Compile Data Set for Download or QSAR
Report error Found 18 Enz. Inhib. hit(s) with all data for entry = 50011408
TargetPotassium voltage-gated channel subfamily E/KQT member 1(Human)
Aventis Pharma Deutschland

Curated by ChEMBL
LigandPNGBDBM50106236((3R,4S)-Ethanesulfonic acid (6-benzyloxy-3-hydroxy...)
Affinity DataIC50: 50nMAssay Description:Inhibition of human IKs-channel expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily E/KQT member 1(Human)
Aventis Pharma Deutschland

Curated by ChEMBL
LigandPNGBDBM50099582(N-[(3R,4S)-3-Hydroxy-2,2-dimethyl-6-(4,4,4-trifluo...)
Affinity DataIC50: 120nMAssay Description:Inhibition of human IKs-channel expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily E/KQT member 1(Human)
Aventis Pharma Deutschland

Curated by ChEMBL
LigandPNGBDBM50106233(N-(6-Benzyloxy-3-hydroxy-2,2-dimethyl-chroman-4-yl...)
Affinity DataIC50: 200nMAssay Description:Inhibition of human IKs-channel expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily E/KQT member 1(Human)
Aventis Pharma Deutschland

Curated by ChEMBL
LigandPNGBDBM50106231(N-[3-Hydroxy-2,2-dimethyl-6-(4,4,4-trifluoro-butox...)
Affinity DataIC50: 240nMAssay Description:Inhibition of human IKs-channel expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily E/KQT member 1(Human)
Aventis Pharma Deutschland

Curated by ChEMBL
LigandPNGBDBM50106232(N-(6-Butoxy-3-hydroxy-2,2-dimethyl-chroman-4-yl)-N...)
Affinity DataIC50: 250nMAssay Description:Inhibition of human IKs-channel expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily E/KQT member 1(Human)
Aventis Pharma Deutschland

Curated by ChEMBL
LigandPNGBDBM50106237((3S,4R)-Ethanesulfonic acid (6-benzyloxy-3-hydroxy...)
Affinity DataIC50: 400nMAssay Description:Inhibition of human IKs-channel expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily E/KQT member 1(Human)
Aventis Pharma Deutschland

Curated by ChEMBL
LigandPNGBDBM50106234((3S,4R)-(+)-N-[3-Hydroxy-2,2-dimethyl-6-(4,4,4-tri...)
Affinity DataIC50: 440nMAssay Description:Inhibition of human IKs-channel expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily E/KQT member 1(Human)
Aventis Pharma Deutschland

Curated by ChEMBL
LigandPNGBDBM50106228((3R,4S)-Ethanesulfonic acid (6-fluoro-3-hydroxy-2,...)
Affinity DataIC50: 700nMAssay Description:Inhibition of human IKs-channel expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily E/KQT member 1(Human)
Aventis Pharma Deutschland

Curated by ChEMBL
LigandPNGBDBM50106235(N-(3-Hydroxy-2,2-dimethyl-6-propoxy-chroman-4-yl)-...)
Affinity DataIC50: 900nMAssay Description:Inhibition of human IKs-channel expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily E/KQT member 1(Human)
Aventis Pharma Deutschland

Curated by ChEMBL
LigandPNGBDBM50106226(N-(6-Chloro-3-hydroxy-2,2-dimethyl-chroman-4-yl)-N...)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of human IKs-channel expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily E/KQT member 1(Human)
Aventis Pharma Deutschland

Curated by ChEMBL
LigandPNGBDBM50106229(Ethanesulfonic acid (6-fluoro-3-hydroxy-2,2-dimeth...)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of human IKs-channel expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily E/KQT member 1(Human)
Aventis Pharma Deutschland

Curated by ChEMBL
LigandPNGBDBM50106223((3S,4R)-Ethanesulfonic acid (6-fluoro-3-hydroxy-2,...)
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition of human IKs-channel expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily E/KQT member 1(Human)
Aventis Pharma Deutschland

Curated by ChEMBL
LigandPNGBDBM50106224(Ethanesulfonic acid (3-hydroxy-2,2-dimethyl-chroma...)
Affinity DataIC50: 3.10E+3nMAssay Description:Inhibition of human IKs-channel expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily E/KQT member 1(Human)
Aventis Pharma Deutschland

Curated by ChEMBL
LigandPNGBDBM50099567(Ethanesulfonic acid (6-cyano-3-hydroxy-2,2-dimethy...)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of human IKs-channel expressed in Xenopus oocytes,(Experiment 2)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily E/KQT member 1(Human)
Aventis Pharma Deutschland

Curated by ChEMBL
LigandPNGBDBM50106227((3R,4S)-Ethanesulfonic acid (6-cyano-3-hydroxy-2,2...)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of human IKs-channel expressed in Xenopus oocytes,(Experiment 1)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily E/KQT member 1(Human)
Aventis Pharma Deutschland

Curated by ChEMBL
LigandPNGBDBM50106230(Ethanesulfonic acid (6-cyano-3-hydroxy-2,2-dimethy...)
Affinity DataIC50: 6.90E+3nMAssay Description:Inhibition of human IKs-channel expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily E/KQT member 1(Human)
Aventis Pharma Deutschland

Curated by ChEMBL
LigandPNGBDBM50099567(Ethanesulfonic acid (6-cyano-3-hydroxy-2,2-dimethy...)
Affinity DataIC50: 4.45E+4nMAssay Description:Inhibition of human IKs-channel expressed in Xenopus oocytes,(Experiment 1)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily E/KQT member 1(Human)
Aventis Pharma Deutschland

Curated by ChEMBL
LigandPNGBDBM50106225(Butane-1-sulfonic acid (6-cyano-3-hydroxy-2,2-dime...)
Affinity DataIC50: 5.80E+4nMAssay Description:Inhibition of human IKs-channel expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed