Compile Data Set for Download or QSAR
Report error Found 30 Enz. Inhib. hit(s) with all data for entry = 50011684
TargetIntegrin alpha-V/beta-3(Human)
Knoll

Curated by ChEMBL
LigandPNGBDBM50109298([5-({[4-(1H-Benzoimidazol-2-ylamino)-cyclohexylmet...)
Affinity DataIC50: 1.60nMAssay Description:Affinity against alpha V-beta3 integrin via competitive ELISA using vitronectin as natural ligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-3(Human)
Knoll

Curated by ChEMBL
LigandPNGBDBM50109296((5-{[4-(1H-Benzoimidazol-2-ylamino)-benzylcarbamoy...)
Affinity DataIC50: 7nMAssay Description:Affinity against alpha V-beta3 integrin via competitive ELISA using vitronectin as natural ligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-3(Human)
Knoll

Curated by ChEMBL
LigandPNGBDBM50109296((5-{[4-(1H-Benzoimidazol-2-ylamino)-benzylcarbamoy...)
Affinity DataIC50: 7.30nMAssay Description:Affinity against alpha V-beta3 integrin via competitive ELISA using vitronectin as natural ligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-3(Human)
Knoll

Curated by ChEMBL
LigandPNGBDBM50109305((5-{[5-(1H-Benzoimidazol-2-ylamino)-pentylcarbamoy...)
Affinity DataIC50: 13nMAssay Description:Affinity against alpha V-beta3 integrin via competitive ELISA using vitronectin as natural ligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-3(Human)
Knoll

Curated by ChEMBL
LigandPNGBDBM50109307((5-{[4-(1H-Benzoimidazol-2-ylamino)-butylcarbamoyl...)
Affinity DataIC50: 15nMAssay Description:Affinity against alpha V-beta3 integrin via competitive ELISA using vitronectin as natural ligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-3(Human)
Knoll

Curated by ChEMBL
LigandPNGBDBM50109303((5-{[4-(3-Benzyl-ureido)-benzylcarbamoyl]-methyl}-...)
Affinity DataIC50: 23nMAssay Description:Affinity against alpha V-beta3 integrin via competitive ELISA using vitronectin as natural ligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-3(Human)
Knoll

Curated by ChEMBL
LigandPNGBDBM50109298([5-({[4-(1H-Benzoimidazol-2-ylamino)-cyclohexylmet...)
Affinity DataIC50: 40nMAssay Description:Adhesion of recombinant alphaV-beta3 integrin expressed in CHO-K1 to osteopontin (OPN)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-3(Human)
Knoll

Curated by ChEMBL
LigandPNGBDBM50109293((5-{[4-(1H-Benzoimidazol-2-yl)-benzylcarbamoyl]-me...)
Affinity DataIC50: 74nMAssay Description:Affinity against alpha V-beta3 integrin via competitive ELISA using vitronectin as natural ligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-3(Human)
Knoll

Curated by ChEMBL
LigandPNGBDBM50109301({5-[(4-Guanidino-benzylcarbamoyl)-methyl]-6-oxo-6,...)
Affinity DataIC50: 84nMAssay Description:Affinity against alpha V-beta3 integrin via competitive ELISA using vitronectin as natural ligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-3(Human)
Knoll

Curated by ChEMBL
LigandPNGBDBM50109300([5-({[4-(1H-Benzoimidazol-2-yl)-thiophen-2-ylmethy...)
Affinity DataIC50: 100nMAssay Description:Affinity against alpha V-beta3 integrin via competitive ELISA using vitronectin as natural ligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-3(Human)
Knoll

Curated by ChEMBL
LigandPNGBDBM50109296((5-{[4-(1H-Benzoimidazol-2-ylamino)-benzylcarbamoy...)
Affinity DataIC50: 100nMAssay Description:Cell adhesion of alphaV-beta3 integrin expressed in CHO-K1 cell to osteopontin (OPN)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-3(Human)
Knoll

Curated by ChEMBL
LigandPNGBDBM50109299([5-({[6-(1H-Benzoimidazol-2-yl)-pyridin-3-ylmethyl...)
Affinity DataIC50: 200nMAssay Description:Affinity against alpha V-beta3 integrin via competitive ELISA using vitronectin as natural ligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-3(Human)
Knoll

Curated by ChEMBL
LigandPNGBDBM50109312((5-{[4-(5,6-Dimethyl-1H-benzoimidazol-2-yl)-benzyl...)
Affinity DataIC50: 220nMAssay Description:Affinity against alpha V-beta3 integrin via competitive ELISA using vitronectin as natural ligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-3(Human)
Knoll

Curated by ChEMBL
LigandPNGBDBM50109289([6-Oxo-5-({[4-(pyridin-2-ylaminomethyl)-thiophen-2...)
Affinity DataIC50: 220nMAssay Description:Affinity against alpha V-beta3 integrin via competitive ELISA using vitronectin as natural ligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-3(Human)
Knoll

Curated by ChEMBL
LigandPNGBDBM50109310([5-({2-[4-(1H-Benzoimidazol-2-yl)-phenyl]-ethylcar...)
Affinity DataIC50: 380nMAssay Description:Affinity against alpha V-beta3 integrin via competitive ELISA using vitronectin as natural ligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-3(Human)
Knoll

Curated by ChEMBL
LigandPNGBDBM50109304([5-({[4-(3H-Imidazo[4,5-b]pyridin-2-yl)-thiophen-2...)
Affinity DataIC50: 500nMAssay Description:Affinity against alpha V-beta3 integrin via competitive ELISA using vitronectin as natural ligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-3(Human)
Knoll

Curated by ChEMBL
LigandPNGBDBM50109290([5-({[5-(1H-Benzoimidazol-2-yl)-thiophen-2-ylmethy...)
Affinity DataIC50: 500nMAssay Description:Affinity against alpha V-beta3 integrin via competitive ELISA using vitronectin as natural ligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-3(Human)
Knoll

Curated by ChEMBL
LigandPNGBDBM50109302((5-{[4-(5-Chloro-1H-benzoimidazol-2-yl)-benzylcarb...)
Affinity DataIC50: 620nMAssay Description:Affinity against alpha V-beta3 integrin via competitive ELISA using vitronectin as natural ligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-3(Human)
Knoll

Curated by ChEMBL
LigandPNGBDBM50109291((5-{[(4-Carbamimidoyl-thiophen-2-ylmethyl)-carbamo...)
Affinity DataIC50: 1.00E+3nMAssay Description:Affinity against alpha V-beta3 integrin via competitive ELISA using vitronectin as natural ligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-3(Human)
Knoll

Curated by ChEMBL
LigandPNGBDBM50109297((5-{[(1H-Benzoimidazol-2-ylmethyl)-carbamoyl]-meth...)
Affinity DataIC50: 1.00E+3nMAssay Description:Affinity against alpha V-beta3 integrin via competitive ELISA using vitronectin as natural ligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-3(Human)
Knoll

Curated by ChEMBL
LigandPNGBDBM50109306([5-({[4-(1H-Benzoimidazol-2-yl)-thiazol-2-ylmethyl...)
Affinity DataIC50: 1.00E+3nMAssay Description:Affinity against alpha V-beta3 integrin via competitive ELISA using vitronectin as natural ligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-3(Human)
Knoll

Curated by ChEMBL
LigandPNGBDBM50109309((6-Oxo-5-{[3-(pyridin-2-ylamino)-propylcarbamoyl]-...)
Affinity DataIC50: 1.00E+3nMAssay Description:Affinity against alpha V-beta3 integrin via competitive ELISA using vitronectin as natural ligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-3(Human)
Knoll

Curated by ChEMBL
LigandPNGBDBM50109295((6-Oxo-5-{[4-(pyridin-2-ylamino)-benzylcarbamoyl]-...)
Affinity DataIC50: 5.00E+3nMAssay Description:Affinity against alpha V-beta3 integrin via competitive ELISA using vitronectin as natural ligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-3(Human)
Knoll

Curated by ChEMBL
LigandPNGBDBM50109311((5-{[4-(1H-Benzoimidazol-2-yl)-phenylcarbamoyl]-me...)
Affinity DataIC50: 5.00E+3nMAssay Description:Affinity against alpha V-beta3 integrin via competitive ELISA using vitronectin as natural ligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-3(Human)
Knoll

Curated by ChEMBL
LigandPNGBDBM50109294((5-{[3-(1H-Benzoimidazol-2-yl)-benzylcarbamoyl]-me...)
Affinity DataIC50: 1.00E+4nMAssay Description:Affinity against alpha V-beta3 integrin via competitive ELISA using vitronectin as natural ligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-3(Human)
Knoll

Curated by ChEMBL
LigandPNGBDBM50109308({5-[(4-Benzyloxycarbonylamino-benzylcarbamoyl)-met...)
Affinity DataIC50: 1.00E+4nMAssay Description:Affinity against alpha V-beta3 integrin via competitive ELISA using vitronectin as natural ligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-3(Human)
Knoll

Curated by ChEMBL
LigandPNGBDBM50109292({5-[(4-Benzylcarbamoyloxy-benzylcarbamoyl)-methyl]...)
Affinity DataIC50: 1.00E+4nMAssay Description:Affinity against alpha V-beta3 integrin via competitive ELISA using vitronectin as natural ligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-3(Human)
Knoll

Curated by ChEMBL
LigandPNGBDBM50109288((5-{4-[4-(3-Benzyl-ureido)-phenyl]-butyl}-6-oxo-6,...)
Affinity DataIC50: 1.00E+4nMAssay Description:Affinity against alpha V-beta3 integrin via competitive ELISA using vitronectin as natural ligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrin alpha-IIb/beta-3(Human)
Knoll

Curated by ChEMBL
LigandPNGBDBM50109298([5-({[4-(1H-Benzoimidazol-2-ylamino)-cyclohexylmet...)
Affinity DataIC50: 1.00E+6nMAssay Description:Displacement of alphaIIb-beta3 integrin from fibrinogen by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrin alpha-IIb/beta-3(Human)
Knoll

Curated by ChEMBL
LigandPNGBDBM50109296((5-{[4-(1H-Benzoimidazol-2-ylamino)-benzylcarbamoy...)
Affinity DataIC50: 1.00E+6nMAssay Description:Displacement of alphaIIb-beta3 integrin from fibrinogen by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed