Compile Data Set for Download or QSAR
Report error Found 12 Enz. Inhib. hit(s) with all data for entry = 50010773
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50098571(His-Ser-Gln-Gly-Thr-Phe-Thr-Ser-Asp-Tyr-Ser-Lys-Ty...)
Affinity DataIC50: 1.5nMAssay Description:inhibition of [125]glucagon specific binding.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50098563(Ser-Gln-Gly-Thr-Phe-Thr-Ser-Glu-Tyr-Ser-Lys-Tyr-Le...)
Affinity DataIC50: 3.75nMAssay Description:Compound was evaluated for its ability to displace radiolabeled glucagonMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50098573(N-trinitrophenyl-His-Ser-Gln-Gly-Thr-Phe-Thr-Ser-A...)
Affinity DataIC50: 15nMAssay Description:Compound was evaluated for its ability to displace radiolabeled glucagon (inactive up to 100 uM)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50098566(phenylbutyryl-Tyr-Ser-Lys-Tyr-Leu-Asp-Ser-Arg-Arg-...)
Affinity DataIC50: 21.2nMAssay Description:IC50 value was expressed as inhibition of [125]glucagon specific binding.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50098572(Ac-Phe-Thr-Ser-Asp-Tyr-Ser-Lys-Tyr-Leu-Asp-Ser-Arg...)
Affinity DataIC50: 31nMAssay Description:IC50 value was expressed as inhibition of [125]glucagon specific binding.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50098570(Ser-Gln-Gly-Thr-Thr-Ser-Glu-Tyr-Ser-Lys-Tyr-Leu-As...)
Affinity DataIC50: 48nMAssay Description:Compound was evaluated for its ability to displace radiolabeled glucagonMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50098565(Ac-Tyr-Ser-Lys-Tyr-Leu-Asp-Ser-Arg-Arg-Ala-Gln-Asp...)
Affinity DataIC50: 60nMAssay Description:IC50 value was expressed as inhibition of [125]glucagon specific binding.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50098567(phenylhexanoyl-Tyr-Ser-Lys-Tyr-Leu-Asp-Ser-Arg-Arg...)
Affinity DataIC50: 131nMAssay Description:IC50 value was expressed as inhibition of [125]glucagon specific binding.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50098564(Phenacetyl-Tyr-Ser-Lys-Tyr-Leu-Asp-Ser-Arg-Arg-Ala...)
Affinity DataIC50: 249nMAssay Description:IC50 value was expressed as inhibition of [125]glucagon specific binding.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50098574(phenylbutyryl-Tyr-Ser-Lys-2-Nal-Leu-Asp-Ser-Arg-Ar...)
Affinity DataIC50: 781nMAssay Description:IC50 value was expressed for inhibition of [125]glucagon specific binding.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50098569(Ac-Nal-Ser-Lys-Nal-Leu-Asp-Ser-Arg-Arg-Ala-Gln-Asp...)
Affinity DataIC50: 800nMAssay Description:IC50 value was expressed as inhibition of [125]glucagon specific binding.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50098568(Ac-Arg-Arg-Ala-Gln-Asp-Phe-Val-Gln-Trp-Leu-Met-Asn...)
Affinity DataIC50: 2.30E+3nMAssay Description:IC50 value was expressed as inhibition of [125]glucagon specific binding.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed