Compile Data Set for Download or QSAR
Report error Found 16 Enz. Inhib. hit(s) with all data for entry = 50003576
TargetNischarin(Human)
Louis Pasteur University

Curated by ChEMBL
LigandPNGBDBM50070328(CHEBI:8862 | Rilmenidine)
Affinity DataKi:  74nMAssay Description:Displacement of [3H]clonidine from imidazoline receptor I-1 of bovine chromaffin cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetNischarin(Human)
Louis Pasteur University

Curated by ChEMBL
LigandPNGBDBM50473238(CHEMBL40399)
Affinity DataKi:  170nMAssay Description:Displacement of [3H]clonidine from imidazoline receptor I-1 of bovine chromaffin cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetNischarin(Human)
Louis Pasteur University

Curated by ChEMBL
LigandPNGBDBM50473241(CHEMBL288951)
Affinity DataKi:  513nMAssay Description:Displacement of [3H]clonidine from imidazoline receptor I-1 of bovine chromaffin cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetNischarin(Human)
Louis Pasteur University

Curated by ChEMBL
LigandPNGBDBM50070357(CHEMBL288139)
Affinity DataKi:  537nMAssay Description:Displacement of [3H]clonidine from imidazoline receptor I-1 of bovine chromaffin cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetNischarin(Human)
Louis Pasteur University

Curated by ChEMBL
LigandPNGBDBM50473239(CHEMBL442156)
Affinity DataKi:  646nMAssay Description:Displacement of [3H]clonidine from imidazoline receptor I-1 of bovine chromaffin cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetNischarin(Human)
Louis Pasteur University

Curated by ChEMBL
LigandPNGBDBM50473240(CHEMBL40337)
Affinity DataKi:  1.59E+3nMAssay Description:Displacement of [3H]clonidine from imidazoline receptor I-1 of bovine chromaffin cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A/B(Human)
Louis Pasteur University

Curated by ChEMBL
LigandPNGBDBM50070357(CHEMBL288139)
Affinity DataKi: <1.00E+4nMAssay Description:Displacement of [3H]idazoxan from I2 imidazoline binding sites (I2Bs) of rabbit renal cortex membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetNischarin(Human)
Louis Pasteur University

Curated by ChEMBL
LigandPNGBDBM50473237(CHEMBL40393)
Affinity DataKi: <1.00E+4nMAssay Description:Displacement of [3H]clonidine from imidazoline receptor I-1 of bovine chromaffin cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A/B(Human)
Louis Pasteur University

Curated by ChEMBL
LigandPNGBDBM50473238(CHEMBL40399)
Affinity DataKi: <1.00E+4nMAssay Description:Displacement of [3H]idazoxan from I2 imidazoline binding sites (I2Bs) of rabbit renal cortex membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A/B(Human)
Louis Pasteur University

Curated by ChEMBL
LigandPNGBDBM50070328(CHEBI:8862 | Rilmenidine)
Affinity DataKi: <1.00E+4nMAssay Description:Displacement of [3H]idazoxan from I2 imidazoline binding sites (I2Bs) of rabbit renal cortex membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A/B(Human)
Louis Pasteur University

Curated by ChEMBL
LigandPNGBDBM50473237(CHEMBL40393)
Affinity DataKi: <1.00E+4nMAssay Description:Displacement of [3H]idazoxan from I2 imidazoline binding sites (I2Bs) of rabbit renal cortex membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A/B(Human)
Louis Pasteur University

Curated by ChEMBL
LigandPNGBDBM50473241(CHEMBL288951)
Affinity DataKi: <1.00E+4nMAssay Description:Displacement of [3H]idazoxan from I2 imidazoline binding sites (I2Bs) of rabbit renal cortex membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A/B(Human)
Louis Pasteur University

Curated by ChEMBL
LigandPNGBDBM50473239(CHEMBL442156)
Affinity DataKi: <1.00E+4nMAssay Description:Displacement of [3H]idazoxan from I2 imidazoline binding sites (I2Bs) of rabbit renal cortex membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A/B(Human)
Louis Pasteur University

Curated by ChEMBL
LigandPNGBDBM50473242(CHEMBL40287)
Affinity DataKi: <1.00E+4nMAssay Description:Displacement of [3H]idazoxan from I2 imidazoline binding sites (I2Bs) of rabbit renal cortex membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A/B(Human)
Louis Pasteur University

Curated by ChEMBL
LigandPNGBDBM50473240(CHEMBL40337)
Affinity DataKi: <1.00E+4nMAssay Description:Displacement of [3H]idazoxan from I2 imidazoline binding sites (I2Bs) of rabbit renal cortex membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetNischarin(Human)
Louis Pasteur University

Curated by ChEMBL
LigandPNGBDBM50473242(CHEMBL40287)
Affinity DataKi: <1.00E+4nMAssay Description:Displacement of [3H]clonidine from imidazoline receptor I-1 of bovine chromaffin cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed