Compile Data Set for Download or QSAR
Report error Found 28 Enz. Inhib. hit(s) with all data for entry = 50012198
TargetSubstance-P receptor(Human)
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM50115967(2-[(3,5-Bis-trifluoromethyl-benzoyl)-methyl-amino]...)
Affinity DataIC50: 0.600nMAssay Description:inhibition of [3H]Sar-SP binding to Tachykinin receptor 1 of bovine retina membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSubstance-P receptor(Human)
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM50115966(4'-Chloro-2-(3,4,5-trimethoxy-benzoylamino)-biphen...)
Affinity DataIC50: 0.700nMAssay Description:inhibition of [3H]Sar-SP binding to Tachykinin receptor 1 of bovine retina membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSubstance-P receptor(Human)
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM50403920(CHEMBL2112212)
Affinity DataIC50: 0.800nMAssay Description:inhibition of [3H]Sar-SP binding to Tachykinin receptor 1 of bovine retina membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSubstance-P receptor(Human)
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM50403918(CHEMBL2113739)
Affinity DataIC50: 1nMAssay Description:inhibition of [3H]Sar-SP binding to Tachykinin receptor 1 of bovine retina membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSubstance-P receptor(Human)
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM50115965(2-[(3,5-Bis-trifluoromethyl-benzoyl)-methyl-amino]...)
Affinity DataIC50: 1nMAssay Description:inhibition of [3H]Sar-SP binding to Tachykinin receptor 1 of bovine retina membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSubstance-P receptor(Human)
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM50115959(2-[(3,5-Bis-trifluoromethyl-benzoyl)-methyl-amino]...)
Affinity DataIC50: 1.5nMAssay Description:inhibition of [3H]Sar-SP binding to Tachykinin receptor 1 of bovine retina membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSubstance-P receptor(Human)
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM50403916(CHEMBL2113740)
Affinity DataIC50: 2.70nMAssay Description:inhibition of [3H]Sar-SP binding to Tachykinin receptor 1 of bovine retina membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSubstance-P receptor(Human)
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM50115957(2-[(3,5-Bis-trifluoromethyl-benzoyl)-methyl-amino]...)
Affinity DataIC50: 3nMAssay Description:inhibition of [3H]Sar-SP binding to Tachykinin receptor 1 of bovine retina membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSubstance-P receptor(Human)
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM50115969(N-[4-(N-Cyclohexyl-hydrazinocarbonyl)-4'-fluoro-bi...)
Affinity DataIC50: 3.5nMAssay Description:inhibition of [3H]Sar-SP binding to Tachykinin receptor 1 of bovine retina membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSubstance-P receptor(Human)
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM50115964(2-[(3,5-Bis-trifluoromethyl-benzoyl)-methyl-amino]...)
Affinity DataIC50: 4nMAssay Description:inhibition of [3H]Sar-SP binding to Tachykinin receptor 1 of bovine retina membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSubstance-P receptor(Human)
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM50403919(CHEMBL2112211)
Affinity DataIC50: 6nMAssay Description:inhibition of [3H]Sar-SP binding to Tachykinin receptor 1 of bovine retina membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSubstance-P receptor(Human)
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM50115970(N-[4'-Chloro-4-(2-cyclohexylamino-acetyl)-biphenyl...)
Affinity DataIC50: 9nMAssay Description:inhibition of [3H]Sar-SP binding to Tachykinin receptor 1 of bovine retina membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSubstance-P receptor(Human)
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM50403917(CHEMBL2112209)
Affinity DataIC50: 13nMAssay Description:inhibition of [3H]Sar-SP binding to Tachykinin receptor 1 of bovine retina membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSubstance-K receptor(Human)
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM50403918(CHEMBL2113739)
Affinity DataIC50: 28nMAssay Description:Binding affinity was determined by measuring the inhibition of 125 I-NKA binding to transfected CHO cells expressing human recombinant Tachykinin rec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSubstance-K receptor(Human)
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM50115970(N-[4'-Chloro-4-(2-cyclohexylamino-acetyl)-biphenyl...)
Affinity DataIC50: 30nMAssay Description:Binding affinity was determined by measuring the inhibition of 125 I-NKA binding to transfected CHO cells expressing human recombinant Tachykinin rec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSubstance-P receptor(Human)
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM50115963(2-[(3,5-Bis-trifluoromethyl-benzoyl)-methyl-amino]...)
Affinity DataIC50: 34nMAssay Description:inhibition of [3H]Sar-SP binding to Tachykinin receptor 1 of bovine retina membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSubstance-K receptor(Human)
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM50403920(CHEMBL2112212)
Affinity DataIC50: 43nMAssay Description:Binding affinity was determined by measuring the inhibition of 125 I-NKA binding to transfected CHO cells expressing human recombinant Tachykinin rec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSubstance-K receptor(Human)
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM50115957(2-[(3,5-Bis-trifluoromethyl-benzoyl)-methyl-amino]...)
Affinity DataIC50: 51nMAssay Description:Binding affinity was determined by measuring the inhibition of 125 I-NKA binding to transfected CHO cells expressing human recombinant Tachykinin rec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSubstance-K receptor(Human)
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM50403916(CHEMBL2113740)
Affinity DataIC50: 70nMAssay Description:Binding affinity was determined by measuring the inhibition of 125 I-NKA binding to transfected CHO cells expressing human recombinant Tachykinin rec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSubstance-K receptor(Human)
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM50115965(2-[(3,5-Bis-trifluoromethyl-benzoyl)-methyl-amino]...)
Affinity DataIC50: 108nMAssay Description:Binding affinity was determined by measuring the inhibition of 125 I-NKA binding to transfected CHO cells expressing human recombinant Tachykinin rec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSubstance-K receptor(Human)
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM50403917(CHEMBL2112209)
Affinity DataIC50: 162nMAssay Description:Binding affinity was determined by measuring the inhibition of 125 I-NKA binding to transfected CHO cells expressing human recombinant Tachykinin rec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSubstance-K receptor(Human)
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM50115963(2-[(3,5-Bis-trifluoromethyl-benzoyl)-methyl-amino]...)
Affinity DataIC50: 168nMAssay Description:Binding affinity was determined by measuring the inhibition of 125 I-NKA binding to transfected CHO cells expressing human recombinant Tachykinin rec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSubstance-K receptor(Human)
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM50403919(CHEMBL2112211)
Affinity DataIC50: 181nMAssay Description:Binding affinity was determined by measuring the inhibition of 125 I-NKA binding to transfected CHO cells expressing human recombinant Tachykinin rec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSubstance-K receptor(Human)
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM50115964(2-[(3,5-Bis-trifluoromethyl-benzoyl)-methyl-amino]...)
Affinity DataIC50: 500nMAssay Description:Binding affinity was determined by measuring the inhibition of 125 I-NKA binding to transfected CHO cells expressing human recombinant Tachykinin rec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSubstance-K receptor(Human)
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM50115959(2-[(3,5-Bis-trifluoromethyl-benzoyl)-methyl-amino]...)
Affinity DataIC50: 560nMAssay Description:Binding affinity was determined by measuring the inhibition of 125 I-NKA binding to transfected CHO cells expressing human recombinant Tachykinin rec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSubstance-K receptor(Human)
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM50115966(4'-Chloro-2-(3,4,5-trimethoxy-benzoylamino)-biphen...)
Affinity DataIC50: 1.00E+3nMAssay Description:Binding affinity was determined by measuring the inhibition of 125 I-NKA binding to transfected CHO cells expressing human recombinant Tachykinin rec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSubstance-K receptor(Human)
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM50115969(N-[4-(N-Cyclohexyl-hydrazinocarbonyl)-4'-fluoro-bi...)
Affinity DataIC50: 1.00E+3nMAssay Description:Binding affinity was determined by measuring the inhibition of 125 I-NKA binding to transfected CHO cells expressing human recombinant Tachykinin rec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSubstance-K receptor(Human)
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM50115967(2-[(3,5-Bis-trifluoromethyl-benzoyl)-methyl-amino]...)
Affinity DataIC50: 1.00E+3nMAssay Description:Binding affinity was determined by measuring the inhibition of 125 I-NKA binding to transfected CHO cells expressing human recombinant Tachykinin rec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed