Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 50011701
TargetProtein kinase C delta type(Mouse)
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50057514(13-Hydroxymethyl-10-isopropyl-9-methyl-5-octyl-3,9...)
Affinity DataKi:  0.100nMAssay Description:Displacement of [3H]- PDBu from Protein kinase C delta C1b domainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRAS guanyl-releasing protein 1(Rat)
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50057514(13-Hydroxymethyl-10-isopropyl-9-methyl-5-octyl-3,9...)
Affinity DataKi:  0.850nMAssay Description:Binding affinity against RAS guanyl releasing protein using [3H]- PDBu as the labeled ligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein kinase C delta type(Mouse)
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50057511(CHEMBL27266 | 13-Hydroxymethyl-10-isopropyl-9-meth...)
Affinity DataKi:  2.01nMAssay Description:Displacement of [3H]- PDBu from Protein kinase C delta C1b domainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRAS guanyl-releasing protein 1(Rat)
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50057511(CHEMBL27266 | 13-Hydroxymethyl-10-isopropyl-9-meth...)
Affinity DataKi:  2.54nMAssay Description:Binding affinity against RAS guanyl releasing protein using [3H]- PDBu as the labeled ligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRAS guanyl-releasing protein 1(Rat)
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50057509(8-Dec-1-ynyl-5-hydroxymethyl-2-isopropyl-1-methyl-...)
Affinity DataKi:  6.15nMAssay Description:Binding affinity against RAS guanyl releasing protein using [3H]- PDBu as the labeled ligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein kinase C delta type(Mouse)
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50057509(8-Dec-1-ynyl-5-hydroxymethyl-2-isopropyl-1-methyl-...)
Affinity DataKi:  10.7nMAssay Description:Displacement of [3H]- PDBu from Protein kinase C delta C1b domainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRAS guanyl-releasing protein 1(Rat)
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50096601(8-Dec-1-ynyl-5-hydroxymethyl-2-isopropyl-7-methoxy...)
Affinity DataKi:  13.9nMAssay Description:Binding affinity against RAS guanyl releasing protein using [3H]- PDBu as the labeled ligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein kinase C delta type(Mouse)
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50096601(8-Dec-1-ynyl-5-hydroxymethyl-2-isopropyl-7-methoxy...)
Affinity DataKi:  35.1nMAssay Description:Displacement of [3H]- PDBu from Protein kinase C delta C1b domainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed