Compile Data Set for Download or QSAR
Report error Found 18 Enz. Inhib. hit(s) with all data for entry = 50011418
TargetTubulin alpha-1A chain(Pig)
University of North Carolina

Curated by ChEMBL
LigandPNGBDBM50035218(podophyllotoxin | CHEMBL61 | Podophyllinic acid la...)
Affinity DataIC50: 460nMAssay Description:Inhibition of tubulin polymerization. (ITP)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTubulin alpha-1A chain(Pig)
University of North Carolina

Curated by ChEMBL
LigandPNGBDBM50005480(combretastin A4 | CHEMBL67 | 2-Methoxy-5-[2-(3,4,5...)
Affinity DataIC50: 530nMAssay Description:Inhibition of tubulin polymerization (ITP)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTubulin alpha-1A chain(Pig)
University of North Carolina

Curated by ChEMBL
LigandPNGBDBM50041119(2-(2-fluorophenyl)-6,7-methylenedioxyquinolin-4-on...)
Affinity DataIC50: 680nMAssay Description:Inhibition of tubulin polymerization (ITP)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTubulin alpha-1A chain(Pig)
University of North Carolina

Curated by ChEMBL
LigandPNGBDBM50014846(7alphaH-colchicine | (S)-N-(5,6,7,9-tetrahydro-1,2...)
Affinity DataIC50: 800nMAssay Description:Inhibition of tubulin polymerization (ITP)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTubulin alpha-1A chain(Pig)
University of North Carolina

Curated by ChEMBL
LigandPNGBDBM50106310(2,2-Dimethyl-propionic acid 6-(2-fluoro-phenyl)-8-...)
Affinity DataIC50: 3.20E+3nMAssay Description:Inhibition of tubulin polymerization. (ITP)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTubulin alpha-1A chain(Pig)
University of North Carolina

Curated by ChEMBL
LigandPNGBDBM50012666(2-Styryl-3H-quinazolin-4-one | CHEMBL47360 | 2-((E...)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of tubulin polymerization. (ITP)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTubulin alpha-1A chain(Pig)
University of North Carolina

Curated by ChEMBL
LigandPNGBDBM48563(CHEMBL277148 | MLS000084697 | cid_161091 | SMR0000...)
Affinity DataIC50: 7.30E+3nMAssay Description:Inhibition of tubulin polymerization (ITP)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTubulin alpha-1A chain(Pig)
University of North Carolina

Curated by ChEMBL
LigandPNGBDBM50106308(4-[6-(2-Fluoro-phenyl)-[1,3]dioxolo[4,5-g]quinolin...)
Affinity DataIC50: 1.20E+4nMAssay Description:Inhibition of tubulin polymerization. (ITP)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTubulin alpha-1A chain(Pig)
University of North Carolina

Curated by ChEMBL
LigandPNGBDBM50106307(2-Phenyl-2,3-dihydro-1H-quinazolin-4-one | CHEMBL1...)
Affinity DataIC50: 1.40E+4nMAssay Description:Inhibition of tubulin polymerization. (ITP)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTubulin alpha-1A chain(Pig)
University of North Carolina

Curated by ChEMBL
LigandPNGBDBM50106306([6-(2-Fluoro-phenyl)-[1,3]dioxolo[4,5-g]quinolin-8...)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of tubulin polymerization. (ITP)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTubulin alpha-1A chain(Pig)
University of North Carolina

Curated by ChEMBL
LigandPNGBDBM50106311(6-(2-Fluoro-phenyl)-5H-[1,3]dioxolo[4,5-g]quinolin...)
Affinity DataIC50: 2.40E+4nMAssay Description:Inhibition of tubulin polymerization. (ITP)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTubulin alpha-1A chain(Pig)
University of North Carolina

Curated by ChEMBL
LigandPNGBDBM50041119(2-(2-fluorophenyl)-6,7-methylenedioxyquinolin-4-on...)
Affinity DataIC50: 3.90E+4nMAssay Description:Percent inhibition of colchicine binding(ICB) at 5 uM [3H]colchicine concentrationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTubulin alpha-1A chain(Pig)
University of North Carolina

Curated by ChEMBL
LigandPNGBDBM50106303(4-[6-(2-Fluoro-phenyl)-[1,3]dioxolo[4,5-g]quinolin...)
Affinity DataIC50: 4.00E+4nMAssay Description:Inhibition of tubulin polymerization. (ITP)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTubulin alpha-1A chain(Pig)
University of North Carolina

Curated by ChEMBL
LigandPNGBDBM50044965(1-Methyl-2-phenyl-1H-quinolin-4-one | CHEMBL277048)
Affinity DataIC50: 4.00E+4nMAssay Description:Inhibition of tubulin polymerization. (ITP)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTubulin alpha-1A chain(Pig)
University of North Carolina

Curated by ChEMBL
LigandPNGBDBM50106305(2-Phenyl-3H-quinazolin-4-one | CHEMBL127066 | 2-ph...)
Affinity DataIC50: 4.00E+4nMAssay Description:Inhibition of tubulin polymerization. (ITP)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTubulin alpha-1A chain(Pig)
University of North Carolina

Curated by ChEMBL
LigandPNGBDBM50106304([6-(2-Fluoro-phenyl)-[1,3]dioxolo[4,5-g]quinolin-8...)
Affinity DataIC50: 4.00E+4nMAssay Description:Inhibition of tubulin polymerization. (ITP)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTubulin alpha-1A chain(Pig)
University of North Carolina

Curated by ChEMBL
LigandPNGBDBM50106309(2-(2-fluorophenyl)-6-(pyrrolidin-1-yl)quinolin-4(1...)
Affinity DataIC50: 7.60E+4nMAssay Description:Inhibition of colchicine binding(ICB). Tubulin concentration was 1 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTubulin alpha-1A chain(Pig)
University of North Carolina

Curated by ChEMBL
LigandPNGBDBM50106309(2-(2-fluorophenyl)-6-(pyrrolidin-1-yl)quinolin-4(1...)
Affinity DataIC50: 9.30E+4nMAssay Description:Inhibition of colchicine binding(ICB). [3H]colchicine concentration was 5 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed