Compile Data Set for Download or QSAR
Report error Found 14 Enz. Inhib. hit(s) with all data for entry = 50011671
TargetInterstitial collagenase(Human)
Organon K.K.

Curated by ChEMBL
LigandPNGBDBM50031795((N-(2-HYDROXAMATEMETHYLENE-4-METHYL-PENTOYL)PHENYL...)
Affinity DataIC50: 3nMAssay Description:Inhibition of Matrix metalloprotease-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProcathepsin L(Human)
Organon K.K.

Curated by ChEMBL
LigandPNGBDBM50109171([(S)-1-((S)-1-Methyl-2-oxo-ethylcarbamoyl)-2-pheny...)
Affinity DataIC50: 3nMAssay Description:Inhibition of Cathepsin L from human kidneyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProcathepsin L(Human)
Organon K.K.

Curated by ChEMBL
LigandPNGBDBM50109168((R)-N*1*-[(S)-1-((S)-1-Formyl-3-methyl-butylcarbam...)
Affinity DataIC50: 7nMAssay Description:Inhibition of Cathepsin L from human kidneyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetInterstitial collagenase(Human)
Organon K.K.

Curated by ChEMBL
LigandPNGBDBM50109167((R)-N*4*-Hydroxy-2-isobutyl-N*1*-[(S)-1-(2-oxo-eth...)
Affinity DataIC50: 12nMAssay Description:Inhibition of Matrix metalloprotease-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProcathepsin L(Human)
Organon K.K.

Curated by ChEMBL
LigandPNGBDBM50109169((R)-N*4*-Hydroxy-2-isobutyl-N*1*-[(S)-1-((S)-1-met...)
Affinity DataIC50: 15nMAssay Description:Inhibition of Cathepsin L from human kidneyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProcathepsin L(Human)
Organon K.K.

Curated by ChEMBL
LigandPNGBDBM50109170(N*4*-Hydroxy-2-isobutyl-N*1*-[3-methyl-1-(1-methyl...)
Affinity DataIC50: 23nMAssay Description:Inhibition of Cathepsin L from human kidneyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetInterstitial collagenase(Human)
Organon K.K.

Curated by ChEMBL
LigandPNGBDBM50109169((R)-N*4*-Hydroxy-2-isobutyl-N*1*-[(S)-1-((S)-1-met...)
Affinity DataIC50: 25nMAssay Description:Inhibition of Matrix metalloprotease-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetInterstitial collagenase(Human)
Organon K.K.

Curated by ChEMBL
LigandPNGBDBM50109172((R)-N*1*-[(S)-1-((S)-2,2-Diethoxy-1-methyl-ethylca...)
Affinity DataIC50: 29nMAssay Description:Inhibition of Matrix metalloprotease-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetInterstitial collagenase(Human)
Organon K.K.

Curated by ChEMBL
LigandPNGBDBM50109170(N*4*-Hydroxy-2-isobutyl-N*1*-[3-methyl-1-(1-methyl...)
Affinity DataIC50: 47nMAssay Description:Inhibition of Matrix metalloprotease-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProcathepsin L(Human)
Organon K.K.

Curated by ChEMBL
LigandPNGBDBM50031795((N-(2-HYDROXAMATEMETHYLENE-4-METHYL-PENTOYL)PHENYL...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of Cathepsin L from human kidneyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetInterstitial collagenase(Human)
Organon K.K.

Curated by ChEMBL
LigandPNGBDBM50109171([(S)-1-((S)-1-Methyl-2-oxo-ethylcarbamoyl)-2-pheny...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of Matrix metalloprotease-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProcathepsin L(Human)
Organon K.K.

Curated by ChEMBL
LigandPNGBDBM50109172((R)-N*1*-[(S)-1-((S)-2,2-Diethoxy-1-methyl-ethylca...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of Cathepsin L from human kidneyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetInterstitial collagenase(Human)
Organon K.K.

Curated by ChEMBL
LigandPNGBDBM50109168((R)-N*1*-[(S)-1-((S)-1-Formyl-3-methyl-butylcarbam...)
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of Matrix metalloprotease-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProcathepsin L(Human)
Organon K.K.

Curated by ChEMBL
LigandPNGBDBM50109167((R)-N*4*-Hydroxy-2-isobutyl-N*1*-[(S)-1-(2-oxo-eth...)
Affinity DataIC50: 4.30E+3nMAssay Description:Inhibition of Cathepsin L from human kidneyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed