Compile Data Set for Download or QSAR
Report error Found 42 Enz. Inhib. hit(s) with all data for entry = 50011239
TargetGlucagon receptor(Rat)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50104096BDBM50104096(3-Chloro-4-hydroxy-benzoic acid (4-hydroxy-naphtha...)
Affinity DataIC50: 27nMAssay Description:Binding affinity towards rat Glucagon ReceptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50104096BDBM50104096(3-Chloro-4-hydroxy-benzoic acid (4-hydroxy-naphtha...)
Affinity DataIC50: 200nMAssay Description:Binding affinity towards human Glucagon Receptor by the displacement of [125I]-glucagonMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50104082BDBM50104082(3-Fluoro-4-hydroxy-benzoic acid (4-hydroxy-naphtha...)
Affinity DataIC50: 390nMAssay Description:Binding affinity for human Glucagon ReceptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50104080BDBM50104080(4-Hydroxy-3-methoxy-benzoic acid (4-hydroxy-naphth...)
Affinity DataIC50: 720nMAssay Description:Binding affinity for human Glucagon ReceptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50104064BDBM50104064(3-Bromo-4-hydroxy-benzoic acid (4-hydroxy-naphthal...)
Affinity DataIC50: 830nMAssay Description:Binding affinity for human Glucagon ReceptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50104088BDBM50104088(4-Hydroxy-benzoic acid (4-hydroxy-naphthalen-1-ylm...)
Affinity DataIC50: 1.20E+3nMAssay Description:Binding affinity for human Glucagon ReceptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50104063BDBM50104063(4-Hydroxy-benzoic acid naphthalen-1-ylmethylene-hy...)
Affinity DataIC50: 1.80E+3nMAssay Description:Binding affinity for human Glucagon ReceptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50104099BDBM50104099(3-Amino-4-hydroxy-benzoic acid (4-hydroxy-naphthal...)
Affinity DataIC50: 2.00E+3nMAssay Description:Binding affinity for human Glucagon ReceptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50104081BDBM50104081(4-Hydroxy-3-methoxy-benzoic acid (4-methoxy-naphth...)
Affinity DataIC50: 2.90E+3nMAssay Description:Binding affinity for human Glucagon ReceptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50104068BDBM50104068(3,4-Dihydroxy-benzoic acid (4-hydroxy-naphthalen-1...)
Affinity DataIC50: 3.40E+3nMAssay Description:Binding affinity for human Glucagon ReceptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50104094BDBM50104094(4-Hydroxy-3-methoxy-benzoic acid naphthalen-1-ylme...)
Affinity DataIC50: 4.80E+3nMAssay Description:Binding affinity for human Glucagon ReceptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50104066BDBM50104066(4-Hydroxy-3-methoxy-benzoic acid [3-(3-trifluorome...)
Affinity DataIC50: 4.90E+3nMAssay Description:Binding affinity for human Glucagon ReceptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50104069BDBM50104069(4-Hydroxy-benzoic acid (4-methoxy-naphthalen-1-ylm...)
Affinity DataIC50: 4.90E+3nMAssay Description:Binding affinity for human Glucagon ReceptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50104077BDBM50104077(4-Hydroxy-3-methoxy-benzoic acid (9-ethyl-9H-carba...)
Affinity DataIC50: 6.30E+3nMAssay Description:Binding affinity for human Glucagon ReceptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50104061BDBM50104061(4-Hydroxy-3-methoxy-benzoic acid (4-dimethylamino-...)
Affinity DataIC50: 8.10E+3nMAssay Description:Binding affinity for human Glucagon ReceptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50104071BDBM50104071(4-Hydroxy-3-methoxy-benzoic acid quinolin-4-ylmeth...)
Affinity DataIC50: 1.00E+4nMAssay Description:Binding affinity for human Glucagon ReceptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50104083BDBM50104083(4-Hydroxy-3-methoxy-benzoic acid [5-(3-chloro-4-me...)
Affinity DataIC50: 1.20E+4nMAssay Description:Binding affinity for human Glucagon ReceptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50104073BDBM50104073(4-Hydroxy-3-methoxy-benzoic acid (1H-indol-3-ylmet...)
Affinity DataIC50: 2.30E+4nMAssay Description:Binding affinity for human Glucagon ReceptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50104087BDBM50104087(4-Hydroxy-3-methoxy-benzoic acid biphenyl-4-ylmeth...)
Affinity DataIC50: 2.60E+4nMAssay Description:Binding affinity for human Glucagon ReceptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50104086BDBM50104086(2,4-Dihydroxy-benzoic acid (4-hydroxy-naphthalen-1...)
Affinity DataIC50: 2.80E+4nMAssay Description:Binding affinity for human Glucagon ReceptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50104093BDBM50104093(4-Hydroxy-3-methoxy-benzoic acid (4-tert-butyl-ben...)
Affinity DataIC50: 2.90E+4nMAssay Description:Binding affinity for human Glucagon ReceptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50104089BDBM50104089(3,5-Dichloro-4-hydroxy-benzoic acid (4-hydroxy-nap...)
Affinity DataIC50: 3.40E+4nMAssay Description:Binding affinity for human Glucagon ReceptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50104079BDBM50104079(4-Hydroxy-3-methoxy-benzoic acid (4-isopropyl-benz...)
Affinity DataIC50: 4.30E+4nMAssay Description:Binding affinity for human Glucagon ReceptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50104091BDBM50104091(4-Hydroxy-3-methoxy-benzoic acid (4-trifluorometho...)
Affinity DataIC50: 4.30E+4nMAssay Description:Binding affinity for human Glucagon ReceptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50104097BDBM50104097(3-Chloro-4-hydroxy-5-methoxy-benzoic acid(4-hydrox...)
Affinity DataIC50: 6.00E+4nMAssay Description:Binding affinity for human Glucagon ReceptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50104098BDBM50104098(5-Hydroxy-1H-indole-2-carboxylic acid (4-hydroxy-n...)
Affinity DataIC50: 1.00E+5nMAssay Description:Binding affinity for human Glucagon ReceptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50104067BDBM50104067(3-Methoxy-benzoic acid (4-methoxy-naphthalen-1-ylm...)
Affinity DataIC50: 1.00E+5nMAssay Description:Binding affinity for human Glucagon ReceptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50104095BDBM50104095(Naphthalene-1-carboxylic acid (4-hydroxy-3-methoxy...)
Affinity DataIC50: 1.00E+5nMAssay Description:Binding affinity for human Glucagon ReceptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50104062BDBM50104062(4-Hydroxy-3-methoxy-benzoic acid (4-methoxy-benzyl...)
Affinity DataIC50: 1.00E+5nMAssay Description:Binding affinity for human Glucagon ReceptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50104092BDBM50104092(4-Hydroxy-3-methoxy-benzoic acid (1-naphthalen-1-y...)
Affinity DataIC50: 1.00E+5nMAssay Description:Binding affinity for human Glucagon ReceptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50104065BDBM50104065(4-Hydroxy-benzoic acid N'-naphthalen-1-ylmethyl-hy...)
Affinity DataIC50: 1.00E+5nMAssay Description:Binding affinity for human Glucagon ReceptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50104090BDBM50104090(6-Hydroxy-nicotinic acid (4-hydroxy-naphthalen-1-y...)
Affinity DataIC50: 1.00E+5nMAssay Description:Binding affinity for human Glucagon ReceptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50104084BDBM50104084(1H-Indole-5-carboxylic acid (4-hydroxy-naphthalen-...)
Affinity DataIC50: 1.00E+5nMAssay Description:Binding affinity for human Glucagon ReceptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50104085BDBM50104085(4-Hydroxy-3-methoxy-benzoic acid (4-styryl-benzyli...)
Affinity DataIC50: 1.00E+5nMAssay Description:Binding affinity for human Glucagon ReceptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50104078BDBM50104078(4-(4-Hydroxy-naphthalen-1-ylmethylene-hydrazinocar...)
Affinity DataIC50: 1.00E+5nMAssay Description:Binding affinity for human Glucagon ReceptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50104075BDBM50104075(4-Hydroxy-3-methoxy-benzoic acid (2,4-dioxo-1,2,3,...)
Affinity DataIC50: 1.00E+5nMAssay Description:Binding affinity for human Glucagon ReceptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50104072BDBM50104072(4-Hydroxy-3-methoxy-benzoic acid (5-methyl-1H-imid...)
Affinity DataIC50: 1.00E+5nMAssay Description:Binding affinity for human Glucagon ReceptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50104076BDBM50104076(Quinoxaline-6-carboxylic acid (4-hydroxy-naphthale...)
Affinity DataIC50: 1.00E+5nMAssay Description:Binding affinity for human Glucagon ReceptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50104074BDBM50104074(4-Hydroxy-3-methoxy-benzoic acid (3-hydroxy-4-meth...)
Affinity DataIC50: 1.00E+5nMAssay Description:Binding affinity for human Glucagon ReceptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50104070BDBM50104070(4-Hydroxy-3-morpholin-4-ylmethyl-benzoic acid (4-h...)
Affinity DataIC50: 1.00E+5nMAssay Description:Binding affinity for human Glucagon ReceptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50104101BDBM50104101(4-Hydroxy-3-methoxy-benzoic acid (4-hydroxy-benzyl...)
Affinity DataIC50: 1.00E+5nMAssay Description:Binding affinity for human Glucagon ReceptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50104100BDBM50104100(4-Amino-benzoic acid (4-hydroxy-naphthalen-1-ylmet...)
Affinity DataIC50: 1.00E+5nMAssay Description:Binding affinity for human Glucagon ReceptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed