Compile Data Set for Download or QSAR
Report error Found 42 Enz. Inhib. hit(s) with all data for entry = 50010831
TargetNeuropeptide Y receptor type 2(Human)
University of Cincinnati and Va Medical Centers

Curated by ChEMBL
LigandPNGBDBM50409214(GR-231118 | CHEMBL2110365)
Affinity DataEC50:  983nMAssay Description:Agonist potency for the inhibition of Forskolin stimulated cAMP synthesis in cells expressing cloned Y2 receptorsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 4(Human)
University of Cincinnati and Va Medical Centers

Curated by ChEMBL
LigandPNGBDBM50099198(Tyr-Pro-Ser-Lys-Pro-Asp-Asn-Pro-Gly-Glu-Asp-Ala-Pr...)
Affinity DataEC50:  0.460nMAssay Description:Agonist potency for the inhibition of Forskolin stimulated cAMP synthesis in cells expressing cloned Y2 receptorsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
University of Cincinnati and Va Medical Centers

Curated by ChEMBL
LigandPNGBDBM50409214(GR-231118 | CHEMBL2110365)
Affinity DataEC50:  2.05E+3nMAssay Description:Agonist potency for the inhibition of Forskolin stimulated cAMP synthesis in cells expressing cloned Y5 receptorsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 4(Human)
University of Cincinnati and Va Medical Centers

Curated by ChEMBL
LigandPNGBDBM50099198(Tyr-Pro-Ser-Lys-Pro-Asp-Asn-Pro-Gly-Glu-Asp-Ala-Pr...)
Affinity DataEC50:  0.160nMAssay Description:Agonist potency for the inhibition of Forskolin stimulated cAMP synthesis in cells expressing cloned Y4 receptorsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 4(Human)
University of Cincinnati and Va Medical Centers

Curated by ChEMBL
LigandPNGBDBM50409214(GR-231118 | CHEMBL2110365)
Affinity DataEC50:  2.5nMAssay Description:Agonist potency for the inhibition of Forskolin stimulated cAMP synthesis in cells expressing cloned Y4 receptorsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
University of Cincinnati and Va Medical Centers

Curated by ChEMBL
LigandPNGBDBM50099198(Tyr-Pro-Ser-Lys-Pro-Asp-Asn-Pro-Gly-Glu-Asp-Ala-Pr...)
Affinity DataEC50:  7.89nMAssay Description:Agonist potency for the inhibition of Forskolin stimulated cAMP synthesis in cells expressing cloned Y5 receptorsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 1(Human)
University of Cincinnati and Va Medical Centers

Curated by ChEMBL
LigandPNGBDBM50409214(GR-231118 | CHEMBL2110365)
Affinity DataKi:  0.0700nMAssay Description:Affinity for cloned Y1 receptor using [125I]PYY as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 4(Human)
University of Cincinnati and Va Medical Centers

Curated by ChEMBL
LigandPNGBDBM50099198(Tyr-Pro-Ser-Lys-Pro-Asp-Asn-Pro-Gly-Glu-Asp-Ala-Pr...)
Affinity DataKi:  0.0800nMAssay Description:Affinity for cloned Y4 receptor using [125I]PP as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 2(Human)
University of Cincinnati and Va Medical Centers

Curated by ChEMBL
LigandPNGBDBM50099198(Tyr-Pro-Ser-Lys-Pro-Asp-Asn-Pro-Gly-Glu-Asp-Ala-Pr...)
Affinity DataKi:  0.230nMAssay Description:Affinity for cloned Y2 receptor using [125I]PYY as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 4(Human)
University of Cincinnati and Va Medical Centers

Curated by ChEMBL
LigandPNGBDBM50409214(GR-231118 | CHEMBL2110365)
Affinity DataKi:  0.260nMAssay Description:Affinity for cloned Y4 receptor using [125I]PP as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 1(Human)
University of Cincinnati and Va Medical Centers

Curated by ChEMBL
LigandPNGBDBM50099197(Ile-Glu-Pro-Dpr-Tyr-Arg-Leu-Arg-Tyr-OMeIle-Glu-Pro...)
Affinity DataKi:  0.270nMAssay Description:Affinity for cloned Y1 receptor using [125I]PYY as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 1(Human)
University of Cincinnati and Va Medical Centers

Curated by ChEMBL
LigandPNGBDBM50099200(Ile-Glu-Pro-Dpr-Tyr-Arg-Leu-Arg-(CH2-NH)-Tyr-NH2Il...)
Affinity DataKi:  0.460nMAssay Description:Affinity for cloned Y1 receptor using [125I]PYY as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 1(Human)
University of Cincinnati and Va Medical Centers

Curated by ChEMBL
LigandPNGBDBM50099198(Tyr-Pro-Ser-Lys-Pro-Asp-Asn-Pro-Gly-Glu-Asp-Ala-Pr...)
Affinity DataKi:  0.520nMAssay Description:Affinity for cloned Y1 receptor using [125I]PYY as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
University of Cincinnati and Va Medical Centers

Curated by ChEMBL
LigandPNGBDBM50099198(Tyr-Pro-Ser-Lys-Pro-Asp-Asn-Pro-Gly-Glu-Asp-Ala-Pr...)
Affinity DataKi:  2.21nMAssay Description:Affinity for cloned Y5 receptor using [125I]PYY as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 1(Human)
University of Cincinnati and Va Medical Centers

Curated by ChEMBL
LigandPNGBDBM50099201(Ile-Asn-Pro-Cys-Tyr-Arg-Leu-Arg-(CH2-NH)-Tyr-NH2Il...)
Affinity DataKi:  2.30nMAssay Description:Affinity for cloned Y1 receptor using [125I]PYY as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 1(Human)
University of Cincinnati and Va Medical Centers

Curated by ChEMBL
LigandPNGBDBM50099199(Ile-Asn-Pro-Cys-Tyr-Arg-Leu-Arg-Tyr-OMeIle-Asn-Pro...)
Affinity DataKi:  4.80nMAssay Description:Affinity for cloned Y1 receptor using [125I]PYY as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 1(Human)
University of Cincinnati and Va Medical Centers

Curated by ChEMBL
LigandPNGBDBM50034121(Ile-Asn-Pro-Ile-Tyr-Arg-Leu-Arg-Tyr-NH2 | CHEMBL38...)
Affinity DataKi:  5nMAssay Description:Affinity for cloned Y1 receptor using [125I]PYY as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 4(Human)
University of Cincinnati and Va Medical Centers

Curated by ChEMBL
LigandPNGBDBM50034121(Ile-Asn-Pro-Ile-Tyr-Arg-Leu-Arg-Tyr-NH2 | CHEMBL38...)
Affinity DataKi:  5.80nMAssay Description:Affinity for cloned Y4 receptor using [125I]PP as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 2(Human)
University of Cincinnati and Va Medical Centers

Curated by ChEMBL
LigandPNGBDBM50034121(Ile-Asn-Pro-Ile-Tyr-Arg-Leu-Arg-Tyr-NH2 | CHEMBL38...)
Affinity DataKi:  11.3nMAssay Description:Affinity for cloned Y2 receptor using [125I]PYY as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 1(Human)
University of Cincinnati and Va Medical Centers

Curated by ChEMBL
LigandPNGBDBM50099203(Ile-Asn-Pro-Ile-Tyr-Arg-Leu-Arg-Tyr-OMe | CHEMBL43...)
Affinity DataKi:  25.7nMAssay Description:Affinity for cloned Y1 receptor using [125I]PYY as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 4(Human)
University of Cincinnati and Va Medical Centers

Curated by ChEMBL
LigandPNGBDBM50099197(Ile-Glu-Pro-Dpr-Tyr-Arg-Leu-Arg-Tyr-OMeIle-Glu-Pro...)
Affinity DataKi:  33.4nMAssay Description:Affinity for cloned Y4 receptor using [125I]PP as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 1(Human)
University of Cincinnati and Va Medical Centers

Curated by ChEMBL
LigandPNGBDBM50099202(Ile-Asn-Pro-Ile-Tyr-Arg-Leu-Arg-(CH2-NH)Tyr-NH2 | ...)
Affinity DataKi:  34.8nMAssay Description:Affinity for cloned Y1 receptor using [125I]PYY as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 2(Human)
University of Cincinnati and Va Medical Centers

Curated by ChEMBL
LigandPNGBDBM50409214(GR-231118 | CHEMBL2110365)
Affinity DataKi:  55nMAssay Description:Affinity for cloned Y2 receptor using [125I]PYY as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 4(Human)
University of Cincinnati and Va Medical Centers

Curated by ChEMBL
LigandPNGBDBM50099201(Ile-Asn-Pro-Cys-Tyr-Arg-Leu-Arg-(CH2-NH)-Tyr-NH2Il...)
Affinity DataKi:  65nMAssay Description:Affinity for cloned Y4 receptor using [125I]PP as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 4(Human)
University of Cincinnati and Va Medical Centers

Curated by ChEMBL
LigandPNGBDBM50099200(Ile-Glu-Pro-Dpr-Tyr-Arg-Leu-Arg-(CH2-NH)-Tyr-NH2Il...)
Affinity DataKi:  65.5nMAssay Description:Affinity for cloned Y4 receptor using [125I]PP as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 4(Human)
University of Cincinnati and Va Medical Centers

Curated by ChEMBL
LigandPNGBDBM50099199(Ile-Asn-Pro-Cys-Tyr-Arg-Leu-Arg-Tyr-OMeIle-Asn-Pro...)
Affinity DataKi:  99nMAssay Description:Affinity for cloned Y4 receptor using [125I]PP as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
University of Cincinnati and Va Medical Centers

Curated by ChEMBL
LigandPNGBDBM50409214(GR-231118 | CHEMBL2110365)
Affinity DataKi:  115nMAssay Description:Affinity for cloned Y5 receptor using [125I]PYY as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
University of Cincinnati and Va Medical Centers

Curated by ChEMBL
LigandPNGBDBM50099199(Ile-Asn-Pro-Cys-Tyr-Arg-Leu-Arg-Tyr-OMeIle-Asn-Pro...)
Affinity DataKi:  464nMAssay Description:Affinity for cloned Y5 receptor using [125I]PYY as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 2(Human)
University of Cincinnati and Va Medical Centers

Curated by ChEMBL
LigandPNGBDBM50099200(Ile-Glu-Pro-Dpr-Tyr-Arg-Leu-Arg-(CH2-NH)-Tyr-NH2Il...)
Affinity DataKi:  624nMAssay Description:Affinity for cloned Y2 receptor using [125I]PYY as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
University of Cincinnati and Va Medical Centers

Curated by ChEMBL
LigandPNGBDBM50099197(Ile-Glu-Pro-Dpr-Tyr-Arg-Leu-Arg-Tyr-OMeIle-Glu-Pro...)
Affinity DataKi:  662nMAssay Description:Affinity for cloned Y5 receptor using [125I]PYY as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 2(Human)
University of Cincinnati and Va Medical Centers

Curated by ChEMBL
LigandPNGBDBM50099201(Ile-Asn-Pro-Cys-Tyr-Arg-Leu-Arg-(CH2-NH)-Tyr-NH2Il...)
Affinity DataKi:  822nMAssay Description:Affinity for cloned Y2 receptor using [125I]PYY as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
University of Cincinnati and Va Medical Centers

Curated by ChEMBL
LigandPNGBDBM50034121(Ile-Asn-Pro-Ile-Tyr-Arg-Leu-Arg-Tyr-NH2 | CHEMBL38...)
Affinity DataKi: >1.00E+3nMAssay Description:Affinity for cloned Y5 receptor using [125I]PYY as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 2(Human)
University of Cincinnati and Va Medical Centers

Curated by ChEMBL
LigandPNGBDBM50099197(Ile-Glu-Pro-Dpr-Tyr-Arg-Leu-Arg-Tyr-OMeIle-Glu-Pro...)
Affinity DataKi:  1.04E+3nMAssay Description:Affinity for cloned Y2 receptor using [125I]PYY as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 2(Human)
University of Cincinnati and Va Medical Centers

Curated by ChEMBL
LigandPNGBDBM50099199(Ile-Asn-Pro-Cys-Tyr-Arg-Leu-Arg-Tyr-OMeIle-Asn-Pro...)
Affinity DataKi:  1.12E+3nMAssay Description:Affinity for cloned Y2 receptor using [125I]PYY as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 2(Human)
University of Cincinnati and Va Medical Centers

Curated by ChEMBL
LigandPNGBDBM50099203(Ile-Asn-Pro-Ile-Tyr-Arg-Leu-Arg-Tyr-OMe | CHEMBL43...)
Affinity DataKi:  1.42E+3nMAssay Description:Affinity for cloned Y2 receptor using [125I]PYY as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 2(Human)
University of Cincinnati and Va Medical Centers

Curated by ChEMBL
LigandPNGBDBM50099202(Ile-Asn-Pro-Ile-Tyr-Arg-Leu-Arg-(CH2-NH)Tyr-NH2 | ...)
Affinity DataKi:  1.65E+3nMAssay Description:Affinity for cloned Y2 receptor using [125I]PYY as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
University of Cincinnati and Va Medical Centers

Curated by ChEMBL
LigandPNGBDBM50099201(Ile-Asn-Pro-Cys-Tyr-Arg-Leu-Arg-(CH2-NH)-Tyr-NH2Il...)
Affinity DataKi:  2.34E+3nMAssay Description:Affinity for cloned Y5 receptor using [125I]PYY as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 4(Human)
University of Cincinnati and Va Medical Centers

Curated by ChEMBL
LigandPNGBDBM50099203(Ile-Asn-Pro-Ile-Tyr-Arg-Leu-Arg-Tyr-OMe | CHEMBL43...)
Affinity DataKi:  2.40E+3nMAssay Description:Affinity for cloned Y4 receptor using [125I]PP as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 4(Human)
University of Cincinnati and Va Medical Centers

Curated by ChEMBL
LigandPNGBDBM50099202(Ile-Asn-Pro-Ile-Tyr-Arg-Leu-Arg-(CH2-NH)Tyr-NH2 | ...)
Affinity DataKi:  3.74E+3nMAssay Description:Affinity for cloned Y4 receptor using [125I]PP as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
University of Cincinnati and Va Medical Centers

Curated by ChEMBL
LigandPNGBDBM50099202(Ile-Asn-Pro-Ile-Tyr-Arg-Leu-Arg-(CH2-NH)Tyr-NH2 | ...)
Affinity DataKi:  5.08E+3nMAssay Description:Affinity for cloned Y5 receptor using [125I]PYY as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
University of Cincinnati and Va Medical Centers

Curated by ChEMBL
LigandPNGBDBM50099203(Ile-Asn-Pro-Ile-Tyr-Arg-Leu-Arg-Tyr-OMe | CHEMBL43...)
Affinity DataKi:  7.10E+3nMAssay Description:Affinity for cloned Y5 receptor using [125I]PYY as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
University of Cincinnati and Va Medical Centers

Curated by ChEMBL
LigandPNGBDBM50099200(Ile-Glu-Pro-Dpr-Tyr-Arg-Leu-Arg-(CH2-NH)-Tyr-NH2Il...)
Affinity DataKi:  7.89E+3nMAssay Description:Affinity for cloned Y5 receptor using [125I]PYY as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed