Compile Data Set for Download or QSAR
Report error Found 36 Enz. Inhib. hit(s) with all data for entry = 50011358
TargetMuscarinic acetylcholine receptor M1(Human)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50004665(1-[4-(2-oxo-pyrrolidin-1-yl)-but-2-ynyl]-pyrrolidi...)
Affinity DataIC50: 2.30nMAssay Description:Ability to displace [3H]oxotremorine from Muscarinic acetylcholine receptor M1 expressed in CHO cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50105712(3-[(Z)-3-Chloro-isoxazol-5-ylmethoxyimino]-1-azoni...)
Affinity DataIC50: 23nMAssay Description:Ability to displace [3H]oxotremorine from Muscarinic acetylcholine receptor M1 expressed in CHO cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50105708(3-[(3-Chloro-isoxazol-5-ylmethoxyimino)-methyl]-1-...)
Affinity DataIC50: 44nMAssay Description:Ability to displace [3H]oxotremorine from Muscarinic acetylcholine receptor M1 expressed in CHO cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50105710(3-[(Z)-3-Chloro-isoxazol-5-ylmethoxyimino]-1-azoni...)
Affinity DataIC50: 57nMAssay Description:Ability to displace [3H]oxotremorine from Muscarinic acetylcholine receptor M1 expressed in CHO cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50105721(3-[(Z)-3-Bromo-isoxazol-5-ylmethoxyimino]-1-azonia...)
Affinity DataIC50: 72nMAssay Description:Ability to displace [3H]oxotremorine from Muscarinic acetylcholine receptor M1 expressed in CHO cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50105716(3-[(Z)-3-Bromo-isoxazol-5-ylmethoxyimino]-1-azonia...)
Affinity DataIC50: 79nMAssay Description:Ability to displace [3H]oxotremorine from Muscarinic acetylcholine receptor M1 expressed in CHO cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50105713(3-[(Z)-3-Cyano-isoxazol-5-ylmethoxyimino]-1-azonia...)
Affinity DataIC50: 81nMAssay Description:Ability to displace [3H]oxotremorine from Muscarinic acetylcholine receptor M1 expressed in CHO cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50105722(3-[(Z)-3-Cyano-isoxazol-5-ylmethoxyimino]-1-azonia...)
Affinity DataIC50: 82nMAssay Description:Ability to displace [3H]oxotremorine from Muscarinic acetylcholine receptor M1 expressed in CHO cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM46858(cid_9301 | ARECOLINE HYDROBROMIDE | SMR000058258 |...)
Affinity DataIC50: 115nMAssay Description:Ability to displace [3H]oxotremorine from Muscarinic acetylcholine receptor M1 expressed in CHO cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50105717(3-[(Z)-3-Methoxy-isoxazol-5-ylmethoxyimino]-1-azon...)
Affinity DataIC50: 131nMAssay Description:Ability to displace [3H]oxotremorine from Muscarinic acetylcholine receptor M1 expressed in CHO cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50105720(3-[(3-Methoxy-isoxazol-5-ylmethoxyimino)-methyl]-1...)
Affinity DataIC50: 287nMAssay Description:Ability to displace [3H]oxotremorine from Muscarinic acetylcholine receptor M1 expressed in CHO cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50105709(3-[(3-Cyano-isoxazol-5-ylmethoxyimino)-methyl]-1-a...)
Affinity DataIC50: 341nMAssay Description:Ability to displace [3H]oxotremorine from Muscarinic acetylcholine receptor M1 expressed in CHO cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50105718(3-[(Z)-3-Methoxy-isoxazol-5-ylmethoxyimino]-1-azon...)
Affinity DataIC50: 362nMAssay Description:Ability to displace [3H]oxotremorine from Muscarinic acetylcholine receptor M1 expressed in CHO cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50105715(3-[(3-Bromo-isoxazol-5-ylmethoxyimino)-methyl]-1-a...)
Affinity DataIC50: 385nMAssay Description:Ability to displace [3H]oxotremorine from Muscarinic acetylcholine receptor M1 expressed in CHO cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50105719(3-[(3-Chloro-isoxazol-5-ylmethoxyimino)-methyl]-1-...)
Affinity DataIC50: 795nMAssay Description:Ability to displace [3H]oxotremorine from Muscarinic acetylcholine receptor M1 expressed in CHO cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50105707(3-[(3-Bromo-isoxazol-5-ylmethoxyimino)-methyl]-1-a...)
Affinity DataIC50: 1.22E+3nMAssay Description:Ability to displace [3H]oxotremorine from Muscarinic acetylcholine receptor M1 expressed in CHO cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50105714(3-[(3-Methoxy-isoxazol-5-ylmethoxyimino)-methyl]-1...)
Affinity DataIC50: 1.64E+3nMAssay Description:Ability to displace [3H]oxotremorine from Muscarinic acetylcholine receptor M1 expressed in CHO cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50105711(3-[(3-Cyano-isoxazol-5-ylmethoxyimino)-methyl]-1-a...)
Affinity DataIC50: 1.86E+3nMAssay Description:Ability to displace [3H]oxotremorine from Muscarinic acetylcholine receptor M1 expressed in CHO cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50105707(3-[(3-Bromo-isoxazol-5-ylmethoxyimino)-methyl]-1-a...)
