Compile Data Set for Download or QSAR
Report error Found 26 Enz. Inhib. hit(s) with all data for entry = 50035224
TargetTyrosine-protein kinase Lck(Human)
Roche Products

Curated by ChEMBL
LigandPNGBDBM50112960((1S,3R)-3-({(1S,9S)-9-[(S)-2-Acetylamino-3-(4-phos...)
Affinity DataIC50: 30nMAssay Description:Inhibitory activity towards p56 Lck tyrosine kinase SH2 domain using scintillation proximity assay (SPA)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetTyrosine-protein kinase Lck(Human)
Roche Products

Curated by ChEMBL
LigandPNGBDBM50112980((1R,3R)-3-({(1S,9S)-9-[(S)-2-Acetylamino-3-(4-phos...)
Affinity DataIC50: 100nMAssay Description:Inhibitory activity towards p56 Lck tyrosine kinase SH2 domain using scintillation proximity assay (SPA)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetTyrosine-protein kinase Lck(Human)
Roche Products

Curated by ChEMBL
LigandPNGBDBM50112966(EPQpYEEIPIYL | CHEMBL2372049)
Affinity DataIC50: 360nMAssay Description:Inhibitory activity towards p56 Lck tyrosine kinase SH2 domain using scintillation proximity assay (SPA)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetTyrosine-protein kinase Lck(Human)
Roche Products

Curated by ChEMBL
LigandPNGBDBM50112959(Phosphoric acid mono-(4-{(S)-2-acetylamino-2-[(4S,...)
Affinity DataIC50: 400nMAssay Description:Inhibitory activity towards p56 Lck tyrosine kinase SH2 domain using scintillation proximity assay (SPA)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetTyrosine-protein kinase Lck(Human)
Roche Products

Curated by ChEMBL
LigandPNGBDBM50112974(Phosphoric acid mono-(4-{(S)-2-acetylamino-2-[(4S,...)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibitory activity towards p56 Lck tyrosine kinase SH2 domain using scintillation proximity assay (SPA)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetTyrosine-protein kinase Lck(Human)
Roche Products

Curated by ChEMBL
LigandPNGBDBM50112973(Phosphoric acid mono-[4-((S)-2-acetylamino-2-{(4S,...)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibitory activity towards p56 Lck tyrosine kinase SH2 domain using scintillation proximity assay (SPA)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetTyrosine-protein kinase Lck(Human)
Roche Products

Curated by ChEMBL
LigandPNGBDBM50112975(Phosphoric acid mono-(4-{(S)-2-acetylamino-2-[(4S,...)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibitory activity towards p56 Lck tyrosine kinase SH2 domain using scintillation proximity assay (SPA)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetTyrosine-protein kinase Lck(Human)
Roche Products

Curated by ChEMBL
LigandPNGBDBM50112971(Phosphoric acid mono-(4-{(S)-2-acetylamino-2-[(4S,...)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibitory activity towards p56 Lck tyrosine kinase SH2 domain using scintillation proximity assay (SPA)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetTyrosine-protein kinase Lck(Human)
Roche Products

Curated by ChEMBL
LigandPNGBDBM50112968(Phosphoric acid mono-{4-[(S)-2-acetylamino-2-((4S,...)
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibitory activity towards p56 Lck tyrosine kinase SH2 domain using scintillation proximity assay (SPA)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetTyrosine-protein kinase Lck(Human)
Roche Products

Curated by ChEMBL
LigandPNGBDBM50112964(Phosphoric acid mono-(4-{(S)-2-acetylamino-2-[(4S,...)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibitory activity towards p56 Lck tyrosine kinase SH2 domain using scintillation proximity assay (SPA)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetTyrosine-protein kinase Lck(Human)
Roche Products

Curated by ChEMBL
LigandPNGBDBM50112958(Phosphoric acid mono-(4-{(S)-2-acetylamino-2-[(4S,...)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibitory activity towards p56 Lck tyrosine kinase SH2 domain using scintillation proximity assay (SPA)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetTyrosine-protein kinase Lck(Human)
Roche Products

Curated by ChEMBL
LigandPNGBDBM50112972((S)-4-{(S)-2-[(S)-2-Acetylamino-3-(4-phosphonooxy-...)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibitory activity towards p56 Lck tyrosine kinase SH2 domain using scintillation proximity assay (SPA)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetTyrosine-protein kinase Lck(Human)
Roche Products

Curated by ChEMBL
LigandPNGBDBM50112969(Phosphoric acid mono-{4-[(S)-2-acetylamino-2-((4S,...)
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibitory activity towards p56 Lck tyrosine kinase SH2 domain using scintillation proximity assay (SPA)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetTyrosine-protein kinase Lck(Human)
Roche Products

Curated by ChEMBL
LigandPNGBDBM50112970(Phosphoric acid mono-(4-{(S)-2-acetylamino-2-[(4S,...)
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibitory activity towards p56 Lck tyrosine kinase SH2 domain using scintillation proximity assay (SPA)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetTyrosine-protein kinase Lck(Human)
Roche Products

Curated by ChEMBL
LigandPNGBDBM50112981(Phosphoric acid mono-{4-[(S)-2-acetylamino-2-((4S,...)
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibitory activity towards p56 Lck tyrosine kinase SH2 domain using scintillation proximity assay (SPA)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetTyrosine-protein kinase Lck(Human)
Roche Products

Curated by ChEMBL
LigandPNGBDBM50112961(Phosphoric acid mono-[4-((S)-2-acetylamino-2-{(4S,...)
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibitory activity towards p56 Lck tyrosine kinase SH2 domain using scintillation proximity assay (SPA)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetTyrosine-protein kinase Lck(Human)
Roche Products

Curated by ChEMBL
LigandPNGBDBM50112979((1S,3S)-3-({(1S,9S)-9-[(S)-2-Acetylamino-3-(4-phos...)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibitory activity towards p56 Lck tyrosine kinase SH2 domain using scintillation proximity assay (SPA)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetTyrosine-protein kinase Lck(Human)
Roche Products

Curated by ChEMBL
LigandPNGBDBM50366781(CHEMBL1790100)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibitory activity towards p56 Lck tyrosine kinase SH2 domain using scintillation proximity assay (SPA)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetTyrosine-protein kinase Lck(Human)
Roche Products

Curated by ChEMBL
LigandPNGBDBM50112962((1R,3S)-3-({(1S,9S)-9-[(S)-2-Acetylamino-3-(4-phos...)
Affinity DataIC50: 2.80E+3nMAssay Description:Inhibitory activity towards p56 Lck tyrosine kinase SH2 domain using scintillation proximity assay (SPA)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetTyrosine-protein kinase Lck(Human)
Roche Products

Curated by ChEMBL
LigandPNGBDBM50112976(Phosphoric acid mono-{4-[(S)-2-acetylamino-2-((4S,...)
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibitory activity towards p56 Lck tyrosine kinase SH2 domain using scintillation proximity assay (SPA)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetTyrosine-protein kinase Lck(Human)
Roche Products

Curated by ChEMBL
LigandPNGBDBM50112977(3-({(1S,9S)-9-[(S)-2-Acetylamino-3-(4-phosphonooxy...)
Affinity DataIC50: 7.30E+3nMAssay Description:Inhibitory activity towards p56 Lck tyrosine kinase SH2 domain using scintillation proximity assay (SPA)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetTyrosine-protein kinase Lck(Human)
Roche Products

Curated by ChEMBL
LigandPNGBDBM50112977(3-({(1S,9S)-9-[(S)-2-Acetylamino-3-(4-phosphonooxy...)
Affinity DataIC50: 7.70E+3nMAssay Description:Inhibitory activity towards p56 Lck tyrosine kinase SH2 domain using scintillation proximity assay (SPA)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetTyrosine-protein kinase Lck(Human)
Roche Products

Curated by ChEMBL
LigandPNGBDBM50112965(Phosphoric acid mono-{4-[(S)-2-acetylamino-2-((4S,...)
Affinity DataIC50: 8.50E+3nMAssay Description:Inhibitory activity towards p56 Lck tyrosine kinase SH2 domain using scintillation proximity assay (SPA)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetTyrosine-protein kinase Lck(Human)
Roche Products

Curated by ChEMBL
LigandPNGBDBM50112963(Phosphoric acid mono-(4-{(S)-2-acetylamino-2-[(4S,...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibitory activity towards p56 Lck tyrosine kinase SH2 domain using scintillation proximity assay (SPA)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetTyrosine-protein kinase Lck(Human)
Roche Products

Curated by ChEMBL
LigandPNGBDBM50112957((S)-4-[(S)-2-Acetylamino-3-(4-phosphonooxy-phenyl)...)
Affinity DataIC50: 1.70E+4nMAssay Description:Inhibitory activity towards p56 Lck tyrosine kinase SH2 domain using scintillation proximity assay (SPA)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetTyrosine-protein kinase Lck(Human)
Roche Products

Curated by ChEMBL
LigandPNGBDBM50112967((S)-4-[(S)-2-Acetylamino-3-(4-phosphonooxy-phenyl)...)
Affinity DataIC50: 3.50E+5nMAssay Description:Inhibitory activity towards p56 Lck tyrosine kinase SH2 domain using scintillation proximity assay (SPA)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed