Compile Data Set for Download or QSAR
Report error Found 12 Enz. Inhib. hit(s) with all data for entry = 50003612
TargetSimilar to alpha-tubulin isoform 1(Bovine)
Australian National University

Curated by ChEMBL
LigandPNGBDBM50473762(CHEMBL90904)
Affinity DataIC50: 410nMAssay Description:Inhibition of tubulin (10 uM) polymerization, after a 20 min incubation at 30 degrees CentigradeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetSimilar to alpha-tubulin isoform 1(Bovine)
Australian National University

Curated by ChEMBL
LigandPNGBDBM50473763(CHEMBL409088)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of tubulin (10 uM) polymerization, after a 20 min incubation at 30 degrees CentigradeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetSimilar to alpha-tubulin isoform 1(Bovine)
Australian National University

Curated by ChEMBL
LigandPNGBDBM50473764(CHEMBL89341)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of tubulin (10 uM) polymerization, after a 20 min incubation at 30 degrees CentigradeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetSimilar to alpha-tubulin isoform 1(Bovine)
Australian National University

Curated by ChEMBL
LigandPNGBDBM50005480(combretastin A4 | CHEMBL67 | 2-Methoxy-5-[2-(3,4,5...)
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of tubulin (10 uM) polymerization, after a 20 min incubation at 30 degrees CentigradeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetSimilar to alpha-tubulin isoform 1(Bovine)
Australian National University

Curated by ChEMBL
LigandPNGBDBM50473768(CHEMBL314534)
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of tubulin (10 uM) polymerization, after a 20 min incubation at 30 degrees CentigradeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetSimilar to alpha-tubulin isoform 1(Bovine)
Australian National University

Curated by ChEMBL
LigandPNGBDBM50103821([2-(3-Hydroxy-4-methoxy-phenyl)-6-methoxy-benzo[b]...)
Affinity DataIC50: 3.40E+3nMAssay Description:Inhibition of tubulin (10 uM) polymerization, after a 20 min incubation at 30 degrees CentigradeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetSimilar to alpha-tubulin isoform 1(Bovine)
Australian National University

Curated by ChEMBL
LigandPNGBDBM50473769(CHEMBL327414)
Affinity DataIC50: 4.10E+3nMAssay Description:Inhibition of tubulin (10 uM) polymerization, after a 20 min incubation at 30 degrees CentigradeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetSimilar to alpha-tubulin isoform 1(Bovine)
Australian National University

Curated by ChEMBL
LigandPNGBDBM50473766(CHEMBL90441)
Affinity DataIC50: 8.80E+3nMAssay Description:Inhibition of tubulin (10 uM) polymerization, after a 20 min incubation at 30 degrees CentigradeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetSimilar to alpha-tubulin isoform 1(Bovine)
Australian National University

Curated by ChEMBL
LigandPNGBDBM50473761(CHEMBL89039)
Affinity DataIC50: 4.00E+4nMAssay Description:Inhibition of tubulin (10 uM) polymerization, after a 20 min incubation at 30 degrees CentigradeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetSimilar to alpha-tubulin isoform 1(Bovine)
Australian National University

Curated by ChEMBL
LigandPNGBDBM50103823([6-Methoxy-2-(4-methoxy-phenyl)-benzo[b]thiophen-3...)
Affinity DataIC50: 4.00E+4nMAssay Description:Inhibition of tubulin (10 uM) polymerization, after a 20 min incubation at 30 degrees CentigradeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetSimilar to alpha-tubulin isoform 1(Bovine)
Australian National University

Curated by ChEMBL
LigandPNGBDBM50473765(CHEMBL90926)
Affinity DataIC50: 4.00E+4nMAssay Description:Inhibition of tubulin (10 uM) polymerization, after a 20 min incubation at 30 degrees CentigradeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetSimilar to alpha-tubulin isoform 1(Bovine)
Australian National University

Curated by ChEMBL
LigandPNGBDBM50473767(CHEMBL327181)
Affinity DataIC50: 4.00E+4nMAssay Description:Inhibition of tubulin (10 uM) polymerization, after a 20 min incubation at 30 degrees CentigradeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed