Compile Data Set for Download or QSAR
Report error Found 29 Enz. Inhib. hit(s) with all data for entry = 50003617
TargetSubstance-K receptor(Human)
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Curated by ChEMBL
LigandPNGBDBM50472916(CHEMBL223221 | MEN-11690)
Affinity DataKi:  0.100nMAssay Description:Inhibitory affinity constant (pKi) against tachykinin receptor 2 (NK-2R) using heterologous competition experimentsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetSubstance-K receptor(Human)
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Curated by ChEMBL
LigandPNGBDBM50473829(MEN-11995 | CHEMBL389459)
Affinity DataKi:  0.158nMAssay Description:Inhibitory affinity constant (pKi) against tachykinin receptor 2 (NK-2R) using heterologous competition experimentsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetSubstance-K receptor(Human)
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Curated by ChEMBL
LigandPNGBDBM50473828(MEN-11990 | CHEMBL116812)
Affinity DataKi:  0.316nMAssay Description:Inhibitory affinity constant (pKi) against tachykinin receptor 2 (NK-2R) using heterologous competition experimentsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetSubstance-K receptor(Human)
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Curated by ChEMBL
LigandPNGBDBM50473824(MEN-11959 | CHEMBL406024)
Affinity DataKi:  0.398nMAssay Description:Inhibitory affinity constant (pKi) against tachykinin receptor 2 (NK-2R) using heterologous competition experimentsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetSubstance-K receptor(Human)
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Curated by ChEMBL
LigandPNGBDBM50473818(MEN-11842 | CHEMBL406287)
Affinity DataKi:  0.794nMAssay Description:Inhibitory affinity constant (pKi) against tachykinin receptor 2 (NK-2R) using heterologous competition experimentsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetSubstance-K receptor(Human)
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Curated by ChEMBL
LigandPNGBDBM50473833(MEN-11830 | CHEMBL420859)
Affinity DataKi:  1.60nMAssay Description:Inhibitory affinity constant (pKi) against tachykinin receptor 2 (NK-2R) using heterologous competition experimentsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetSubstance-K receptor(Human)
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Curated by ChEMBL
LigandPNGBDBM50472917(CHEMBL323884 | MEN-11749)
Affinity DataKi:  1.60nMAssay Description:Inhibitory affinity constant (pKi) against tachykinin receptor 2 (NK-2R) using heterologous competition experimentsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetSubstance-K receptor(Human)
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Curated by ChEMBL
LigandPNGBDBM50404020(MEN-11558 | CHEMBL435324)
Affinity DataKi:  2nMAssay Description:Inhibitory affinity constant (pKi) against tachykinin receptor 2 (NK-2R) using heterologous competition experimentsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetSubstance-K receptor(Human)
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Curated by ChEMBL
LigandPNGBDBM50473823(MEN-11691 | CHEMBL420308)
Affinity DataKi:  3.20nMAssay Description:Inhibitory affinity constant (pKi) against tachykinin receptor 2 (NK-2R) using heterologous competition experimentsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetSubstance-K receptor(Human)
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Curated by ChEMBL
LigandPNGBDBM50473822(MEN-11799 | CHEMBL438559)
Affinity DataKi:  3.20nMAssay Description:Inhibitory affinity constant (pKi) against tachykinin receptor 2 (NK-2R) using heterologous competition experimentsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetSubstance-K receptor(Human)
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Curated by ChEMBL
LigandPNGBDBM50473830(MEN-11703 | CHEMBL323677)
Affinity DataKi:  3.20nMAssay Description:Inhibitory affinity constant (pKi) against tachykinin receptor 2 (NK-2R) using heterologous competition experimentsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetSubstance-K receptor(Human)
Menarini Ricerche

Curated by ChEMBL
LigandPNGBDBM50473836(MEN-11701 | CHEMBL324313)
Affinity DataKi:  3.20nMAssay Description:Inhibitory affinity constant (pKi) against tachykinin receptor 2 (NK-2R) using heterologous competition experimentsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetSubstance-K receptor(Human)
Menarini Ricerche

Curated by ChEMBL
LigandPNGBDBM50473839(MEN-11987 | CHEMBL116871)
Affinity DataKi:  4nMAssay Description:Inhibitory affinity constant (pKi) against tachykinin receptor 2 (NK-2R) using heterologous competition experimentsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetSubstance-K receptor(Human)
Menarini Ricerche

Curated by ChEMBL
LigandPNGBDBM50473821(MEN-11986 | CHEMBL114068)
Affinity DataKi:  4nMAssay Description:Inhibitory affinity constant (pKi) against tachykinin receptor 2 (NK-2R) using heterologous competition experimentsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetSubstance-K receptor(Human)
Menarini Ricerche

Curated by ChEMBL
LigandPNGBDBM50473825(MEN-11983 | CHEMBL113765)
Affinity DataKi:  5nMAssay Description:Inhibitory affinity constant (pKi) against tachykinin receptor 2 (NK-2R) using heterologous competition experimentsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetSubstance-K receptor(Human)
Menarini Ricerche

Curated by ChEMBL
LigandPNGBDBM50473831(MEN-11757 | CHEMBL432986)
Affinity DataKi:  6.30nMAssay Description:Inhibitory affinity constant (pKi) against tachykinin receptor 2 (NK-2R) using heterologous competition experimentsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetSubstance-K receptor(Human)
Menarini Ricerche

Curated by ChEMBL
LigandPNGBDBM50472912(CHEMBL116564 | MEN-11712)
Affinity DataKi:  7.90nMAssay Description:Inhibitory affinity constant (pKi) against tachykinin receptor 2 (NK-2R) using heterologous competition experimentsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetSubstance-K receptor(Human)
Menarini Ricerche

Curated by ChEMBL
LigandPNGBDBM50473837(MEN-11877 | CHEMBL324532)
Affinity DataKi:  7.90nMAssay Description:Inhibitory affinity constant (pKi) against tachykinin receptor 2 (NK-2R) using heterologous competition experimentsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetSubstance-K receptor(Human)
Menarini Ricerche

Curated by ChEMBL
LigandPNGBDBM50473838(MEN-11708 | CHEMBL116629)
Affinity DataKi:  10nMAssay Description:Inhibitory affinity constant (pKi) against tachykinin receptor 2 (NK-2R) using heterologous competition experimentsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetSubstance-K receptor(Human)
Menarini Ricerche

Curated by ChEMBL
LigandPNGBDBM50473832(MEN-11755 | CHEMBL116969)
Affinity DataKi:  13nMAssay Description:Inhibitory affinity constant (pKi) against tachykinin receptor 2 (NK-2R) using heterologous competition experimentsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetSubstance-K receptor(Human)
Menarini Ricerche

Curated by ChEMBL
LigandPNGBDBM50473827(MEN-11668 | CHEMBL323836)
Affinity DataKi:  13nMAssay Description:Inhibitory affinity constant (pKi) against tachykinin receptor 2 (NK-2R) using heterologous competition experimentsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetSubstance-K receptor(Human)
Menarini Ricerche

Curated by ChEMBL
LigandPNGBDBM50473834(MEN-11733 | CHEMBL324106)
Affinity DataKi:  316nMAssay Description:Inhibitory affinity constant (pKi) against tachykinin receptor 2 (NK-2R) using heterologous competition experimentsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetSubstance-K receptor(Human)
Menarini Ricerche

Curated by ChEMBL
LigandPNGBDBM50472914(CHEMBL114442 | MEN-11667)
Affinity DataKi:  316nMAssay Description:Inhibitory affinity constant (pKi) against tachykinin receptor 2 (NK-2R) using heterologous competition experimentsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetSubstance-K receptor(Human)
Menarini Ricerche

Curated by ChEMBL
LigandPNGBDBM50473826(MEN-11715 | CHEMBL116855)
Affinity DataKi:  316nMAssay Description:Inhibitory affinity constant (pKi) against tachykinin receptor 2 (NK-2R) using heterologous competition experimentsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetSubstance-K receptor(Human)
Menarini Ricerche

Curated by ChEMBL
LigandPNGBDBM50473820(MEN-11716 | CHEMBL117039)
Affinity DataKi:  398nMAssay Description:Inhibitory affinity constant (pKi) against tachykinin receptor 2 (NK-2R) using heterologous competition experimentsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetSubstance-K receptor(Human)
Menarini Ricerche

Curated by ChEMBL
LigandPNGBDBM50473819(MEN-11532 | CHEMBL326790)
Affinity DataKi:  631nMAssay Description:Inhibitory affinity constant (pKi) against tachykinin receptor 2 (NK-2R) using heterologous competition experimentsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetSubstance-K receptor(Human)
Menarini Ricerche

Curated by ChEMBL
LigandPNGBDBM50472915(CHEMBL114036 | MEN-11540)
Affinity DataKi:  794nMAssay Description:Inhibitory affinity constant (pKi) against tachykinin receptor 2 (NK-2R) using heterologous competition experimentsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetSubstance-K receptor(Human)
Menarini Ricerche

Curated by ChEMBL
LigandPNGBDBM50472918(CHEMBL324804 | MEN-11970)
Affinity DataKi:  1.26E+3nMAssay Description:Inhibitory affinity constant (pKi) against tachykinin receptor 2 (NK-2R) using heterologous competition experimentsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetSubstance-K receptor(Human)
Menarini Ricerche

Curated by ChEMBL
LigandPNGBDBM50473835(MEN-11523 | CHEMBL420685)
Affinity DataKi:  3.98E+3nMAssay Description:Inhibitory affinity constant (pKi) against tachykinin receptor 2 (NK-2R) using heterologous competition experimentsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed