Compile Data Set for Download or QSAR
Report error Found 16 Enz. Inhib. hit(s) with all data for entry = 50011262
TargetEstrogen receptor beta(Human)
University of Illinois

Curated by ChEMBL
LigandPNGBDBM50104326(4-{3-(4-hydroxy-phenyl)-4-ethyl-5-[4-(2-piperidin-...)
Affinity DataKi:  0.0600nMAssay Description:Displacement of [3H]estradiol from Estrogen receptor betaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
University of Illinois

Curated by ChEMBL
LigandPNGBDBM50104326(4-{3-(4-hydroxy-phenyl)-4-ethyl-5-[4-(2-piperidin-...)
Affinity DataKi:  0.360nMAssay Description:Displacement of [3H]estradiol from Estrogen receptor alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEstrogen receptor beta(Human)
University of Illinois

Curated by ChEMBL
LigandPNGBDBM50104329(4-{3-Ethyl-5-phenyl-4-[4-(2-piperidin-1-yl-ethoxy)...)
Affinity DataKi:  0.430nMAssay Description:Displacement of [3H]estradiol from Estrogen receptor betaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEstrogen receptor beta(Human)
University of Illinois

Curated by ChEMBL
LigandPNGBDBM50104324(4-{5-(4-hydroxy-phenyl)-4-methyl-3-[4-(2-piperidin...)
Affinity DataKi:  0.470nMAssay Description:Displacement of [3H]estradiol from Estrogen receptor betaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEstrogen receptor beta(Human)
University of Illinois

Curated by ChEMBL
LigandPNGBDBM50104325(4-[5-(4-hydroxy-phenyl)-4-ethyl-3-(4-methoxy-pheny...)
Affinity DataKi:  0.910nMAssay Description:Displacement of [3H]estradiol from Estrogen receptor betaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
University of Illinois

Curated by ChEMBL
LigandPNGBDBM50104325(4-[5-(4-hydroxy-phenyl)-4-ethyl-3-(4-methoxy-pheny...)
Affinity DataKi:  2.5nMAssay Description:Displacement of [3H]estradiol from Estrogen receptor alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEstrogen receptor beta(Human)
University of Illinois

Curated by ChEMBL
LigandPNGBDBM50104327(4-{5-(4-hydroxy-phenyl)-4-ethyl-3-[4-(2-piperidin-...)
Affinity DataKi:  3.10nMAssay Description:Displacement of [3H]estradiol from Estrogen receptor betaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
University of Illinois

Curated by ChEMBL
LigandPNGBDBM50104329(4-{3-Ethyl-5-phenyl-4-[4-(2-piperidin-1-yl-ethoxy)...)
Affinity DataKi:  3.80nMAssay Description:Displacement of [3H]estradiol from Estrogen receptor alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEstrogen receptor beta(Human)
University of Illinois

Curated by ChEMBL
LigandPNGBDBM50104323(4-{5-(4-hydroxy-phenyl)-4-propyl-3-[4-(2-piperidin...)
Affinity DataKi:  4nMAssay Description:Displacement of [3H]estradiol from Estrogen receptor betaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEstrogen receptor beta(Human)
University of Illinois

Curated by ChEMBL
LigandPNGBDBM50104328(4-{4-Ethyl-5-phenyl-3-[4-(2-piperidin-1-yl-ethoxy)...)
Affinity DataKi:  20nMAssay Description:Displacement of [3H]estradiol from Estrogen receptor betaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
University of Illinois

Curated by ChEMBL
LigandPNGBDBM50104324(4-{5-(4-hydroxy-phenyl)-4-methyl-3-[4-(2-piperidin...)
Affinity DataKi:  32nMAssay Description:Displacement of [3H]estradiol from Estrogen receptor alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
University of Illinois

Curated by ChEMBL
LigandPNGBDBM50104323(4-{5-(4-hydroxy-phenyl)-4-propyl-3-[4-(2-piperidin...)
Affinity DataKi:  34nMAssay Description:Displacement of [3H]estradiol from Estrogen receptor alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
University of Illinois

Curated by ChEMBL
LigandPNGBDBM50104328(4-{4-Ethyl-5-phenyl-3-[4-(2-piperidin-1-yl-ethoxy)...)
Affinity DataKi:  60nMAssay Description:Displacement of [3H]estradiol from Estrogen receptor alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
University of Illinois

Curated by ChEMBL
LigandPNGBDBM50104327(4-{5-(4-hydroxy-phenyl)-4-ethyl-3-[4-(2-piperidin-...)
Affinity DataIC50: 65nMAssay Description:Displacement of [3H]estradiol from Estrogen receptor alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
University of Illinois

Curated by ChEMBL
LigandPNGBDBM50104327(4-{5-(4-hydroxy-phenyl)-4-ethyl-3-[4-(2-piperidin-...)
Affinity DataKi:  75nMAssay Description:Displacement of [3H]estradiol from Estrogen receptor alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEstrogen receptor beta(Human)
University of Illinois

Curated by ChEMBL
LigandPNGBDBM50104327(4-{5-(4-hydroxy-phenyl)-4-ethyl-3-[4-(2-piperidin-...)
Affinity DataIC50: 480nMAssay Description:Inhibitory activity against Estrogen receptor betaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed