Compile Data Set for Download or QSAR
Report error Found 24 Enz. Inhib. hit(s) with all data for entry = 50037050
TargetKappa-type opioid receptor(Guinea pig)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM82551(C18130 | CAS_105618-26-6 | NORBNI | NOR-BNI (HCI)2)
Affinity DataKi:  1.09nMAssay Description:Ability to displace [3H]U-69593 from Opioid receptor kappa 1 of guinea pig brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50116621(3-[7-Amino-4-methyl-2-(3-phenyl-propyl)-2-aza-bicy...)
Affinity DataKi:  3.30nMAssay Description:Ability to displace [3H]DAMGO from Opioid receptor mu 1 of rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50116622(N-[5-(3-Hydroxy-phenyl)-4-methyl-2-phenethyl-2-aza...)
Affinity DataKi:  4.30nMAssay Description:Ability to displace [3H]U-69593 from Opioid receptor kappa 1 of guinea pig brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50116624(3-Guanidino-N-[5-(3-hydroxy-phenyl)-4-methyl-2-phe...)
Affinity DataKi:  5.20nMAssay Description:Ability to displace [3H]DAMGO from Opioid receptor mu 1 of rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50116623(4-Dimethylamino-N-[5-(3-hydroxy-phenyl)-4-methyl-2...)
Affinity DataKi:  12nMAssay Description:Ability to displace [3H]U-69593 from Opioid receptor kappa 1 of guinea pig brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50116620(4-Guanidino-N-[5-(3-hydroxy-phenyl)-4-methyl-2-phe...)
Affinity DataKi:  13.2nMAssay Description:Ability to displace [3H]U-69593 from Opioid receptor kappa 1 of guinea pig brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50116621(3-[7-Amino-4-methyl-2-(3-phenyl-propyl)-2-aza-bicy...)
Affinity DataKi:  14.7nMAssay Description:Ability to displace [3H]DADLE from Opioid receptor delta 1 of rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50116624(3-Guanidino-N-[5-(3-hydroxy-phenyl)-4-methyl-2-phe...)
Affinity DataKi:  23.3nMAssay Description:Ability to displace [3H]U-69593 from Opioid receptor kappa 1 of guinea pig brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50116622(N-[5-(3-Hydroxy-phenyl)-4-methyl-2-phenethyl-2-aza...)
Affinity DataKi:  36nMAssay Description:Ability to displace [3H]U-69593 from Opioid receptor kappa 1 of guinea pig brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50116624(3-Guanidino-N-[5-(3-hydroxy-phenyl)-4-methyl-2-phe...)
Affinity DataKi:  56.5nMAssay Description:Ability to displace [3H]DADLE from Opioid receptor delta 1 of rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50116623(4-Dimethylamino-N-[5-(3-hydroxy-phenyl)-4-methyl-2...)
Affinity DataKi:  57nMAssay Description:Ability to displace [3H]DAMGO from Opioid receptor mu 1 of rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM82551(C18130 | CAS_105618-26-6 | NORBNI | NOR-BNI (HCI)2)
Affinity DataKi:  65nMAssay Description:Ability to displace [3H]DAMGO from Opioid receptor mu 1 of rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM82551(C18130 | CAS_105618-26-6 | NORBNI | NOR-BNI (HCI)2)
Affinity DataKi:  86nMAssay Description:Ability to displace [3H]DADLE from Opioid receptor delta 1 of rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50116620(4-Guanidino-N-[5-(3-hydroxy-phenyl)-4-methyl-2-phe...)
Affinity DataKi:  87nMAssay Description:Ability to displace [3H]DAMGO from Opioid receptor mu 1 of rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50116621(3-[7-Amino-4-methyl-2-(3-phenyl-propyl)-2-aza-bicy...)
Affinity DataKi:  122nMAssay Description:Ability to displace [3H]U-69593 from Opioid receptor kappa 1 of guinea pig brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50116622(N-[5-(3-Hydroxy-phenyl)-4-methyl-2-phenethyl-2-aza...)
Affinity DataKi:  147nMAssay Description:Ability to displace [3H]DAMGO from Opioid receptor mu 1 of rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50116621(3-[7-Amino-4-methyl-2-(3-phenyl-propyl)-2-aza-bicy...)
Affinity DataKi:  207nMAssay Description:Ability to displace [3H]DAMGO from Opioid receptor mu 1 of rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50116621(3-[7-Amino-4-methyl-2-(3-phenyl-propyl)-2-aza-bicy...)
Affinity DataKi:  246nMAssay Description:Ability to displace [3H]DADLE from Opioid receptor delta 1 of rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50116622(N-[5-(3-Hydroxy-phenyl)-4-methyl-2-phenethyl-2-aza...)
Affinity DataKi:  775nMAssay Description:Ability to displace [3H]DAMGO from Opioid receptor mu 1 of rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50116621(3-[7-Amino-4-methyl-2-(3-phenyl-propyl)-2-aza-bicy...)
Affinity DataKi:  893nMAssay Description:Ability to displace [3H]U-69593 from Opioid receptor kappa 1 of guinea pig brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50116623(4-Dimethylamino-N-[5-(3-hydroxy-phenyl)-4-methyl-2...)
Affinity DataKi:  1.46E+3nMAssay Description:Ability to displace [3H]DADLE from Opioid receptor delta 1 of rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50116620(4-Guanidino-N-[5-(3-hydroxy-phenyl)-4-methyl-2-phe...)
Affinity DataKi:  1.74E+3nMAssay Description:Ability to displace [3H]DADLE from Opioid receptor delta 1 of rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50116622(N-[5-(3-Hydroxy-phenyl)-4-methyl-2-phenethyl-2-aza...)
Affinity DataKi:  2.18E+3nMAssay Description:Ability to displace [3H]DADLE from Opioid receptor delta 1 of rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50116622(N-[5-(3-Hydroxy-phenyl)-4-methyl-2-phenethyl-2-aza...)
Affinity DataKi: >3.40E+3nMAssay Description:Ability to displace [3H]DADLE from Opioid receptor delta 1 of rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed