Compile Data Set for Download or QSAR
Report error Found 9 Enz. Inhib. hit(s) with all data for entry = 50010814
TargetD(3) dopamine receptor(Human)
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50099011(1-Methyl-cyclohexanecarboxylic acid {(R)-2-[4-(4-m...)
Affinity DataIC50: 489nMAssay Description:Percent inhibition towards dopamine D3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50099011(1-Methyl-cyclohexanecarboxylic acid {(R)-2-[4-(4-m...)
Affinity DataIC50: 1.10E+3nMAssay Description:Percent inhibition towards dopamine D4 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50099011(1-Methyl-cyclohexanecarboxylic acid {(R)-2-[4-(4-m...)
Affinity DataIC50: 3.52E+3nMAssay Description:Percent inhibition towards dopamine D2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50099016(Cyclohexanecarboxylic acid {(S)-1-benzyl-2-[4-(4-c...)
Affinity DataKi:  0.800nMAssay Description:Ability to displace [3H]8-OH-DPAT from CHO cells stably transfected with human 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50099015(Cyclohexanecarboxylic acid {(R)-1-benzyl-2-[4-(4-m...)
Affinity DataKi:  1.5nMAssay Description:Ability to displace [3H]8-OH-DPAT from CHO cells stably transfected with human 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50099011(1-Methyl-cyclohexanecarboxylic acid {(R)-2-[4-(4-m...)
Affinity DataKi:  3nMAssay Description:Ability to displace [3H]8-OH-DPAT from CHO cells stably transfected with human 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50099014(Cyclohexanecarboxylic acid {(R)-1-benzyl-2-[4-(4-c...)
Affinity DataKi:  4.5nMAssay Description:Ability to displace [3H]8-OH-DPAT from CHO cells stably transfected with human 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50099013(N-{(R)-1-Benzyl-2-[4-(4-methoxy-[1,2,5]thiadiazol-...)
Affinity DataKi:  9.90nMAssay Description:Ability to displace [3H]8-OH-DPAT from CHO cells stably transfected with human 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50099012(N-{(S)-1-Benzyl-2-[4-(4-chloro-[1,2,5]thiadiazol-3...)
Affinity DataKi:  425nMAssay Description:Ability to displace [3H]8-OH-DPAT from CHO cells stably transfected with human 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed