Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 4030
TargetLeucine--tRNA ligase(Thermus thermophilus)
Wayne State University

LigandPNGBDBM19(KDR Kinase Inhibitor, 3 | Neomycin | (2S,3S,4R,5R,...)
Affinity DataKd:  5nMpH: 7.5 T: 2°CAssay Description:Binding assay of Aminoglycoside antibiotics and kanamycin A derivatives for the bacterial A site RNA.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2011
Entry Details Article
PubMed
TargetLeucine--tRNA ligase(Thermus thermophilus)
Wayne State University

LigandPNGBDBM43823(N-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-piperidinos...)
Affinity DataKd:  1.10E+3nMpH: 7.5 T: 2°CAssay Description:Binding assay of Aminoglycoside antibiotics and kanamycin A derivatives for the bacterial A site RNA.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2011
Entry Details Article
PubMed
TargetLeucine--tRNA ligase(Thermus thermophilus)
Wayne State University

LigandPNGBDBM43824(N-[(E)-N''''-(1,3-benzothiazol-2-yl)carbamimidoyl]...)
Affinity DataKd:  1.30E+6nMpH: 7.5 T: 2°CAssay Description:Binding assay of Aminoglycoside antibiotics and kanamycin A derivatives for the bacterial A site RNA.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2011
Entry Details Article
PubMed
TargetLeucine--tRNA ligase(Thermus thermophilus)
Wayne State University

LigandPNGBDBM43825(methyl (Z)-3-(3-chloro-2-methylanilino)-2-[3-chlor...)
Affinity DataKd:  2.00E+6nMpH: 7.5 T: 2°CAssay Description:Binding assay of Aminoglycoside antibiotics and kanamycin A derivatives for the bacterial A site RNA.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2011
Entry Details Article
PubMed
TargetLeucine--tRNA ligase(Thermus thermophilus)
Wayne State University

LigandPNGBDBM43827(MLS000567315 | cid_2565969 | (E)-3-(1-benzyl-3-phe...)
Affinity DataKd:  1.70E+6nMpH: 7.5 T: 2°CAssay Description:Binding assay of Aminoglycoside antibiotics and kanamycin A derivatives for the bacterial A site RNA.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2011
Entry Details Article
PubMed
TargetLeucine--tRNA ligase(Thermus thermophilus)
Wayne State University

LigandPNGBDBM43826(MLS000568202 | 2-[[5-(diethylsulfamoyl)-1-(4-metho...)
Affinity DataKd:  6.00E+5nMpH: 7.5 T: 2°CAssay Description:Binding assay of Aminoglycoside antibiotics and kanamycin A derivatives for the bacterial A site RNA.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2011
Entry Details Article
PubMed