinity DataEC50:  1nMAssay Description:Agonist potency towards human Melanocortin 4 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed