Compile Data Set for Download or QSAR
Report error Found 19 Enz. Inhib. hit(s) with all data for entry = 50011953
TargetGlucagon receptor(Human)
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50109326((R)-1-[4-(4-Fluoro-phenyl)-2,6-diisopropyl-5-propy...)
Affinity DataIC50: 65nMAssay Description:Tested for its ability to inhibit cAMP production in human glucagon receptor expressed CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50109326((R)-1-[4-(4-Fluoro-phenyl)-2,6-diisopropyl-5-propy...)
Affinity DataIC50: 110nMAssay Description:Tested for its inhibitory activity against human glucagon receptor (hGR) expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50112476(5-Fluoro-2-(3-hydroxymethyl-2,6-diisopropyl-5-pent...)
Affinity DataIC50: 120nMAssay Description:Tested for its ability to inhibit cAMP production in human glucagon receptor expressed CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50112476(5-Fluoro-2-(3-hydroxymethyl-2,6-diisopropyl-5-pent...)
Affinity DataIC50: 190nMAssay Description:Tested for its inhibitory activity against human glucagon receptor (hGR) expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50109331([4-(4-Fluoro-phenyl)-2,6-diisopropyl-5-pentyl-pyri...)
Affinity DataIC50: 400nMAssay Description:Tested for its ability to inhibit cAMP production in human glucagon receptor expressed CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50112484(2-(3-Hydroxymethyl-2,6-diisopropyl-5-pentyl-pyridi...)
Affinity DataIC50: 500nMAssay Description:Tested for its inhibitory activity against human glucagon receptor (hGR) expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50109331([4-(4-Fluoro-phenyl)-2,6-diisopropyl-5-pentyl-pyri...)
Affinity DataIC50: 700nMAssay Description:Tested for its inhibitory activity against human glucagon receptor (hGR) expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50112475([4-(4-Chloro-phenyl)-2,6-diisopropyl-5-pentyl-pyri...)
Affinity DataIC50: 800nMAssay Description:Tested for its inhibitory activity against human glucagon receptor (hGR) expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50112479((2,6-Diisopropyl-5-pentyl-4-p-tolyl-pyridin-3-yl)-...)
Affinity DataIC50: 1.00E+3nMAssay Description:Tested for its inhibitory activity against human glucagon receptor (hGR) expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50112478([4-(3,4-Difluoro-phenyl)-2,6-diisopropyl-5-pentyl-...)
Affinity DataIC50: 1.10E+3nMAssay Description:Tested for its inhibitory activity against human glucagon receptor (hGR) expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50109336((2,6-Diisopropyl-5-pentyl-4-phenyl-pyridin-3-yl)-m...)
Affinity DataIC50: 1.40E+3nMAssay Description:Tested for its inhibitory activity against human glucagon receptor (hGR) expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50112485([4-(2-Amino-phenyl)-2,6-diisopropyl-5-pentyl-pyrid...)
Affinity DataIC50: 2.30E+3nMAssay Description:Tested for its inhibitory activity against human glucagon receptor (hGR) expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50112483([4-(3-Fluoro-phenyl)-2,6-diisopropyl-5-pentyl-pyri...)
Affinity DataIC50: 3.00E+3nMAssay Description:Tested for its inhibitory activity against human glucagon receptor (hGR) expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50112481(3-(3-Hydroxymethyl-2,6-diisopropyl-5-pentyl-pyridi...)
Affinity DataIC50: 6.00E+3nMAssay Description:Tested for its inhibitory activity against human glucagon receptor (hGR) expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50112477(4-(4-Fluoro-phenyl)-2,6-diisopropyl-5-(2-methyl-pr...)
Affinity DataIC50: 7.00E+3nMAssay Description:Tested for its inhibitory activity against human glucagon receptor (hGR) expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50112480([4-(2-Fluoro-phenyl)-2,6-diisopropyl-5-pentyl-pyri...)
Affinity DataIC50: 9.00E+3nMAssay Description:Tested for its inhibitory activity against human glucagon receptor (hGR) expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50112482([4-(2,4-Difluoro-phenyl)-2,6-diisopropyl-5-pentyl-...)
Affinity DataIC50: 1.10E+4nMAssay Description:Tested for its inhibitory activity against human glucagon receptor (hGR) expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50112473([4-(4-Fluoro-3-hydroxymethyl-phenyl)-2,6-diisoprop...)
Affinity DataIC50: 1.90E+4nMAssay Description:Tested for its inhibitory activity against human glucagon receptor (hGR) expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50112474([2,6-Diisopropyl-4-(3-methoxy-phenyl)-5-pentyl-pyr...)
Affinity DataIC50: 4.80E+4nMAssay Description:Tested for its inhibitory activity against human glucagon receptor (hGR) expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed