Compile Data Set for Download or QSAR
Report error Found 34 Enz. Inhib. hit(s) with all data for entry = 50012247
TargetNeuropeptide Y receptor type 5(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50116590(N-(9-Methanesulfonyl-9H-carbazol-3-yl)-3-pyridin-4...)
Affinity DataIC50: 1nMAssay Description:Binding affinity to the human Neuropeptide Y receptor Y5 (NPY5)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50116610(N-(9-Isopropyl-9H-carbazol-3-yl)-3-pyridin-4-yl-pr...)
Affinity DataIC50: 1nMAssay Description:Binding affinity to the human Neuropeptide Y receptor Y5 (NPY5)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50116619(Morpholine-4-carboxylic acid (9-isopropyl-8-methyl...)
Affinity DataIC50: 2nMAssay Description:Binding affinity to the human Neuropeptide Y receptor Y5 (NPY5)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50116602(Morpholine-4-carboxylic acid (9-isopropyl-9H-carba...)
Affinity DataIC50: 2nMAssay Description:Binding affinity to the human Neuropeptide Y receptor Y5 (NPY5)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50116600(N-(9-Ethyl-9H-carbazol-3-yl)-3-pyridin-4-yl-propio...)
Affinity DataIC50: 2nMAssay Description:Binding affinity to the human Neuropeptide Y receptor Y5 (NPY5)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50116617(N-(9-Acetyl-9H-carbazol-3-yl)-3-pyridin-4-yl-propi...)
Affinity DataIC50: 3nMAssay Description:Binding affinity to the human Neuropeptide Y receptor Y5 (NPY5)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50116605(Morpholine-4-carboxylic acid (6-fluoro-9-isopropyl...)
Affinity DataIC50: 3nMAssay Description:Binding affinity to the human Neuropeptide Y receptor Y5 (NPY5)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50116592(Morpholine-4-carboxylic acid (9-isopropyl-4-methyl...)
Affinity DataIC50: 3nMAssay Description:Binding affinity to the human Neuropeptide Y receptor Y5 (NPY5)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50116592(Morpholine-4-carboxylic acid (9-isopropyl-4-methyl...)
Affinity DataIC50: 6nMAssay Description:Compound was evaluated for functional antagonism of Neuropeptide Y receptor Y5 activity in cellular Ca fluxMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 5(Rat)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50116600(N-(9-Ethyl-9H-carbazol-3-yl)-3-pyridin-4-yl-propio...)
Affinity DataIC50: 7nMAssay Description:Binding affinity against rat Neuropeptide Y receptor Y5More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50116597(Morpholine-4-carboxylic acid (9-ethyl-9H-carbazol-...)
Affinity DataIC50: 7nMAssay Description:Binding affinity to the human Neuropeptide Y receptor Y5 (NPY5)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50116608(N-(9-Dimethylsulfamoyl-9H-carbazol-3-yl)-3-pyridin...)
Affinity DataIC50: 8nMAssay Description:Binding affinity to the human Neuropeptide Y receptor Y5 (NPY5)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50116600(N-(9-Ethyl-9H-carbazol-3-yl)-3-pyridin-4-yl-propio...)
Affinity DataIC50: 11nMAssay Description:In vitro human Neuropeptide Y receptor Y5 functional antagonism (reporter gene assay)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50116607(Morpholine-4-carboxylic acid (2,4-difluoro-9-isopr...)
Affinity DataIC50: 12nMAssay Description:Binding affinity to the human Neuropeptide Y receptor Y5 (NPY5)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50116603(Morpholine-4-carboxylic acid (9-methanesulfonyl-9H...)
Affinity DataIC50: 15nMAssay Description:Binding affinity to the human Neuropeptide Y receptor Y5 (NPY5)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50116612(N-(9-Methyl-9H-carbazol-3-yl)-3-pyridin-4-yl-propi...)
Affinity DataIC50: 33nMAssay Description:Binding affinity to the human Neuropeptide Y receptor Y5 (NPY5)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50116592(Morpholine-4-carboxylic acid (9-isopropyl-4-methyl...)
Affinity DataIC50: 37nMAssay Description:The compound was evaluated in vitro for: human Neuropeptide Y receptor Y5 functional antagonismMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50116618(Morpholine-4-carboxylic acid [9-(tetrahydro-furan-...)
Affinity DataIC50: 40nMAssay Description:Binding affinity to the human Neuropeptide Y receptor Y5 (NPY5)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50116609(Morpholine-4-carboxylic acid [9-(2,2-dimethyl-prop...)
Affinity DataIC50: 78nMAssay Description:Binding affinity to the human Neuropeptide Y receptor Y5 (NPY5)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50116613(N-(9H-Carbazol-3-yl)-3-pyridin-4-yl-propionamide |...)
Affinity DataIC50: 230nMAssay Description:Binding affinity to the human Neuropeptide Y receptor Y5 (NPY5)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50116594(Morpholine-4-carboxylic acid (4-ethoxy-9-isopropyl...)
Affinity DataIC50: 270nMAssay Description:Binding affinity to the human Neuropeptide Y receptor Y5 (NPY5)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50116604(N-(4-Benzoyl-phenyl)-3-pyridin-4-yl-propionamide |...)
Affinity DataIC50: 300nMAssay Description:Binding affinity to the human Neuropeptide Y receptor Y5 (NPY5)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50116615(Morpholine-4-carboxylic acid (9-dimethylsulfamoyl-...)
Affinity DataIC50: 350nMAssay Description:Binding affinity to the human Neuropeptide Y receptor Y5 (NPY5)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50116598(N-(4-Benzoyl-phenyl)-2-(pyridin-4-ylsulfanyl)-acet...)
Affinity DataIC50: 350nMAssay Description:Binding affinity to the human Neuropeptide Y receptor Y5 (NPY5)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50116599(Morpholine-4-carboxylic acid (9-isopropyl-2,4-dime...)
Affinity DataIC50: 390nMAssay Description:Binding affinity to the human Neuropeptide Y receptor Y5 (NPY5)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50116616(N-(9-Ethyl-9H-carbazol-1-yl)-3-pyridin-4-yl-propio...)
Affinity DataIC50: 440nMAssay Description:Binding affinity to the human Neuropeptide Y receptor Y5 (NPY5)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50116606(9-Ethyl-9H-carbazole-3-carboxylic acid (2-pyridin-...)
Affinity DataIC50: 700nMAssay Description:Binding affinity to the human Neuropeptide Y receptor Y5 (NPY5)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50116611(Morpholine-4-carboxylic acid (9-isopropyl-1,4-dime...)
Affinity DataIC50: 710nMAssay Description:Binding affinity to the human Neuropeptide Y receptor Y5 (NPY5)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50116601(Morpholine-4-carboxylic acid (4,9-diisopropyl-9H-c...)
Affinity DataIC50: 770nMAssay Description:Binding affinity to the human Neuropeptide Y receptor Y5 (NPY5)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50116593(N-(9-Ethyl-9H-carbazol-2-yl)-3-pyridin-4-yl-propio...)
Affinity DataIC50: 800nMAssay Description:Binding affinity to the human Neuropeptide Y receptor Y5 (NPY5)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50116595(N-(9-Ethyl-9H-carbazol-3-yl)-N-methyl-3-pyridin-4-...)
Affinity DataIC50: 2.20E+3nMAssay Description:Binding affinity to the human Neuropeptide Y receptor Y5 (NPY5)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50116591(2-(9-Ethyl-9H-carbazol-3-yl)-N-pyridin-4-ylmethyl-...)
Affinity DataIC50: 2.25E+3nMAssay Description:Binding affinity to the human Neuropeptide Y receptor Y5 (NPY5)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50116614(N-(9-Ethyl-9H-carbazol-3-ylmethyl)-2-pyridin-4-yl-...)
Affinity DataIC50: 3.40E+3nMAssay Description:Binding affinity to the human Neuropeptide Y receptor Y5 (NPY5)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50116596(N-(9-Ethyl-9H-carbazol-4-yl)-3-pyridin-4-yl-propio...)
Affinity DataIC50: 1.00E+4nMAssay Description:Binding affinity to the human Neuropeptide Y receptor Y5 (NPY5)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed