Compile Data Set for Download or QSAR
Report error Found 29 Enz. Inhib. hit(s) with all data for entry = 5337
TargetAlpha-2C adrenergic receptor(Human)
Novartis Pharma

Curated by PDSP Ki Database
LigandPNGBDBM50034043(CHEMBL14376 | 1-(4-{3-[4-(6-Fluoro-benzo[d]isoxazo...)
Affinity DataKi:  16.2nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Novartis Pharma

Curated by PDSP Ki Database
LigandPNGBDBM50034043(CHEMBL14376 | 1-(4-{3-[4-(6-Fluoro-benzo[d]isoxazo...)
Affinity DataKi:  21.4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Novartis Pharma

Curated by PDSP Ki Database
LigandPNGBDBM50034043(CHEMBL14376 | 1-(4-{3-[4-(6-Fluoro-benzo[d]isoxazo...)
Affinity DataKi:  63.1nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 7(Human)
Novartis Pharma

Curated by PDSP Ki Database
LigandPNGBDBM50034043(CHEMBL14376 | 1-(4-{3-[4-(6-Fluoro-benzo[d]isoxazo...)
Affinity DataKi:  112nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2012
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Human)
Novartis Pharma

Curated by PDSP Ki Database
LigandPNGBDBM50034043(CHEMBL14376 | 1-(4-{3-[4-(6-Fluoro-benzo[d]isoxazo...)
Affinity DataKi:  162nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2012
Entry Details Article
PubMed
TargetAlpha-2B adrenergic receptor(Human)
Novartis Pharma

Curated by PDSP Ki Database
LigandPNGBDBM50034043(CHEMBL14376 | 1-(4-{3-[4-(6-Fluoro-benzo[d]isoxazo...)
Affinity DataKi:  162nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2012
Entry Details Article
PubMed
TargetSodium-dependent noradrenaline transporter(Human)
Novartis Pharma

Curated by PDSP Ki Database
LigandPNGBDBM50034043(CHEMBL14376 | 1-(4-{3-[4-(6-Fluoro-benzo[d]isoxazo...)
Affinity DataKi:  1.48E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2012
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
Novartis Pharma

Curated by PDSP Ki Database
LigandPNGBDBM50034043(CHEMBL14376 | 1-(4-{3-[4-(6-Fluoro-benzo[d]isoxazo...)
Affinity DataKi:  2.95E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Human)
Novartis Pharma

Curated by PDSP Ki Database
LigandPNGBDBM50034043(CHEMBL14376 | 1-(4-{3-[4-(6-Fluoro-benzo[d]isoxazo...)
Affinity DataKi:  3.31E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
Novartis Pharma

Curated by PDSP Ki Database
LigandPNGBDBM50034043(CHEMBL14376 | 1-(4-{3-[4-(6-Fluoro-benzo[d]isoxazo...)
Affinity DataKi:  4.90E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M4(Human)
Novartis Pharma

Curated by PDSP Ki Database
LigandPNGBDBM50034043(CHEMBL14376 | 1-(4-{3-[4-(6-Fluoro-benzo[d]isoxazo...)
Affinity DataKi:  8.32E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2012
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Novartis Pharma

Curated by PDSP Ki Database
LigandPNGBDBM50034043(CHEMBL14376 | 1-(4-{3-[4-(6-Fluoro-benzo[d]isoxazo...)
Affinity DataKi:  9.33E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2012
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Novartis Pharma

Curated by PDSP Ki Database
LigandPNGBDBM50034043(CHEMBL14376 | 1-(4-{3-[4-(6-Fluoro-benzo[d]isoxazo...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
Novartis Pharma

Curated by PDSP Ki Database
LigandPNGBDBM50034043(CHEMBL14376 | 1-(4-{3-[4-(6-Fluoro-benzo[d]isoxazo...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2012
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
Novartis Pharma

Curated by PDSP Ki Database
LigandPNGBDBM50034043(CHEMBL14376 | 1-(4-{3-[4-(6-Fluoro-benzo[d]isoxazo...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
Novartis Pharma

Curated by PDSP Ki Database
LigandPNGBDBM50034043(CHEMBL14376 | 1-(4-{3-[4-(6-Fluoro-benzo[d]isoxazo...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Novartis Pharma

Curated by PDSP Ki Database
LigandPNGBDBM50034043(CHEMBL14376 | 1-(4-{3-[4-(6-Fluoro-benzo[d]isoxazo...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2012
Entry Details Article
PubMed
TargetNeuromedin-K receptor(Human)
Novartis Pharma

Curated by PDSP Ki Database
LigandPNGBDBM50034043(CHEMBL14376 | 1-(4-{3-[4-(6-Fluoro-benzo[d]isoxazo...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2012
Entry Details Article
PubMed
TargetSubstance-K receptor(Human)
Novartis Pharma

Curated by PDSP Ki Database
LigandPNGBDBM50034043(CHEMBL14376 | 1-(4-{3-[4-(6-Fluoro-benzo[d]isoxazo...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2012
Entry Details Article
PubMed
TargetSubstance-P receptor(Human)
Novartis Pharma

Curated by PDSP Ki Database
LigandPNGBDBM50034043(CHEMBL14376 | 1-(4-{3-[4-(6-Fluoro-benzo[d]isoxazo...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Novartis Pharma

Curated by PDSP Ki Database
LigandPNGBDBM50034043(CHEMBL14376 | 1-(4-{3-[4-(6-Fluoro-benzo[d]isoxazo...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2012
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Novartis Pharma

Curated by PDSP Ki Database
LigandPNGBDBM50034043(CHEMBL14376 | 1-(4-{3-[4-(6-Fluoro-benzo[d]isoxazo...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2012
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Novartis Pharma

Curated by PDSP Ki Database
LigandPNGBDBM50034043(CHEMBL14376 | 1-(4-{3-[4-(6-Fluoro-benzo[d]isoxazo...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Human)
Novartis Pharma

Curated by PDSP Ki Database
LigandPNGBDBM50034043(CHEMBL14376 | 1-(4-{3-[4-(6-Fluoro-benzo[d]isoxazo...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Human)
Novartis Pharma

Curated by PDSP Ki Database
LigandPNGBDBM50034043(CHEMBL14376 | 1-(4-{3-[4-(6-Fluoro-benzo[d]isoxazo...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2012
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Novartis Pharma

Curated by PDSP Ki Database
LigandPNGBDBM50034043(CHEMBL14376 | 1-(4-{3-[4-(6-Fluoro-benzo[d]isoxazo...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A(Human)
Novartis Pharma

Curated by PDSP Ki Database
LigandPNGBDBM50034043(CHEMBL14376 | 1-(4-{3-[4-(6-Fluoro-benzo[d]isoxazo...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2012
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Novartis Pharma

Curated by PDSP Ki Database
LigandPNGBDBM50034043(CHEMBL14376 | 1-(4-{3-[4-(6-Fluoro-benzo[d]isoxazo...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Novartis Pharma

Curated by PDSP Ki Database
LigandPNGBDBM50034043(CHEMBL14376 | 1-(4-{3-[4-(6-Fluoro-benzo[d]isoxazo...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2012
Entry Details Article
PubMed