Affinity DataIC50: 8.40E+3nMAssay Description:Ability to displace [3H]N-methylscopolamine from Muscarinic acetylcholine receptor M1 expressed in CHO cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50105713(3-[(Z)-3-Cyano-isoxazol-5-ylmethoxyimino]-1-azonia...)
Affinity DataIC50: 8.70E+3nMAssay Description:Ability to displace [3H]N-methylscopolamine from Muscarinic acetylcholine receptor M1 expressed in CHO cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50105721(3-[(Z)-3-Bromo-isoxazol-5-ylmethoxyimino]-1-azonia...)
Affinity DataIC50: 1.15E+4nMAssay Description:Ability to displace [3H]N-methylscopolamine from Muscarinic acetylcholine receptor M1 expressed in CHO cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50105710(3-[(Z)-3-Chloro-isoxazol-5-ylmethoxyimino]-1-azoni...)
Affinity DataIC50: 1.38E+4nMAssay Description:Ability to displace [3H]N-methylscopolamine from Muscarinic acetylcholine receptor M1 expressed in CHO cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50105708(3-[(3-Chloro-isoxazol-5-ylmethoxyimino)-methyl]-1-...)
Affinity DataIC50: 1.49E+4nMAssay Description:Ability to displace [3H]N-methylscopolamine from Muscarinic acetylcholine receptor M1 expressed in CHO cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50105720(3-[(3-Methoxy-isoxazol-5-ylmethoxyimino)-methyl]-1...)
Affinity DataIC50: 1.67E+4nMAssay Description:Ability to displace [3H]N-methylscopolamine from Muscarinic acetylcholine receptor M1 expressed in CHO cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50105715(3-[(3-Bromo-isoxazol-5-ylmethoxyimino)-methyl]-1-a...)
Affinity DataIC50: 1.77E+4nMAssay Description:Ability to displace [3H]N-methylscopolamine from Muscarinic acetylcholine receptor M1 expressed in CHO cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50105719(3-[(3-Chloro-isoxazol-5-ylmethoxyimino)-methyl]-1-...)
Affinity DataIC50: 2.35E+4nMAssay Description:Ability to displace [3H]N-methylscopolamine from Muscarinic acetylcholine receptor M1 expressed in CHO cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50004665(1-[4-(2-oxo-pyrrolidin-1-yl)-but-2-ynyl]-pyrrolidi...)
Affinity DataIC50: 2.71E+4nMAssay Description:Ability to displace [3H]N-methylscopolamine from Muscarinic acetylcholine receptor M1 expressed in CHO cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50105714(3-[(3-Methoxy-isoxazol-5-ylmethoxyimino)-methyl]-1...)
Affinity DataIC50: 2.95E+4nMAssay Description:Ability to displace [3H]N-methylscopolamine from Muscarinic acetylcholine receptor M1 expressed in CHO cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50105722(3-[(Z)-3-Cyano-isoxazol-5-ylmethoxyimino]-1-azonia...)
Affinity DataIC50: 3.25E+4nMAssay Description:Ability to displace [3H]N-methylscopolamine from Muscarinic acetylcholine receptor M1 expressed in CHO cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50105718(3-[(Z)-3-Methoxy-isoxazol-5-ylmethoxyimino]-1-azon...)
Affinity DataIC50: 3.56E+4nMAssay Description:Ability to displace [3H]N-methylscopolamine from Muscarinic acetylcholine receptor M1 expressed in CHO cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50105712(3-[(Z)-3-Chloro-isoxazol-5-ylmethoxyimino]-1-azoni...)
Affinity DataIC50: 3.63E+4nMAssay Description:Ability to displace [3H]N-methylscopolamine from Muscarinic acetylcholine receptor M1 expressed in CHO cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50105717(3-[(Z)-3-Methoxy-isoxazol-5-ylmethoxyimino]-1-azon...)
Affinity DataIC50: 4.05E+4nMAssay Description:Ability to displace [3H]N-methylscopolamine from Muscarinic acetylcholine receptor M1 expressed in CHO cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50105716(3-[(Z)-3-Bromo-isoxazol-5-ylmethoxyimino]-1-azonia...)
Affinity DataIC50: 4.88E+4nMAssay Description:Ability to displace [3H]N-methylscopolamine from Muscarinic acetylcholine receptor M1 expressed in CHO cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM46858(cid_9301 | ARECOLINE HYDROBROMIDE | SMR000058258 |...)
Affinity DataIC50: 1.16E+5nMAssay Description:Ability to displace [3H]N-methylscopolamine from Muscarinic acetylcholine receptor M1 expressed in CHO cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50105709(3-[(3-Cyano-isoxazol-5-ylmethoxyimino)-methyl]-1-a...)
Affinity DataIC50: 1.33E+5nMAssay Description:Ability to displace [3H]N-methylscopolamine from Muscarinic acetylcholine receptor M1 expressed in CHO cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50105711(3-[(3-Cyano-isoxazol-5-ylmethoxyimino)-methyl]-1-a...)
Affinity DataIC50: 1.90E+5nMAssay Description:Ability to displace [3H]N-methylscopolamine from Muscarinic acetylcholine receptor M1 expressed in CHO cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed