Compile Data Set for Download or QSAR
Report error Found 5 Enz. Inhib. hit(s) with all data for entry = 3966
TargetHIV-1 protease(Human immunodeficiency virus)
State University of New York

LigandPNGBDBM517(Crixivan | CHEMBL115 | L-735, 524 | MK639 | Indina...)
Affinity DataKi:  0.370nMAssay Description:Enzyme inhibition assay for silanediols, carbinols, and indinavir using assay system C.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/11/2011
Entry Details Article
PubMed
TargetHIV-1 protease(Human immunodeficiency virus)
State University of New York

LigandPNGBDBM40773(Silanediol, 17b)
Affinity DataKi:  2.70nMAssay Description:Enzyme inhibition assay for silanediols, carbinols, and indinavir using assay system C.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/11/2011
Entry Details Article
PubMed
TargetHIV-1 protease(Human immunodeficiency virus)
State University of New York

LigandPNGBDBM40774(Carbinol, 18b)
Affinity DataKi:  3.80nMAssay Description:Enzyme inhibition assay for silanediols, carbinols, and indinavir using assay system C.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/11/2011
Entry Details Article
PubMed
TargetHIV-1 protease(Human immunodeficiency virus)
State University of New York

LigandPNGBDBM40772(Silanediol, 17a)
Affinity DataKi:  3.20E+3nMAssay Description:Enzyme inhibition assay for silanediols, carbinols, and indinavir using assay system C.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/11/2011
Entry Details Article
PubMed
TargetHIV-1 protease(Human immunodeficiency virus)
State University of New York

LigandPNGBDBM40775(Carbinol, 18a)
Affinity DataKi:  3.20E+3nMAssay Description:Enzyme inhibition assay for silanediols, carbinols, and indinavir using assay system C.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/11/2011
Entry Details Article
PubMed