Compile Data Set for Download or QSAR
Report error Found 12 Enz. Inhib. hit(s) with all data for entry = 50012038
TargetDipeptidyl peptidase 4(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM11694(Cyclohexylglycine-(2S)-cyanopyrolidine 3 | (2S)-1-...)
Affinity DataIC50: 2nMAssay Description:In vitro inhibitory activity against Dipeptidyl peptidase IV (DPP-IV) extracted from Caco-2 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM11694(Cyclohexylglycine-(2S)-cyanopyrolidine 3 | (2S)-1-...)
Affinity DataIC50: 2.80nMAssay Description:In vitro inhibitory activity against Dipeptidyl peptidase IV (DPP-IV) extracted from rat plasmaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM11694(Cyclohexylglycine-(2S)-cyanopyrolidine 3 | (2S)-1-...)
Affinity DataIC50: 3.20nMAssay Description:In vitro inhibitory activity against Dipeptidyl peptidase IV (DPP-IV) extracted from human plasmaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM11113(NVP-DPP728 | cyanopyrrolidine derivative 2 | CHEMB...)
Affinity DataIC50: 6nMAssay Description:In vitro inhibitory activity against Dipeptidyl peptidase IV (DPP-IV) extracted from rat plasma.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM11113(NVP-DPP728 | cyanopyrrolidine derivative 2 | CHEMB...)
Affinity DataIC50: 7nMAssay Description:In vitro inhibitory activity against Dipeptidyl peptidase IV (DPP-IV) extracted from human plasma.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50113678(1-{2-[2-(5-Nitro-pyridin-2-ylamino)-ethylamino]-ac...)
Affinity DataIC50: 8nMAssay Description:In vitro inhibitory activity against Dipeptidyl peptidase IV (DPP-IV) extracted from Caco-2 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50113678(1-{2-[2-(5-Nitro-pyridin-2-ylamino)-ethylamino]-ac...)
Affinity DataIC50: 8.70nMAssay Description:In vitro inhibitory activity against Dipeptidyl peptidase IV (DPP-IV) extracted from human plasmaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50113678(1-{2-[2-(5-Nitro-pyridin-2-ylamino)-ethylamino]-ac...)
Affinity DataIC50: 17nMAssay Description:In vitro inhibitory activity against Dipeptidyl peptidase IV (DPP-IV) extracted from rat plasmaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM11113(NVP-DPP728 | cyanopyrrolidine derivative 2 | CHEMB...)
Affinity DataIC50: 22nMAssay Description:In vitro inhibitory activity against Dipeptidyl peptidase IV (DPP-IV) extracted from Caco-2 cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50113678(1-{2-[2-(5-Nitro-pyridin-2-ylamino)-ethylamino]-ac...)
Affinity DataIC50: 1.20E+4nMAssay Description:In vitro inhibitory activity against Dipeptidylpeptidase II (DPP-II) extracted from bovine kidney homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM11694(Cyclohexylglycine-(2S)-cyanopyrolidine 3 | (2S)-1-...)
Affinity DataIC50: 1.02E+5nMAssay Description:In vitro inhibitory activity against Dipeptidylpeptidase II (DPP-II) extracted from bovine kidney homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM11113(NVP-DPP728 | cyanopyrrolidine derivative 2 | CHEMB...)
Affinity DataIC50: 1.10E+5nMAssay Description:In vitro inhibitory activity against Dipeptidylpeptidase II (DPP-II) extracted from bovine kidney homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed